Rogaratinib: A potent and selective pan‐FGFR inhibitor with broad antitumor activity in FGFR‐overexpressing preclinical cancer models
Grünewald, Sylvia, Politz, Oliver, Bender, Sebastian, Héroult, Mélanie, Lustig, Klemens, Thuss, Uwe, Kneip, Christoph, Kopitz, Charlotte, Zopf, Dieter, Collin, Marie‐Pierre, Boemer, Ulf, Ince, Stuart, Ellinghaus, Peter, Mumberg, Dominik, Hess‐Stumpp, Holger, Ziegelbauer, Karl
Published in International journal of cancer (01.09.2019)
Published in International journal of cancer (01.09.2019)
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Discovery of Rogaratinib (BAY 1163877): a pan‐FGFR Inhibitor
Collin, Marie‐Pierre, Lobell, Mario, Hübsch, Walter, Brohm, Dirk, Schirok, Hartmut, Jautelat, Rolf, Lustig, Klemens, Bömer, Ulf, Vöhringer, Verena, Héroult, Mélanie, Grünewald, Sylvia, Hess‐Stumpp, Holger
Published in ChemMedChem (06.03.2018)
Published in ChemMedChem (06.03.2018)
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Total Synthesis of Spirastrellolide F Methyl Ester--Part 1: Strategic Considerations and Revised Approach to the Southern Hemisphere
O'Neil, Gregory W, Ceccon, Julien, Benson, Stefan, Collin, Marie-Pierre, Fasching, Bernhard, Fürstner, Alois
Published in Angewandte Chemie (International ed.) (21.12.2009)
Published in Angewandte Chemie (International ed.) (21.12.2009)
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Total Synthesis of Spirastrellolide F Methyl Ester--Part 2: Macrocyclization and Completion of the Synthesis
Benson, Stefan, Collin, Marie-Pierre, O'Neil, Gregory W, Ceccon, Julien, Fasching, Bernhard, Fenster, Michaël D.B, Godbout, Cédrickx, Radkowski, Karin, Goddard, Richard, Fürstner, Alois
Published in Angewandte Chemie (International ed.) (21.12.2009)
Published in Angewandte Chemie (International ed.) (21.12.2009)
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Journal Article
Synthesis of 1,2,3-Triazole Analogues of Lincomycin
Collin, Marie-Pierre, Hobbie, Sven N., Böttger, Erik C., Vasella, Andrea
Published in Helvetica chimica acta (01.10.2008)
Published in Helvetica chimica acta (01.10.2008)
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Synthesis and Evaluation of S- and C(1)-Substituted Analogues of Lincomycin
Collin, Marie-Pierre, Hobbie, Sven N., Böttger, Erik C., Vasella, Andrea
Published in Helvetica chimica acta (01.02.2009)
Published in Helvetica chimica acta (01.02.2009)
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Structure–Permeability Relationship of Semipeptidic MacrocyclesUnderstanding and Optimizing Passive Permeability and Efflux Ratio
Le Roux, Antoine, Blaise, Émilie, Boudreault, Pierre-Luc, Comeau, Christian, Doucet, Annie, Giarrusso, Marilena, Collin, Marie-Pierre, Neubauer, Thomas, Kölling, Florian, Göller, Andreas H, Seep, Lea, Tshitenge, Dieudonné T, Wittwer, Matthias, Kullmann, Maximilian, Hillisch, Alexander, Mittendorf, Joachim, Marsault, Eric
Published in Journal of medicinal chemistry (09.07.2020)
Published in Journal of medicinal chemistry (09.07.2020)
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Abstract 4332: Discovery of BAY 1163877 - A pan-FGFR inhibitor: De novo structure-based design and lead optimization of benzothiophenyl-pyrrolotriazines
Collin, Marie-Pierre L., Lobell, Mario, Huebsch, Walter, Brohm, Dirk, Héroult, Mélanie, Lustig, Klemens, Gruenewald, Sylvia, Boemer, Ulf, Jautelat, Rolf, Hess-Stump, Holger, Jaroch, Stefan, Brands, Michael, Ziegelbauer, Karl
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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Second-Generation Total Synthesis of Spirastrellolide F Methyl Ester: The Alkyne Route
Benson, Stefan, Collin, Marie-Pierre, Arlt, Alexander, Gabor, Barbara, Goddard, Richard, Fürstner, Alois
Published in Angewandte Chemie (05.09.2011)
Published in Angewandte Chemie (05.09.2011)
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Journal Article
Total Synthesis of Spirastrellolide F Methyl Ester-Part 1: Strategic Considerations and Revised Approach to the Southern Hemisphere
O'Neil, Gregory W., Ceccon, Julien, Benson, Stefan, Collin, Marie-Pierre, Fasching, Bernhard, Fürstner, Alois
Published in Angewandte Chemie (21.12.2009)
Published in Angewandte Chemie (21.12.2009)
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Journal Article
Total Synthesis of Spirastrellolide F Methyl Ester-Part 2: Macrocyclization and Completion of the Synthesis
Benson, Stefan, Collin, Marie-Pierre, O'Neil, Gregory W., Ceccon, Julien, Fasching, Bernhard, Fenster, Michaël D. B., Godbout, Cédrickx, Radkowski, Karin, Goddard, Richard, Fürstner, Alois
Published in Angewandte Chemie (21.12.2009)
Published in Angewandte Chemie (21.12.2009)
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Journal Article
The Novel Potent and Selective Vasopressin V1a Antagonist BAY2327949 Blocks Arginine Vasopressin-Mediated Decline of Renal Blood Flow and Tissue Oxygenation: PO0647
Cernecka, Hana, Droebner, Karoline, Tinel, Hanna, Pook, Eisabeth, Fuerstner, Chantal, Collin, Marie-Pierre L., Hein, Peter, Eitner, Frank, Kolkhof, Peter
Published in Journal of the American Society of Nephrology (01.10.2020)
Published in Journal of the American Society of Nephrology (01.10.2020)
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Kidney Functional Improvements by a Novel Potent and Selective Vasopressin V1a Antagonist After Ischemia/Reperfusion Injury (I/RI) in Rats: PO0164
Droebner, Karoline, Cernecka, Hana, Fuerstner, Chantal, Collin, Marie-Pierre L., Pavkovic, Mira, Hein, Peter, Eitner, Frank, Kolkhof, Peter
Published in Journal of the American Society of Nephrology (01.10.2020)
Published in Journal of the American Society of Nephrology (01.10.2020)
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Abstract 1079: Preclinical activity of the FGFRinhibitor BAY 1163877 alone or in combination with antihormonal therapy in breast cancer
Politz, Oliver, Ellinghaus, Peter, Bender, Sebastian, Gruenewald, Sylvia, Siegel, Franziska, Collin, Marie-Pierre, Zitzmann-Kolbe, Sabine, Mumberg, Dominik, Ziegelbauer, Karl
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Published in Cancer research (Chicago, Ill.) (01.07.2017)
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Abstract 1739: Preclinical profile of BAY 1163877 - a selective pan-FGFR inhibitor in phase 1 clinical trial
Heroult, Melanie, Ellinghaus, Peter, Sieg, Christian, Brohm, Dirk, Gruenewald, Sylvia, Collin, Marie-Pierre, Boemer, Ulf, Lobell, Mario, Huebsch, Walter, Ocker, Matthias, Ince, Stuart, Haegebarth, Andrea, Jautelat, Rolf, Hess-Stumpp, Holger, Brands, Michael, Ziegelbauer, Karl
Published in Cancer research (Chicago, Ill.) (01.10.2014)
Published in Cancer research (Chicago, Ill.) (01.10.2014)
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