Properties of Bisphosphonates in the 13762 Rat Mammary Carcinoma Model of Tumor-Induced Bone Resorption
ALVAREZ, Enrique, WESTMORE, Michael, ZAMBRANO, Carmen, MA, Linda, SATO, Masahiko, MARTIN, T. John, TEICHER, Beverly A, GALBREATH, Elizabeth J, SELLS GALVIN, Rachelle J, CLAPP, Crystal L, CONSIDINE, Eileen L, SMITH, Shawn J, KEYES, Kristan, IVERSEN, Philip W, DELAFUENTE, Dawn M, SULAIMON, Shola
Published in Clinical cancer research (15.11.2003)
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Published in Clinical cancer research (15.11.2003)
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Discovery of LY2457546: a multi-targeted anti-angiogenic kinase inhibitor with a novel spectrum of activity and exquisite potency in the acute myelogenous leukemia-Flt-3-internal tandem duplication mutant human tumor xenograft model
Burkholder, Timothy P., Clayton, Joshua R., Rempala, Mark E., Henry, James R., Knobeloch, John M., Mendel, David, McLean, Johnathan A., Hao, Yan, Barda, David A., Considine, Eileen L., Uhlik, Mark T., Chen, Yuefeng, Ma, Liandong, Bloem, Laura J., Akunda, Jacqueline K., McCann, Denis J., Sanchez-Felix, Manuel, Clawson, David K., Lahn, Michael M., Starling, James J.
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Published in Investigational new drugs (01.06.2012)
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Acyl Sulfonamide Anti-Proliferatives: Benzene Substituent Structure−Activity Relationships for a Novel Class of Antitumor Agents
Lobb, Karen L, Hipskind, Philip A, Aikins, James A, Alvarez, Enrique, Cheung, Yiu-Yin, Considine, Eileen L, De Dios, Alfonso, Durst, Gregory L, Ferritto, Rafael, Grossman, Cora Sue, Giera, Deborah D, Hollister, Beth A, Huang, Zhongping, Iversen, Philip W, Law, Kevin L, Li, Tiechao, Lin, Ho-Shen, Lopez, Beatriz, Lopez, Jose E, Cabrejas, Luisa M. Martin, McCann, Denis J, Molero, Victoriano, Reilly, John E, Richett, Michael E, Shih, Chuan, Teicher, Beverly, Wikel, James H, White, Wesley T, Mader, Mary M
Published in Journal of medicinal chemistry (21.10.2004)
Published in Journal of medicinal chemistry (21.10.2004)
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Erratum to: Discovery of LY2457546: a multi-targeted anti-angiogenic kinase inhibitor with a novel spectrum of activity and exquisite potency in the acute myelogenous leukemia-Flt-3-internal tandem duplication mutant human tumor xenograft model
Burkholder, Timothy P., Clayton, Joshua R., Rempala, Mark E., Henry, James R., Knobeloch, John M., Mendel, David, McLean, Johnathan A., Hao, Yan, Barda, David A., Considine, Eileen L., Uhlik, Mark T., Chen, Yuefeng, Ma, Liandong, Bloem, Laura J., Akunda, Jacqueline K., McCann, Denis J., Sanchez-Felix, Manuel, Clawson, David K., Lahn, Michael M., Starling, James J.
Published in Investigational new drugs (01.06.2012)
Published in Investigational new drugs (01.06.2012)
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Synthesis of 1,7-annulated indoles and their applications in the studies of cyclin dependent kinase inhibitors
Zhu, Guoxin, Conner, Scott E., Zhou, Xun, Chan, Ho-Kit, Shih, Chuan, Engler, Thomas A., Al-awar, Rima S., Brooks, Harold B., Watkins, Scott A., Spencer, Charles D., Schultz, Richard M., Dempsey, Jack A., Considine, Eileen L., Patel, Bharvin R., Ogg, Catherine A., Vasudevan, Vasu, Lytle, Michelle L.
Published in Bioorganic & medicinal chemistry letters (21.06.2004)
Published in Bioorganic & medicinal chemistry letters (21.06.2004)
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Preparation of novel aza-1,7-annulated indoles and their conversion to potent indolocarbazole kinase inhibitors
Al-awar, Rima S, Ray, James E, Hecker, Kyle A, Joseph, Sajan, Huang, Jianping, Shih, Chuan, Brooks, Harold B, Spencer, Charles D, Watkins, Scott A, Schultz, Richard M, Considine, Eileen L, Faul, Margaret M, Sullivan, Kevin A, Kolis, Stanley P, Carr, Michael A, Zhang, Faming
Published in Bioorganic & medicinal chemistry letters (02.08.2004)
Published in Bioorganic & medicinal chemistry letters (02.08.2004)
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1,7-Annulated indolocarbazoles as cyclin-dependent kinase inhibitors
Al-awar, Rima S., Ray, James E., Hecker, Kyle A., Huang, Jianping, Waid, Philip P., Shih, Chuan, Brooks, Harold B., Spencer, Charles D., Watkins, Scott A., Patel, Bharvin R., Stamm, Nancy B., Ogg, Catherine A., Schultz, Richard M., Considine, Eileen L., Faul, Margaret M., Sullivan, Kevin A., Kolis, Stanley P., Grutsch, John L., Joseph, Sajan
Published in Bioorganic & medicinal chemistry letters (21.06.2004)
Published in Bioorganic & medicinal chemistry letters (21.06.2004)
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Five families with arginine519-cysteine mutation in COL2A1: Evidence for three distinct founders
Bleasel, Jane F., Holderbaum, Daniel, Brancolini, Valeria, Moskowitz, Roland W., Considine, Eileen L., Prockop, Darwin J., Devoto, Marcella, Williams, Charlene J.
Published in Human mutation (1998)
Published in Human mutation (1998)
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Evidence against either a premature stop codon or the absence of obese gene mRNA in human obesity
Considine, R V, Considine, E L, Williams, C J, Nyce, M R, Magosin, S A, Bauer, T L, Rosato, E L, Colberg, J, Caro, J F
Published in The Journal of clinical investigation (01.06.1995)
Published in The Journal of clinical investigation (01.06.1995)
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The hypothalamic leptin receptor in humans: identification of incidental sequence polymorphisms and absence of the db/db mouse and fa/fa rat mutations
CONSIDINE, R. V, CONSIDINE, E. L, WILLIAMS, C. J, HYDE, T. M, CARO, J. F
Published in Diabetes (New York, N.Y.) (01.07.1996)
Published in Diabetes (New York, N.Y.) (01.07.1996)
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Novel, potent and selective cyclin D1/CDK4 inhibitors: indolo[6,7- a]pyrrolo[3,4- c]carbazoles
Engler, Thomas A., Furness, Kelly, Malhotra, Sushant, Sanchez-Martinez, Concha, Shih, Chuan, Xie, Walter, Zhu, Guoxin, Zhou, Xun, Conner, Scott, Faul, Margaret M., Sullivan, Kevin A., Kolis, Stanley P., Brooks, Harold B., Patel, Bharvin, Schultz, Richard M., DeHahn, Tammy B., Kirmani, Kashif, Spencer, Charles D., Watkins, Scott A., Considine, Eileen L., Dempsey, Jack A., Ogg, Catherine A., Stamm, Nancy B., Anderson, Bryan D., Campbell, Robert M., Vasudevan, Vasu, Lytle, Michelle L.
Published in Bioorganic & medicinal chemistry letters (21.07.2003)
Published in Bioorganic & medicinal chemistry letters (21.07.2003)
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Mutation Screening and Identification of a Sequence Variation in the Human OB Gene Coding Region
Considine, Robert V., Considine, Eileen L., Williams, Charlene J., Nyce, Mark R., Zhang, Peili, Opentanova, Irina, Ohannesian, Joanna P., Kolaczynski, Jerzy W., Bauer, Thomas L., Moore, John H., Caro, Jose F.
Published in Biochemical and biophysical research communications (27.03.1996)
Published in Biochemical and biophysical research communications (27.03.1996)
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Spondyloepiphyseal dysplasia and precocious osteoarthritis in a family with an Arg75-->Cys mutation in the procollagen type II gene (COL2A1)
Williams, C J, Considine, E L, Knowlton, R G, Reginato, A, Neumann, G, Harrison, D, Buxton, P, Jimenez, S, Prockop, D J
Published in Human genetics (01.11.1993)
Published in Human genetics (01.11.1993)
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Detection of sequence variants in the gene for human type II procollagen (COL2A1) by direct sequencing of polymerase chain reaction-amplified genomic DNA
Williams, C J, Harrison, D A, Hopkinson, I, Baldwin, C T, Ahmad, N N, Ala-Kokko, L, Korn, R M, Buxton, P G, Dimascio, J, Considine, E L
Published in Human mutation (1992)
Published in Human mutation (1992)
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