Cytotoxicity of Pyrazine-Based Cyclometalated (C^Npz^C)Au(III) Carbene Complexes: Impact of the Nature of the Ancillary Ligand on the Biological Properties
Bertrand, Benoît, Fernandez-Cestau, Julio, Angulo, Jesus, Cominetti, Marco M. D, Waller, Zoë A. E, Searcey, Mark, O’Connell, Maria A, Bochmann, Manfred
Published in Inorganic chemistry (15.05.2017)
Published in Inorganic chemistry (15.05.2017)
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Journal Article
A Peptide–Duocarmycin Conjugate Targeting the Thomsen-Friedenreich Antigen Has Potent and Selective Antitumor Activity
Cartwright, Oliver Charles, Beekman, Andrew Michael, Cominetti, Marco M. D, Russell, David A, Searcey, Mark
Published in Bioconjugate chemistry (15.07.2020)
Published in Bioconjugate chemistry (15.07.2020)
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Journal Article
Peptide directed phthalocyanine-gold nanoparticles for selective photodynamic therapy of EGFR overexpressing cancers
Goddard, Zoë Rachael, Beekman, Andrew Michael, Cominetti, Marco M. D, O'Connell, Maria A, Chambrier, Isabelle, Cook, Michael J, Marín, María J, Russell, David A, Searcey, Mark
Published in MedChemComm (19.11.2020)
Published in MedChemComm (19.11.2020)
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Journal Article
Open-resorcinarenes, a new family of multivalent scaffolds
Cominetti, Marco M. D., Hughes, David L., Matthews, Susan E.
Published in Organic & biomolecular chemistry (02.11.2016)
Published in Organic & biomolecular chemistry (02.11.2016)
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Journal Article
Junctions in DNA: underexplored targets for therapeutic intervention
Ivens, Eleanor, Cominetti, Marco M.D., Searcey, Mark
Published in Bioorganic & medicinal chemistry (01.09.2022)
Published in Bioorganic & medicinal chemistry (01.09.2022)
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Journal Article
The development of potent, competitive CXCR4 antagonists for the prevention of cancer metastasis
Hamshaw, Isabel, Cominetti, Marco M D, Lai, Wing-Yee, Searcey, Mark, Mueller, Anja
Published in Biochemical pharmacology (01.12.2023)
Published in Biochemical pharmacology (01.12.2023)
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Journal Article
Identification of selective protein-protein interaction inhibitors using efficient in silico peptide-directed ligand design
Beekman, Andrew M., Cominetti, Marco M. D., Walpole, Samuel J., Prabhu, Saurabh, O'Connell, Maria A., Angulo, Jesus, Searcey, Mark
Published in Chemical science (Cambridge) (28.04.2019)
Published in Chemical science (Cambridge) (28.04.2019)
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Journal Article
IS4 ‐ FAM , a fluorescent tool to study CXCR4 affinity and competitive antagonism in native cancer cells
Hamshaw, Isabel, Cominetti, Marco M. D., Nana‐Akyin, Princess, Yee Ho, Ernie Ho, Searcey, Mark, Mueller, Anja
Published in Pharmacology research & perspectives (01.10.2024)
Published in Pharmacology research & perspectives (01.10.2024)
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Journal Article
Correction: Identification of selective protein–protein interaction inhibitors using efficient in silico peptide-directed ligand design
Beekman, Andrew M., Cominetti, Marco M. D., Walpole, Samuel J., Prabhu, Saurabh, O’Connell, Maria A., Angulo, Jesus, Searcey, Mark
Published in Chemical science (Cambridge) (05.06.2019)
Published in Chemical science (Cambridge) (05.06.2019)
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Journal Article
Identification of a new p53/MDM2 inhibitor motif inspired by studies of chlorofusin
Cominetti, Marco M.D., Goffin, Sarah A., Raffel, Ewan, Turner, Kerrie D., Ramoutar, Jordann C., O’Connell, Maria A., Howell, Lesley A., Searcey, Mark
Published in Bioorganic & medicinal chemistry letters (01.11.2015)
Published in Bioorganic & medicinal chemistry letters (01.11.2015)
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Journal Article
Open-resorcinarenes, a new family of multivalent scaffoldsElectronic supplementary information (ESI) available: Methods, characterization data and crystallographic data. CCDC 1497840-1497843. For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c6ob02164f
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Journal Article
Identification of selective protein-protein interaction inhibitors using efficient in silico peptide-directed ligand designElectronic supplementary information (ESI) available: Experimental procedures, spectra and processed biophysical assay data. See DOI: 10.1039/c9sc00059c
Beekman, Andrew M, Cominetti, Marco M. D, Walpole, Samuel J, Prabhu, Saurabh, O'Connell, Maria A, Angulo, Jesus, Searcey, Mark
Year of Publication 17.04.2019
Year of Publication 17.04.2019
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Journal Article
Identification of selective protein–protein interaction inhibitors using efficient in silico peptide-directed ligand design† †Electronic supplementary information (ESI) available: Experimental procedures, spectra and processed biophysical assay data. See DOI: 10.1039/c9sc00059c
Beekman, Andrew M., Cominetti, Marco M. D., Walpole, Samuel J., Prabhu, Saurabh, O'Connell, Maria A., Angulo, Jesus, Searcey, Mark
Published in Chemical science (Cambridge) (22.03.2019)
Published in Chemical science (Cambridge) (22.03.2019)
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Journal Article
A small molecule drug conjugate (SMDC) of DUPA and a duocarmycin built on the solid phase† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c9md00279k
Beekman, Andrew Michael, Cominetti, Marco M. D., Cartwright, Oliver Charles, Boger, Dale L., Searcey, Mark
Published in MedChemComm (27.11.2019)
Published in MedChemComm (27.11.2019)
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Journal Article
Base-modified NAD and AMP derivatives and their activity against bacterial DNA ligasesElectronic supplementary information (ESI) available. See DOI: 10.1039/c5ob00294j
Pergolizzi, Giulia, Cominetti, Marco M. D, Butt, Julea N, Field, Robert A, Bowater, Richard P, Wagner, Gerd K
Year of Publication 27.05.2015
Year of Publication 27.05.2015
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Journal Article