Vanillin enones as selective inhibitors of the cancer associated carbonic anhydrase isoforms IX and XII. The out of the active site pocket for the design of selective inhibitors?
Riafrecha, Leonardo E., Le Pors, Macarena S., Lavecchia, Martín J., Bua, Silvia, Supuran, Claudiu T., Colinas, Pedro A.
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2021)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2021)
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Journal Article
Glycosidic carbonic anhydrase IX inhibitors: A sweet approach against cancer
Winum, Jean-Yves, Colinas, Pedro A., Supuran, Claudiu T.
Published in Bioorganic & medicinal chemistry (15.03.2013)
Published in Bioorganic & medicinal chemistry (15.03.2013)
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Journal Article
C-glycosides incorporating the 6-methoxy-2-naphthyl moiety are selective inhibitors of fungal and bacterial carbonic anhydrases
Riafrecha, Leonardo E., Vullo, Daniela, Supuran, Claudiu T., Colinas, Pedro A.
Published in Journal of enzyme inhibition and medicinal chemistry (03.09.2015)
Published in Journal of enzyme inhibition and medicinal chemistry (03.09.2015)
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Journal Article
Attachment of carbohydrates to methoxyaryl moieties leads to highly selective inhibitors of the cancer associated carbonic anhydrase isoforms IX and XII
Riafrecha, Leonardo E., Rodríguez, Oscar M., Vullo, Daniela, Supuran, Claudiu T., Colinas, Pedro A.
Published in Bioorganic & medicinal chemistry (01.10.2014)
Published in Bioorganic & medicinal chemistry (01.10.2014)
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Journal Article
Inhibition of the β-carbonic anhydrases from Mycobacterium tuberculosis with C-cinnamoyl glycosides: Identification of the first inhibitor with anti-mycobacterial activity
Buchieri, María V., Riafrecha, Leonardo E., Rodríguez, Oscar M., Vullo, Daniela, Morbidoni, Héctor R., Supuran, Claudiu T., Colinas, Pedro A.
Published in Bioorganic & medicinal chemistry letters (01.02.2013)
Published in Bioorganic & medicinal chemistry letters (01.02.2013)
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Journal Article
In vitro antitumor activity of N-glycosyl sulfonamides
Crespo, Rosana, de Bravo, Margarita G., Colinas, Pedro A., Bravo, Rodolfo D.
Published in Bioorganic & medicinal chemistry letters (15.11.2010)
Published in Bioorganic & medicinal chemistry letters (15.11.2010)
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Journal Article
Inhibition of β-carbonic anhydrases from Brucella suis with C-cinnamoyl glycosides incorporating the phenol moiety
Riafrecha, Leonardo E., Vullo, Daniela, Ouahrani-Bettache, Safia, Köhler, Stephan, Dumy, Pascal, Winum, Jean-Yves, Supuran, Claudiu T., Colinas, Pedro A.
Published in Journal of enzyme inhibition and medicinal chemistry (02.11.2015)
Published in Journal of enzyme inhibition and medicinal chemistry (02.11.2015)
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Journal Article
Anti-tubercular and antioxidant activities of C-glycosyl carbonic anhydrase inhibitors: towards the development of novel chemotherapeutic agents against Mycobacterium tuberculosis
Zaro, María J., Bortolotti, Ana, Riafrecha, Leonardo E., Concellón, Analía, Morbidoni, Héctor R., Colinas, Pedro A.
Published in Journal of enzyme inhibition and medicinal chemistry (01.11.2016)
Published in Journal of enzyme inhibition and medicinal chemistry (01.11.2016)
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Journal Article
N-β-Glycosyl sulfamides are selective inhibitors of the cancer associated carbonic anhydrase isoforms IX and XII
Rodríguez, Oscar M., Maresca, Alfonso, Témpera, Carlos A., Bravo, Rodolfo D., Colinas, Pedro A., Supuran, Claudiu T.
Published in Bioorganic & medicinal chemistry letters (01.08.2011)
Published in Bioorganic & medicinal chemistry letters (01.08.2011)
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Journal Article
Efficient synthesis of 2,3-unsaturated sulfonamidoglycosides by Amberlyst 15
Témpera, Carlos A., Colinas, Pedro A., Bravo, Rodolfo D.
Published in Tetrahedron letters (13.10.2010)
Published in Tetrahedron letters (13.10.2010)
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Journal Article
A combined theoretical and spectroscopic study of 4,6-di- O-acetyl-2,3-dideoxy- d- erythro-hex-2-enopyranosyl sulfamide: a novel glycosyl carbonic anhydrase IX inhibitor
Lavecchia, Martín J., Diez, Reinaldo Pis, Colinas, Pedro A.
Published in Carbohydrate research (15.02.2011)
Published in Carbohydrate research (15.02.2011)
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Journal Article
Carbonic anhydrase inhibitors. Inhibition of cytosolic isoforms I and II, and extracellular isoforms IV, IX, and XII with sulfamides incorporating sugar moieties
Colinas, Pedro A., Bravo, Rodolfo D., Vullo, Daniela, Scozzafava, Andrea, Supuran, Claudiu T.
Published in Bioorganic & medicinal chemistry letters (15.09.2007)
Published in Bioorganic & medicinal chemistry letters (15.09.2007)
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Journal Article
Conformational behavior of peracetylated β-d-mannopyranosyl methanesulfonamide: implications for the mechanism of sulfonamidoglycosylation of carbohydrate derivatives
Lavecchia, Martín J., Rodríguez, Oscar M., Echeverría, Gustavo A., Pis Diez, Reinaldo, Colinas, Pedro A.
Published in Carbohydrate research (01.11.2012)
Published in Carbohydrate research (01.11.2012)
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