Enhancing Giardicidal Activity and Aqueous Solubility through the Development of “RetroABZ”, a Regioisomer of Albendazole: In Vitro, In Vivo, and In Silico Studies
Martínez-Conde, Carlos, Colín-Lozano, Blanca, Gutiérrez-Hernández, Abraham, Hernández-Núñez, Emanuel, Yépez-Mulia, Lilián, Colorado-Pablo, Luis Fernando, Aguayo-Ortiz, Rodrigo, Escalante, Jaime, Rivera-Leyva, Julio C., Sánchez-Carranza, Jessica Nayelli, Barbosa-Cabrera, Elizabeth, Navarrete-Vazquez, Gabriel
Published in International journal of molecular sciences (01.10.2023)
Published in International journal of molecular sciences (01.10.2023)
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Journal Article
Design, Synthesis and in Combo Antidiabetic Bioevaluation of Multitarget Phenylpropanoic Acids
Colín-Lozano, Blanca, Estrada-Soto, Samuel, Chávez-Silva, Fabiola, Gutiérrez-Hernández, Abraham, Cerón-Romero, Litzia, Giacoman-Martínez, Abraham, Almanza-Pérez, Julio Cesar, Hernández-Núñez, Emanuel, Wang, Zhilong, Xie, Xin, Cappiello, Mario, Balestri, Francesco, Mura, Umberto, Navarrete-Vazquez, Gabriel
Published in Molecules (Basel, Switzerland) (06.02.2018)
Published in Molecules (Basel, Switzerland) (06.02.2018)
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Journal Article
Design, Synthesis, and In Silico Multitarget Pharmacological Simulations of Acid Bioisosteres with a Validated In Vivo Antihyperglycemic Effect
Domínguez-Mendoza, Elix Alberto, Galván-Ciprés, Yelzyn, Martínez-Miranda, Josué, Miranda-González, Cristian, Colín-Lozano, Blanca, Hernández-Núñez, Emanuel, Hernández-Bolio, Gloria I, Palomino-Hernández, Oscar, Navarrete-Vazquez, Gabriel
Published in Molecules (Basel, Switzerland) (04.02.2021)
Published in Molecules (Basel, Switzerland) (04.02.2021)
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Journal Article
Metronidazole and Secnidazole Carbamates: Synthesis, Antiprotozoal Activity, and Molecular Dynamics Studies
Rocha-Garduño, Genaro, Hernández-Martínez, Norma Angélica, Colín-Lozano, Blanca, Estrada-Soto, Samuel, Hernández-Núñez, Emanuel, Prieto-Martínez, Fernando Daniel, Medina-Franco, José L, Chale-Dzul, Juan Bautista, Moo-Puc, Rosa, Navarrete-Vázquez, Gabriel
Published in Molecules (Basel, Switzerland) (12.02.2020)
Published in Molecules (Basel, Switzerland) (12.02.2020)
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Journal Article
Antidiabetic effect of Cordia morelosana, chemical and pharmacological studies
Giles-Rivas, Diana, Estrada-Soto, Samuel, Aguilar-Guadarrama, A. Berenice, Almanza-Pérez, Julio, García-Jiménez, Sara, Colín-Lozano, Blanca, Navarrete-Vázquez, Gabriel, Villalobos-Molina, Rafael
Published in Journal of ethnopharmacology (06.04.2020)
Published in Journal of ethnopharmacology (06.04.2020)
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Journal Article
Synthesis, antiproliferative evaluation and in silico studies of a novel steroidal spiro morpholinone
Cobos-Ontiveros, Luis A., Romero-Hernández, Laura L., Mastranzo-Sánchez, Eduardo B., Colín-Lozano, Blanca, Puerta, Adrián, Padrón, José M., Merino-Montiel, Penélope, Vega Baez, Jose Luis, Montiel-Smith, Sara
Published in Steroids (01.04.2023)
Published in Steroids (01.04.2023)
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Journal Article
Proton pump inhibitors drastically modify triosephosphate isomerase from Giardia lamblia at functional and structural levels, providing molecular leads in the design of new antigiardiasic drugs
García-Torres, Itzhel, de la Mora-de la Mora, Ignacio, Marcial-Quino, Jaime, Gómez-Manzo, Saúl, Vanoye-Carlo, América, Navarrete-Vázquez, Gabriel, Colín-Lozano, Blanca, Gutiérrez-Castrellón, Pedro, Sierra-Palacios, Edgar, López-Velázquez, Gabriel, Enríquez-Flores, Sergio
Published in Biochimica et biophysica acta (01.01.2016)
Published in Biochimica et biophysica acta (01.01.2016)
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Journal Article
Synthesis, In Vitro, In Vivo and In Silico Antidiabetic Bioassays of 4-Nitro(thio)phenoxyisobutyric Acids Acting as Unexpected PPARγ Modulators: An In Combo Study
Colin-Lozano, Blanca, Torres-Gomez, Héctor, Hidalgo-Figueroa, Sergio, Chávez-Silva, Fabiola, Estrada-Soto, Samuel, Almanza-Pérez, Julio Cesar, Navarrete-Vazquez, Gabriel
Published in Pharmaceuticals (Basel, Switzerland) (15.01.2022)
Published in Pharmaceuticals (Basel, Switzerland) (15.01.2022)
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Journal Article
Synthesis, in vitro and in vivo giardicidal activity of nitrothiazole-NSAID chimeras displaying broad antiprotozoal spectrum
Colín-Lozano, Blanca, León-Rivera, Ismael, Chan-Bacab, Manuel Jesús, Ortega-Morales, Benjamín Otto, Moo-Puc, Rosa, López-Guerrero, Vanessa, Hernández-Núñez, Emanuel, Argüello-Garcia, Raúl, Scior, Thomas, Barbosa-Cabrera, Elizabeth, Navarrete-Vázquez, Gabriel
Published in Bioorganic & medicinal chemistry letters (01.08.2017)
Published in Bioorganic & medicinal chemistry letters (01.08.2017)
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Journal Article
Synthesis of nitro(benzo)thiazole acetamides and in vitro antiprotozoal effect against amitochondriate parasites Giardia intestinalis and Trichomonas vaginalis
Navarrete-Vázquez, Gabriel, Chávez-Silva, Fabiola, Colín-Lozano, Blanca, Estrada-Soto, Samuel, Hidalgo-Figueroa, Sergio, Guerrero-Álvarez, Jorge, Méndez, Sara T., Reyes-Vivas, Horacio, Oria-Hernández, Jesús, Canul-Canché, Jaqueline, Ortiz-Andrade, Rolffy, Moo-Puc, Rosa
Published in Bioorganic & medicinal chemistry (01.05.2015)
Published in Bioorganic & medicinal chemistry (01.05.2015)
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Journal Article
Novel Coumarin‐steroid/terpenoid Hybrids: In vitro and in silico Anticancer Studies
Martínez-Lara, Rosa I., Cobos-Ontiveros, Luis A., Meza-Ireta, Silvia A., Martínez-Montiel, Mónica, Colín-Lozano, Blanca, Puerta, Adrián, Padrón, José M., López, Óscar, Vega-Báez, José Luis, Merino-Montiel, Penélope, Montiel-Smith, Sara
Published in Chemistry & biodiversity (13.08.2024)
Published in Chemistry & biodiversity (13.08.2024)
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Journal Article
Molecular Docking Studies of Estrone-Coumarin Derivatives as Aromatase and 17β-HSD1 Inhibitors Related to Hormone Receptor Positive (HR+) Breast Cancer
Meza-Ireta, Silvia Alejandra, Colin-Lozano, Blanca, Merino-Montiel, Penélope, Vega-Báez, José Luis, Montiel-Smith, Sara
Published in Advances in enzyme research (2022)
Published in Advances in enzyme research (2022)
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Journal Article
Steroidal Plant Growth Promoters vs. Phytopathogens, via Enzymatic Regulation; An in Silico Approach
Carrasco-Carballo, Alan, Marín-Merino, Emiliano, Merino-Montiel, Penélope, Colin-Lozano, Blanca, Hilerio, Sandra Luz Cabrera, Hilario-Martínez, Jazmin Ciciolil, Sandoval-Ramírez, Jesús
Published in Advances in enzyme research (2021)
Published in Advances in enzyme research (2021)
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