Methods to measure the intracellular concentration of unlabeled compounds within cultured cells using liquid chromatography/tandem mass spectrometry
Colletti, Lynn M., Liu, Yaya, Koev, Gennadiy, Richardson, Paul L., Chen, Chih-Ming, Kati, Warren
Published in Analytical biochemistry (15.12.2008)
Published in Analytical biochemistry (15.12.2008)
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Estimation of Serum-Free 50-Percent Inhibitory Concentrations for Human Immunodeficiency Virus Protease Inhibitors Lopinavir and Ritonavir
HICKMAN, Dean, VASAVANONDA, Sudthida, NEQUIST, George, COLLETTI, Lynn, KATI, Warren M, BERTZ, Richard, HSU, Ann, KEMPF, Dale J
Published in Antimicrobial Agents and Chemotherapy (01.08.2004)
Published in Antimicrobial Agents and Chemotherapy (01.08.2004)
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Design and synthesis of pseudo-Symmetric HIV protease inhibitors containing a novel hydroxymethylcarbonyl (HMC)-Hydrazide isostere
Hidaka, Koushi, Kimura, Tooru, Hayashi, Yoshio, McDaniel, Keith F, Dekhtyar, Tatyana, Colletti, Lynn, Kiso, Yoshiaki
Published in Bioorganic & medicinal chemistry letters (06.01.2003)
Published in Bioorganic & medicinal chemistry letters (06.01.2003)
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Synthesis and Biological Characterization of Aryl Uracil Inhibitors of Hepatitis C Virus NS5B Polymerase: Discovery of ABT-072, a trans-Stilbene Analog with Good Oral Bioavailability
Randolph, John T, Krueger, A. Chris, Donner, Pamela L, Pratt, John K, Liu, Dachun, Motter, Christopher E, Rockway, Todd W, Tufano, Michael D, Wagner, Rolf, Lim, Hock B, Beyer, Jill M, Mondal, Rubina, Panchal, Neeta S, Colletti, Lynn, Liu, Yaya, Koev, Gennadiy, Kati, Warren M, Hernandez, Lisa E, Beno, David W. A, Longenecker, Kenton L, Stewart, Kent D, Dumas, Emily O, Molla, Akhteruzzaman, Maring, Clarence J
Published in Journal of medicinal chemistry (08.02.2018)
Published in Journal of medicinal chemistry (08.02.2018)
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High potency improvements to weak aryl uracil HCV polymerase inhibitor leads
Donner, Pamela, Randolph, John T., Huang, Peggy, Wagner, Rolf, Maring, Clarence, Lim, Ben Hock, Colletti, Lynn, Liu, Yaya, Mondal, Rubina, Beyer, Jill, Koev, Gennadiy, Marsh, Kennan, Beno, David, Longenecker, Kenton, Pilot-Matias, Tami, Kati, Warren, Molla, Akhter, Kempf, Dale
Published in Bioorganic & medicinal chemistry letters (01.08.2013)
Published in Bioorganic & medicinal chemistry letters (01.08.2013)
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2-Pyridyl P1′-Substituted Symmetry-Based Human Immunodeficiency Virus Protease Inhibitors (A-792611 and A-790742) with Potential for Convenient Dosing and Reduced Side Effects
DeGoey, David A, Grampovnik, David J, Flentge, Charles A, Flosi, William J, Chen, Hui-ju, Yeung, Clinton M, Randolph, John T, Klein, Larry L, Dekhtyar, Tatyana, Colletti, Lynn, Marsh, Kennan C, Stoll, Vincent, Mamo, Mulugeta, Morfitt, David C, Nguyen, Bach, Schmidt, James M, Swanson, Sue J, Mo, Hongmei, Kati, Warren M, Molla, Akhteruzzaman, Kempf, Dale J
Published in Journal of medicinal chemistry (23.04.2009)
Published in Journal of medicinal chemistry (23.04.2009)
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Synthesis, antiviral activity, and pharmacokinetic evaluation of P3 pyridylmethyl analogs of oximinoarylsulfonyl HIV-1 protease inhibitors
Randolph, John T., Huang, Peggy P., Flosi, William J., DeGoey, David, Klein, Larry L., Yeung, Clinton M., Flentge, Charles, Sun, Mingua, Zhao, Chen, Dekhtyar, Tatyana, Mo, Hongmei, Colletti, Lynn, Kati, Warren, Marsh, Kennan C., Molla, Akhteruzzaman, Kempf, Dale J.
Published in Bioorganic & medicinal chemistry (15.06.2006)
Published in Bioorganic & medicinal chemistry (15.06.2006)
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