Tool inhibitors and assays to interrogate the biology of the TRAF2 and NCK interacting kinase
Read, Jon, Collie, Iain T., Nguyen-McCarty, Michelle, Lucaj, Christopher, Robinson, James, Conway, Leslie, Mukherjee, Jayanta, McCall, Eileen, Donohoe, Gerard, Flavell, Elizabeth, Peciak, Karolina, Warwicker, Juli, Dix, Carly, Van den Hoven, Bernard G., Madin, Andrew, Brown, Dean G., Moss, Stephen, Haggarty, Stephen J., Brandon, Nicholas J., Bürli, Roland W.
Published in Bioorganic & medicinal chemistry letters (01.08.2019)
Published in Bioorganic & medicinal chemistry letters (01.08.2019)
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One Scaffold, Three Binding Modes: Novel and Selective Pteridine Reductase 1 Inhibitors Derived from Fragment Hits Discovered by Virtual Screening
Mpamhanga, Chidochangu P, Spinks, Daniel, Tulloch, Lindsay B, Shanks, Emma J, Robinson, David A, Collie, Iain T, Fairlamb, Alan H, Wyatt, Paul G, Frearson, Julie A, Hunter, William N, Gilbert, Ian H, Brenk, Ruth
Published in Journal of medicinal chemistry (23.07.2009)
Published in Journal of medicinal chemistry (23.07.2009)
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Development of a Series of Pyrrolopyridone MAT2A Inhibitors
Atkinson, Stephen J., Bagal, Sharan K., Argyrou, Argyrides, Askin, Sean, Cheung, Tony, Chiarparin, Elisabetta, Coen, Muireann, Collie, Iain T., Dale, Ian L., De Fusco, Claudia, Dillman, Keith, Evans, Laura, Feron, Lyman J., Foster, Alison J., Grondine, Michael, Kantae, Vasudev, Lamont, Gillian M., Lamont, Scott, Lynch, James T., Nilsson Lill, Sten, Robb, Graeme R., Saeh, Jamal, Schimpl, Marianne, Scott, James S., Smith, James, Srinivasan, Bharath, Tentarelli, Sharon, Vazquez-Chantada, Mercedes, Wagner, David, Walsh, Jarrod J., Watson, David, Williamson, Beth
Published in Journal of medicinal chemistry (28.03.2024)
Published in Journal of medicinal chemistry (28.03.2024)
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Development of a 2,4-Diaminothiazole Series for the Treatment of Human African Trypanosomiasis Highlights the Importance of Static–Cidal Screening of Analogues
Cleghorn, Laura A. T., Wall, Richard J., Albrecht, Sébastien, MacGowan, Stuart A., Norval, Suzanne, De Rycker, Manu, Woodland, Andrew, Spinks, Daniel, Thompson, Stephen, Patterson, Stephen, Corpas Lopez, Victoriano, Dey, Gourav, Collie, Iain T., Hallyburton, Irene, Kime, Robert, Simeons, Frederick R. C., Stojanovski, Laste, Frearson, Julie A., Wyatt, Paul G., Read, Kevin D., Gilbert, Ian H., Wyllie, Susan
Published in Journal of medicinal chemistry (13.07.2023)
Published in Journal of medicinal chemistry (13.07.2023)
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The First Potent and Selective Inhibitors of the Glycine Transporter Type 2
Caulfield, Wilson L, Collie, Iain T, Dickins, Rachel S, Epemolu, Ola, McGuire, Ross, Hill, David R, McVey, Gillian, Morphy, J. Richard, Rankovic, Zoran, Sundaram, Hardy
Published in Journal of medicinal chemistry (16.08.2001)
Published in Journal of medicinal chemistry (16.08.2001)
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Discovery of Indoline-2-carboxamide Derivatives as a New Class of Brain-Penetrant Inhibitors of Trypanosoma brucei
Cleghorn, Laura A. T., Albrecht, Sébastien, Stojanovski, Laste, Simeons, Frederick R. J., Norval, Suzanne, Kime, Robert, Collie, Iain T., De Rycker, Manu, Campbell, Lorna, Hallyburton, Irene, Frearson, Julie A., Wyatt, Paul G., Read, Kevin D., Gilbert, Ian H.
Published in Journal of medicinal chemistry (08.10.2015)
Published in Journal of medicinal chemistry (08.10.2015)
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Journal Article
Development of Small-Molecule Trypanosoma brucei N-Myristoyltransferase Inhibitors: Discovery and Optimisation of a Novel Binding Mode
Spinks, Daniel, Smith, Victoria, Thompson, Stephen, Robinson, David A., Luksch, Torsten, Smith, Alasdair, Torrie, Leah S., McElroy, Stuart, Stojanovski, Laste, Norval, Suzanne, Collie, Iain T., Hallyburton, Irene, Rao, Bhavya, Brand, Stephen, Brenk, Ruth, Frearson, Julie A., Read, Kevin D., Wyatt, Paul G., Gilbert, Ian H.
Published in ChemMedChem (01.11.2015)
Published in ChemMedChem (01.11.2015)
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Identification of Inhibitors of the Leishmania cdc2-Related Protein Kinase CRK3
Cleghorn, Laura A. T., Woodland, Andrew, Collie, Iain T., Torrie, Leah S., Norcross, Neil, Luksch, Torsten, Mpamhanga, Chido, Walker, Roderick G., Mottram, Jeremy C., Brenk, Ruth, Frearson, Julie A., Gilbert, Ian H., Wyatt, Paul G.
Published in ChemMedChem (09.12.2011)
Published in ChemMedChem (09.12.2011)
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A Novel Allosteric Inhibitor of the Uridine Diphosphate N‑Acetylglucosamine Pyrophosphorylase from Trypanosoma brucei
Urbaniak, Michael D, Collie, Iain T, Fang, Wenxia, Aristotelous, Tonia, Eskilsson, Susanne, Raimi, Olawale G, Harrison, Justin, Navratilova, Iva Hopkins, Frearson, Julie A, van Aalten, Daan M. F, Ferguson, Michael A. J
Published in ACS chemical biology (20.09.2013)
Published in ACS chemical biology (20.09.2013)
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Design, Synthesis and Biological Evaluation of Novel Inhibitors of Trypanosoma brucei Pteridine Reductase 1
Spinks, Daniel, Ong, Han B., Mpamhanga, Chidochangu P., Shanks, Emma J., Robinson, David A., Collie, Iain T., Read, Kevin D., Frearson, Julie A., Wyatt, Paul G., Brenk, Ruth, Fairlamb, Alan H., Gilbert, Ian H.
Published in ChemMedChem (07.02.2011)
Published in ChemMedChem (07.02.2011)
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Journal Article
Quinol derivatives as potential trypanocidal agents
Capes, Amy, Patterson, Stephen, Wyllie, Susan, Hallyburton, Irene, Collie, Iain T., McCarroll, Andrew J., Stevens, Malcolm F.G., Frearson, Julie A., Wyatt, Paul G., Fairlamb, Alan H., Gilbert, Ian H.
Published in Bioorganic & medicinal chemistry (15.02.2012)
Published in Bioorganic & medicinal chemistry (15.02.2012)
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Journal Article
Cover Picture: Development of Small-Molecule Trypanosoma brucei N-Myristoyltransferase Inhibitors: Discovery and Optimisation of a Novel Binding Mode (ChemMedChem 11/2015)
Spinks, Daniel, Smith, Victoria, Thompson, Stephen, Robinson, David A., Luksch, Torsten, Smith, Alasdair, Torrie, Leah S., McElroy, Stuart, Stojanovski, Laste, Norval, Suzanne, Collie, Iain T., Hallyburton, Irene, Rao, Bhavya, Brand, Stephen, Brenk, Ruth, Frearson, Julie A., Read, Kevin D., Wyatt, Paul G., Gilbert, Ian H.
Published in ChemMedChem (01.11.2015)
Published in ChemMedChem (01.11.2015)
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Journal Article
Optimisation of the Anti-Trypanosoma brucei Activity of the Opioid Agonist U50488
Smith, Victoria C., Cleghorn, Laura A. T., Woodland, Andrew, Spinks, Daniel, Hallyburton, Irene, Collie, Iain T., Yi Mok, N., Norval, Suzanne, Brenk, Ruth, Fairlamb, Alan H., Frearson, Julie A., Read, Kevin D., Gilbert, Ian H., Wyatt, Paul G.
Published in ChemMedChem (04.10.2011)
Published in ChemMedChem (04.10.2011)
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Cover Picture: Synthesis and Evaluation of Indatraline-Based Inhibitors for Trypanothione Reductase / Design, Synthesis and Biological Evaluation of Novel Inhibitors of Trypanosoma brucei Pteridine Reductase 1 / Modified 5′-Trityl Nucleosides as Inhibitors of Plasmodium falciparum dUTPase (ChemMedChem 2/2011)
Walton, Jeffrey G. A., Jones, Deuan C., Kiuru, Paula, Durie, Alastair J., Westwood, Nicholas J., Fairlamb, Alan H., Spinks, Daniel, Ong, Han B., Mpamhanga, Chidochangu P., Shanks, Emma J., Robinson, David A., Collie, Iain T., Read, Kevin D., Frearson, Julie A., Wyatt, Paul G., Brenk, Ruth, Fairlamb, Alan H., Gilbert, Ian H., Ruda, Gian Filippo, Nguyen, Corinne, Ziemkowski, Przemysław, Felczak, Krzysztof, Kasinathan, Ganasan, Musso-Buendia, Alexander, Sund, Christian, Zhou, Xiao Xiong, Kaiser, Marcel, Ruiz-Pérez, Luis M., Brun, Reto, Kulikowski, Tadeusz, Johansson, Nils Gunnar, González-Pacanowska, Dolores, Gilbert, Ian H.
Published in ChemMedChem (07.02.2011)
Published in ChemMedChem (07.02.2011)
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