Discovery of an Orally Bioavailable Inhibitor of Defective in Cullin Neddylation 1 (DCN1)-Mediated Cullin Neddylation
Hammill, Jared T, Bhasin, Deepak, Scott, Daniel C, Min, Jaeki, Chen, Yizhe, Lu, Yan, Yang, Lei, Kim, Ho Shin, Connelly, Michele C, Hammill, Courtney, Holbrook, Gloria, Jeffries, Cynthia, Singh, Bhuvanesh, Schulman, Brenda A, Guy, R. Kiplin
Published in Journal of medicinal chemistry (12.04.2018)
Published in Journal of medicinal chemistry (12.04.2018)
Get full text
Journal Article
Screening and Development of New Inhibitors of FtsZ from M. Tuberculosis
Mathew, Bini, Hobrath, Judith Varady, Ross, Larry, Connelly, Michele C, Lofton, Hava, Rajagopalan, Malini, Guy, R Kiplin, Reynolds, Robert C
Published in PloS one (21.10.2016)
Published in PloS one (21.10.2016)
Get full text
Journal Article
Potent Plasmodium falciparum gametocytocidal activity of diaminonaphthoquinones, lead antimalarial chemotypes identified in an antimalarial compound screen
Tanaka, Takeshi Q, Guiguemde, W Armand, Barnett, David S, Maron, Maxim I, Min, Jaeki, Connelly, Michele C, Suryadevara, Praveen Kumar, Guy, R Kiplin, Williamson, Kim C
Published in Antimicrobial agents and chemotherapy (01.03.2015)
Published in Antimicrobial agents and chemotherapy (01.03.2015)
Get full text
Journal Article
Dihydroquinazolinone Inhibitors of Proliferation of Blood and Liver Stage Malaria Parasites
DERBYSHIRE, Emily R, JAEKI MIN, GUIGUEMDE, W. Armand, CLARK, Julie A, CONNELLY, Michele C, MAGALHAES, Andreia D, GUY, R. Kiplin, CLARDY, Jon
Published in Antimicrobial Agents and Chemotherapy (01.03.2014)
Published in Antimicrobial Agents and Chemotherapy (01.03.2014)
Get full text
Journal Article
MRP4: A previously unidentified factor in resistance to nucleoside-based antiviral drugs
Schuetz, John D, Connelly, Michele C, Sun, Daxi, Paibir, Sheela G, Flynn, Patricia M, Srinivas, R.V, Kumar, Alok, Fridland, Arnold
Published in Nature medicine (01.09.1999)
Published in Nature medicine (01.09.1999)
Get full text
Journal Article
Amide conjugates of ketoprofen and indole as inhibitors of Gli1-mediated transcription in the Hedgehog pathway
Mahindroo, Neeraj, Connelly, Michele C., Punchihewa, Chandanamali, Yang, Lei, Yan, Bing, Fujii, Naoaki
Published in Bioorganic & medicinal chemistry (01.07.2010)
Published in Bioorganic & medicinal chemistry (01.07.2010)
Get full text
Journal Article
Discovery of a Diaminopyrimidine FLT3 Inhibitor Active against Acute Myeloid Leukemia
Jarusiewicz, Jamie A, Jeon, Jae Yoon, Connelly, Michele C, Chen, Yizhe, Yang, Lei, Baker, Sharyn D, Guy, R. Kiplin
Published in ACS omega (31.05.2017)
Published in ACS omega (31.05.2017)
Get full text
Journal Article
Antitrypanosomal Chloronitrobenzamides
Carrillo, Angela K., Kadayat, Tara Man, Hwang, Jong Yeon, Chen, Yizhe, Zhu, Fangyi, Holbrook, Gloria, Gillingwater, Kirsten, Connelly, Michele C., Yang, Lei, Kaiser, Marcel, Guy, R. Kiplin
Published in Journal of medicinal chemistry (14.03.2024)
Published in Journal of medicinal chemistry (14.03.2024)
Get full text
Journal Article
Piperidinyl Ureas Chemically Control Defective in Cullin Neddylation 1 (DCN1)-Mediated Cullin Neddylation
Hammill, Jared T, Scott, Daniel C, Min, Jaeki, Connelly, Michele C, Holbrook, Gloria, Zhu, Fangyi, Matheny, Amy, Yang, Lei, Singh, Bhuvanesh, Schulman, Brenda A, Guy, R. Kiplin
Published in Journal of medicinal chemistry (12.04.2018)
Published in Journal of medicinal chemistry (12.04.2018)
Get full text
Journal Article
Discovery of Novel Antimalarial Compounds Enabled by QSAR-Based Virtual Screening
Zhang, Liying, Fourches, Denis, Sedykh, Alexander, Zhu, Hao, Golbraikh, Alexander, Ekins, Sean, Clark, Julie, Connelly, Michele C, Sigal, Martina, Hodges, Dena, Guiguemde, Armand, Guy, R. Kiplin, Tropsha, Alexander
Published in Journal of chemical information and modeling (25.02.2013)
Published in Journal of chemical information and modeling (25.02.2013)
Get full text
Journal Article
Diverse amide analogs of sulindac for cancer treatment and prevention
Mathew, Bini, Hobrath, Judith V., Connelly, Michele C., Kiplin Guy, R., Reynolds, Robert C.
Published in Bioorganic & medicinal chemistry letters (15.10.2017)
Published in Bioorganic & medicinal chemistry letters (15.10.2017)
Get full text
Journal Article
Optimization of a Novel Series of Ataxia-Telangiectasia Mutated Kinase Inhibitors as Potential Radiosensitizing Agents
Min, Jaeki, Guo, Kexiao, Suryadevara, Praveen K, Zhu, Fangyi, Holbrook, Gloria, Chen, Yizhe, Feau, Clementine, Young, Brandon M, Lemoff, Andrew, Connelly, Michele C, Kastan, Michael B, Guy, R. Kiplin
Published in Journal of medicinal chemistry (28.01.2016)
Published in Journal of medicinal chemistry (28.01.2016)
Get full text
Journal Article
Lead Optimization of 3-Carboxyl-4(1H)-Quinolones to Deliver Orally Bioavailable Antimalarials
Zhang, Yiqun, Clark, Julie A, Connelly, Michele C, Zhu, Fangyi, Min, Jaeki, Guiguemde, W. Armand, Pradhan, Anupam, Iyer, Lalitha, Furimsky, Anna, Gow, Jason, Parman, Toufan, El Mazouni, Farah, Phillips, Margaret A, Kyle, Dennis E, Mirsalis, Jon, Guy, R. Kiplin
Published in Journal of medicinal chemistry (10.05.2012)
Published in Journal of medicinal chemistry (10.05.2012)
Get full text
Journal Article
Oxazole and thiazole analogs of sulindac for cancer prevention
Mathew, Bini, Hobrath, Judith V, Connelly, Michele C, Guy, R Kiplin, Reynolds, Robert C
Published in Future medicinal chemistry (01.04.2018)
Published in Future medicinal chemistry (01.04.2018)
Get full text
Journal Article
Synthesis and Evaluation of 7-Substituted 4-Aminoquinoline Analogues for Antimalarial Activity
Hwang, Jong Yeon, Kawasuji, Takashi, Lowes, David J, Clark, Julie A, Connelly, Michele C, Zhu, Fangyi, Guiguemde, W. Armand, Sigal, Martina S, Wilson, Emily B, DeRisi, Joseph L, Guy, R. Kiplin
Published in Journal of medicinal chemistry (27.10.2011)
Published in Journal of medicinal chemistry (27.10.2011)
Get full text
Journal Article
Optimization of Chloronitrobenzamides (CNBs) as Therapeutic Leads for Human African Trypanosomiasis (HAT)
Hwang, Jong Yeon, Smithson, David, Zhu, Fangyi, Holbrook, Gloria, Connelly, Michele C, Kaiser, Marcel, Brun, Reto, Guy, R. Kiplin
Published in Journal of medicinal chemistry (11.04.2013)
Published in Journal of medicinal chemistry (11.04.2013)
Get full text
Journal Article
Synthesis and Evaluation of Sulfonylnitrophenylthiazoles (SNPTs) as Thyroid Hormone Receptor–Coactivator Interaction Inhibitors
Hwang, Jong Yeon, Attia, Ramy R, Zhu, Fangyi, Yang, Lei, Lemoff, Andrew, Jeffries, Cynthia, Connelly, Michele C, Guy, R. Kiplin
Published in Journal of medicinal chemistry (08.03.2012)
Published in Journal of medicinal chemistry (08.03.2012)
Get full text
Journal Article
Optimization of Propafenone Analogues as Antimalarial Leads
Lowes, David J, Guiguemde, W. Armand, Connelly, Michele C, Zhu, Fangyi, Sigal, Martina S, Clark, Julie A, Lemoff, Andrew S, Derisi, Joseph L, Wilson, Emily B, Guy, R. Kiplin
Published in Journal of medicinal chemistry (10.11.2011)
Published in Journal of medicinal chemistry (10.11.2011)
Get full text
Journal Article
Optimization of the electrophile of chloronitrobenzamide leads active against Trypanosoma brucei
Hwang, Jong Yeon, Smithson, David C., Holbrook, Gloria, Zhu, Fangyi, Connelly, Michele C., Kaiser, Marcel, Brun, Reto, Kiplin Guy, R.
Published in Bioorganic & medicinal chemistry letters (15.07.2013)
Published in Bioorganic & medicinal chemistry letters (15.07.2013)
Get full text
Journal Article