Development of pyrimidone D1 dopamine receptor positive allosteric modulators
Luderman, Kathryn D., Jain, Prashi, Benjamin Free, R., Conroy, Jennie L., Aubé, Jeffrey, Sibley, David R., Frankowski, Kevin J.
Published in Bioorganic & medicinal chemistry letters (01.01.2021)
Published in Bioorganic & medicinal chemistry letters (01.01.2021)
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Identification of Positive Allosteric Modulators of the D 1 Dopamine Receptor That Act at Diverse Binding Sites
Luderman, Kathryn D, Conroy, Jennie L, Free, R Benjamin, Southall, Noel, Ferrer, Marc, Sanchez-Soto, Marta, Moritz, Amy E, Willette, Blair K A, Fyfe, Tim J, Jain, Prashi, Titus, Steve, Hazelwood, Lisa A, Aubé, Jeffrey, Lane, J Robert, Frankowski, Kevin J, Sibley, David R
Published in Molecular pharmacology (01.10.2018)
Published in Molecular pharmacology (01.10.2018)
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Modification of cocaine self-administration by buspirone (buspar®): potential involvement of D3 and D4 dopamine receptors
Bergman, Jack, Roof, Rebecca A., Furman, Cheryse A., Conroy, Jennie L., Mello, Nancy K., Sibley, David R., Skolnick, Phil
Published in The international journal of neuropsychopharmacology (01.03.2013)
Published in The international journal of neuropsychopharmacology (01.03.2013)
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Journal Article
Discovery and characterization of a G protein-biased agonist that inhibits β-arrestin recruitment to the D2 dopamine receptor
Free, R Benjamin, Chun, Lani S, Moritz, Amy E, Miller, Brittney N, Doyle, Trevor B, Conroy, Jennie L, Padron, Adrian, Meade, Julie A, Xiao, Jingbo, Hu, Xin, Dulcey, Andrés E, Han, Yang, Duan, Lihua, Titus, Steve, Bryant-Genevier, Melanie, Barnaeva, Elena, Ferrer, Marc, Javitch, Jonathan A, Beuming, Thijs, Shi, Lei, Southall, Noel T, Marugan, Juan J, Sibley, David R
Published in Molecular pharmacology (01.07.2014)
Published in Molecular pharmacology (01.07.2014)
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(-)-Stepholidine is a potent pan-dopamine receptor antagonist of both G protein- and β-arrestin-mediated signaling
Meade, Julie A., Free, R. Benjamin, Miller, Nicole R., Chun, Lani S., Doyle, Trevor B., Moritz, Amy E., Conroy, Jennie L., Watts, Val J., Sibley, David R.
Published in Psychopharmacology (01.03.2015)
Published in Psychopharmacology (01.03.2015)
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Journal Article
Discovery, Optimization, and Characterization of Novel D2 Dopamine Receptor Selective Antagonists
Xiao, Jingbo, Free, R. Benjamin, Barnaeva, Elena, Conroy, Jennie L, Doyle, Trevor, Miller, Brittney, Bryant-Genevier, Marthe, Taylor, Mercedes K, Hu, Xin, Dulcey, Andrés E, Southall, Noel, Ferrer, Marc, Titus, Steve, Zheng, Wei, Sibley, David R, Marugan, Juan J
Published in Journal of medicinal chemistry (24.04.2014)
Published in Journal of medicinal chemistry (24.04.2014)
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Journal Article
Identification of Positive Allosteric Modulators of the D1 Dopamine Receptor That Act at Diverse Binding Sites
Luderman, Kathryn D, Conroy, Jennie L, Free, R Benjamin, Southall, Noel, Ferrer, Marc, Sanchez-Soto, Marta, Moritz, Amy E, Willette, Blair K A, Fyfe, Tim J, Jain, Prashi, Titus, Steve, Hazelwood, Lisa A, Aubé, Jeffrey, Lane, J Robert, Frankowski, Kevin J, Sibley, David R
Published in Molecular pharmacology (01.10.2018)
Published in Molecular pharmacology (01.10.2018)
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Journal Article
PNA-Based Multivalent Scaffolds Activate the Dopamine D2 Receptor
Dix, Andrew V, Conroy, Jennie L, George Rosenker, Kara M, Sibley, David R, Appella, Daniel H
Published in ACS medicinal chemistry letters (09.04.2015)
Published in ACS medicinal chemistry letters (09.04.2015)
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Journal Article
Brain P450 epoxygenase activity is required for the antinociceptive effects of improgan, a nonopioid analgesic
Hough, Lindsay B., Nalwalk, Julia W., Yang, Jun, Conroy, Jennie L., VanAlstine, Melissa A., Yang, Weizhu, Gargano, Joseph, Shan, Zhixing, Zhang, Shao-Zhong, Wentland, Mark P., Phillips, James G., Knapp, Brian I., Bidlack, Jean M., Zuiderveld, Obbe P., Leurs, Rob, Ding, Xinxin
Published in Pain (Amsterdam) (01.04.2011)
Published in Pain (Amsterdam) (01.04.2011)
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Report of the National Cancer Institute and the Eunice Kennedy Shriver National Institute of Child Health and Human Development–sponsored workshop: gynecology and women’s health–benign conditions and cancer
Samimi, Goli, Sathyamoorthy, Neeraja, Tingen, Candace M., Mazloomdoost, Donna, Conroy, Jennie, Heckman-Stoddard, Brandy, Halvorson, Lisa M.
Published in American journal of obstetrics and gynecology (01.12.2020)
Published in American journal of obstetrics and gynecology (01.12.2020)
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Conference Proceeding
Early detection and intervention evaluation for people at risk of psychosis: multisite randomised controlled trial
Morrison, Anthony P, French, Paul, Stewart, Suzanne L K, Birchwood, Max, Fowler, David, Gumley, Andrew I, Jones, Peter B, Bentall, Richard P, Lewis, Shôn W, Murray, Graham K, Patterson, Paul, Brunet, Kat, Conroy, Jennie, Parker, Sophie, Reilly, Tony, Byrne, Rory, Davies, Linda M, Dunn, Graham
Published in BMJ (Online) (05.04.2012)
Published in BMJ (Online) (05.04.2012)
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Journal Article
Discovery, Optimization, and Characterization of Novel D-2 Dopamine Receptor Selective Antagonists
Xiao, Jingbo, Free, R. Benjamin, Barnaeva, Elena, Conroy, Jennie L., Doyle, Trevor, Miller, Brittney, Bryant-Genevier, Marthe, Taylor, Mercedes K., Hu, Xin, Dulcey, Andres E., Southall, Noel, Ferrer, Marc, Titus, Steve, Zheng, Wei, Sibley, David R., Marugan, Juan J.
Published in Journal of medicinal chemistry (24.04.2014)
Published in Journal of medicinal chemistry (24.04.2014)
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Journal Article
PNA-Based Multivalent Scaffolds Activate the Dopamine D 2 Receptor
Dix, Andrew V., Conroy, Jennie L., George Rosenker, Kara M., Sibley, David R., Appella, Daniel H.
Published in ACS medicinal chemistry letters (09.04.2015)
Published in ACS medicinal chemistry letters (09.04.2015)
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Journal Article
Stepholidine is a potent pan-dopamine receptor antagonist of both G protein- and [beta]-arrestin-mediated signaling
Meade, Julie A, Free, R. Benjamin, Miller, Nicole R, Chun, Lani S, Doyle, Trevor B, Moritz, Amy E, Conroy, Jennie L, Watts, Val J, Sibley, David R
Published in Psychopharmacology (01.03.2015)
Published in Psychopharmacology (01.03.2015)
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Journal Article
Modification of cocaine self-administration by buspirone (buspar registered ): potential involvement of D sub(3) and D sub(4) dopamine receptors
Bergman, Jack, Roof, Rebecca A, Furman, Cheryse A, Conroy, Jennie L, Mello, Nancy K, Sibley, David R, Skolnick, Phil
Published in The international journal of neuropsychopharmacology (01.03.2013)
Published in The international journal of neuropsychopharmacology (01.03.2013)
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Journal Article
EARLY DETECTION AND INTERVENTION EVALUATION FOR PEOPLE AT-RISK OF PSYCHOSIS
Morrison, Anthony P, French, Paul, Stewart, Suzanne L.K, Birchwood, Max, Fowler, David, Gumley, Andrew I, Jones, Peter B, Bentall, Richard P, Lewis, Shôn W, Murray, Graham K, Patterson, Paul, Brunet, Kat, Conroy, Jennie, Parker, Sophie, Reilly, Tony, Byrne, Rory, Davies, Linda M, Dunn, Graham
Published in Schizophrenia research (01.04.2012)
Published in Schizophrenia research (01.04.2012)
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Journal Article
Brain P450 Epoxygenase Activity is Required for the Antinociceptive Effects of Improgan, a Non-Opioid Analgesic
Hough, Lindsay B., Nalwalk, Julia W., Yang, Jun, Conroy, Jennie L., VanAlstine, Melissa A., Yang, Weizhu, Gargano, Joseph, Shan, Zhixing, Zhang, Shao-Zhong, Wentland, Mark P, Phillips, James G., Knapp, Brian I., Bidlack, Jean M., Zuiderveld, Obbe P., Leurs, Rob, Ding, Xinxin
Published in Pain (Amsterdam) (01.04.2011)
Published in Pain (Amsterdam) (01.04.2011)
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Journal Article