Search Results - "Coesemans, Erwin" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Pharmacological Profile of JNJ-27141491 [(S)-3-[3,4-Difluorophenyl)-propyl]-5-isoxazol-5-yl-2-thioxo-2,3-dihydro-1H-imidazole-4-carboxyl Acid Methyl Ester], as a Noncompetitive and Orally Active Antagonist of the Human Chemokine Receptor CCR2

by Buntinx, Mieke, Hermans, Bart, Goossens, Jan, Moechars, Dieder, Gilissen, Ron A H J, Doyon, Julien, Boeckx, Staf, Coesemans, Erwin, Van Lommen, Guy, Van Wauwe, Jean P
Published in The Journal of pharmacology and experimental therapeutics (01.10.2008)

Get full text

Journal Article

Spiro-Azetidine Oxindoles as Long-Acting Injectables for Pre-Exposure Prophylaxis against Respiratory Syncytial Virus Infections

Spiro-Azetidine Oxindoles as Long-Acting Injectables for Pre-Exposure Prophylaxis against Respiratory Syncytial Virus Infections

by Kesteleyn, Bart, Herschke, Florence, Darville, Nicolas, Stoops, Bart, Jacobs, Tom, Jacoby, Edgar, Shaffer, Paul, Lammens, Lieve, Van Rompaey, Dries, Matcha, Kiran, Martinez Lamenca, Carolina, Coesemans, Erwin, Hache, Geerwin, Pieters, Serge, Lecomte, Morgan, Hu, Lili, Demin, Samuel, Milligan, Cynthia, Abeywickrema, Pravien, De Bruyn, Suzanne, Van Den Berg, Joke, Ysebaert, Nina, De Zwart, Loeckie, Nájera, Isabel, Rigaux, Peter, Roymans, Dirk, Jonckers, Tim H. M.
Published in Journal of medicinal chemistry (11.07.2024)

Get full text

Journal Article

Discovery of JNJ-1802, a First-in-Class Pan-Serotype Dengue Virus NS4B Inhibitor

Discovery of JNJ-1802, a First-in-Class Pan-Serotype Dengue Virus NS4B Inhibitor

by Kesteleyn, Bart, Bonfanti, Jean-François, Bardiot, Dorothée, De Boeck, Benoît, Goethals, Olivia, Kaptein, Suzanne J. F., Stoops, Bart, Coesemans, Erwin, Fortin, Jérôme, Muller, Philippe, Doublet, Frédéric, Carlens, Gunter, Koukni, Mohamed, Smets, Wim, Raboisson, Pierre, Chaltin, Patrick, Simmen, Kenny, Loock, Marnix Van, Neyts, Johan, Marchand, Arnaud, Jonckers, Tim H. M.
Published in Journal of medicinal chemistry (14.03.2024)

Get full text

Journal Article

(S)-2--1-(1H-인돌-3-일)에테논유도체의 제조 방법

(S)-2--1-(1H-인돌-3-일)에테논유도체의 제조 방법

by OOST RIK, COESEMANS ERWIN, ERIKSSON CARL ARNE MAGNUS, SCHWEITZER CHAPUT BERTRAND, WU KAI
Year of Publication 04.03.2024

Get full text

Patent

Discovery of Acyl-Indole Derivatives as Pan-Serotype Dengue Virus NS4B Inhibitors

Discovery of Acyl-Indole Derivatives as Pan-Serotype Dengue Virus NS4B Inhibitors

by Kesteleyn, Bart, Bardiot, Dorothée, Bonfanti, Jean-François, De Boeck, Benoît, Goethals, Olivia, Kaptein, Suzanne J. F., Stoops, Bart, Coesemans, Erwin, Fortin, Jérôme, Muller, Philippe, Doublet, Frédéric, Carlens, Gunter, Koukni, Mohamed, Smets, Wim, Raboisson, Pierre, Chaltin, Patrick, Simmen, Kenny, Van Loock, Marnix, Neyts, Johan, Marchand, Arnaud, Jonckers, Tim H. M.
Published in Journal of medicinal chemistry (13.07.2023)

Get full text

Journal Article

Characterization of a dengue NS4B inhibitor originating from an HCV small molecule library

Characterization of a dengue NS4B inhibitor originating from an HCV small molecule library

by Hernandez-Morales, Ilane, Geluykens, Peggy, Clynhens, Marleen, Strijbos, Rudy, Goethals, Olivia, Megens, Sarah, Verheyen, Nick, Last, Stefaan, McGowan, David, Coesemans, Erwin, De Boeck, Benoît, Stoops, Bart, Devogelaere, Benoit, Pauwels, Frederik, Vandyck, Koen, Berke, Jan Martin, Raboisson, Pierre, Simmen, Kenneth, Lory, Pedro, Van Loock, Marnix
Published in Antiviral research (01.11.2017)

Get full text

Journal Article

HBV 감염 또는 HBV-유도성 질환의 치료에 유용한 아미드 유도체

HBV 감염 또는 HBV-유도성 질환의 치료에 유용한 아미드 유도체

by BERKE JAN MARTIN, JACOBY EDGAR, GROSSE SANDRINE CELINE, COESEMANS ERWIN, LAST STEFAAN JULIEN, KESTELEYN BART RUDOLF ROMANIE, DOEBELIN CHRISTELLE CATHERINE CECILE, JONCKERS TIM HUGO MARIA, OBRINGER MICHEL, VERSCHUEREN WIM GASTON
Year of Publication 13.01.2022

Get full text

Patent

뎅기 바이러스 복제 억제제로서의 치환 인돌린 유도체

뎅기 바이러스 복제 억제제로서의 치환 인돌린 유도체

by MARCHAND ARNAUD DIDIER M, BONFANTI JEAN FRANCOIS, COESEMANS ERWIN, KESTELEYN BART RUDOLF ROMANIE, RABOISSON PIERRE JEAN MARIE BERNARD, BARDIOT DOROTHEE ALICE MARIE EVE
Year of Publication 10.12.2019

Get full text

Patent

뎅기 바이러스 복제 억제제로서의 치환 인돌린 유도체

뎅기 바이러스 복제 억제제로서의 치환 인돌린 유도체

by MARCHAND ARNAUD DIDIER M, BONFANTI JEAN FRANCOIS, COESEMANS ERWIN, KESTELEYN BART RUDOLF ROMANIE, DE BOECK BENOIT CHRISTIAN ALBERT GHISLAIN, RABOISSON PIERRE JEAN MARIE BERNARD, BARDIOT DOROTHEE ALICE MARIE EVE
Year of Publication 30.01.2020

Get full text

Patent

뎅기 바이러스 복제 억제제로서의 치환 인돌린 유도체

뎅기 바이러스 복제 억제제로서의 치환 인돌린 유도체

by MARCHAND ARNAUD DIDIER M, BONFANTI JEAN FRANCOIS, COESEMANS ERWIN, KESTELEYN BART RUDOLF ROMANIE, RABOISSON PIERRE JEAN MARIE BERNARD, BARDIOT DOROTHEE ALICE MARIE EVE, MERCEY GUILLAUME JEAN MAURICE, FORTIN JEROME MICHEL CLAUDE
Year of Publication 29.01.2020

Get full text

Patent

뎅기 바이러스 복제 억제제로서 치환된 인돌 화합물 유도체

뎅기 바이러스 복제 억제제로서 치환된 인돌 화합물 유도체

by MARCHAND ARNAUD DIDIER M, BONFANTI JEAN FRANCOIS, COESEMANS ERWIN, KESTELEYN BART RUDOLF ROMANIE, RABOISSON PIERRE JEAN MARIE BERNARD, BARDIOT DOROTHEE ALICE MARIE EVE
Year of Publication 07.12.2018

Get full text

Patent

Synthesis and structure–activity relationship of benzetimide derivatives as human CXCR3 antagonists

Synthesis and structure–activity relationship of benzetimide derivatives as human CXCR3 antagonists

by Bongartz, Jean-Pierre, Buntinx, Mieke, Coesemans, Erwin, Hermans, Bart, Lommen, Guy Van, Wauwe, Jean Van
Published in Bioorganic & medicinal chemistry letters (01.11.2008)

Get full text

Journal Article

Pharmacological Profile of JNJ-27141491 [( S )-3-[3,4-Difluorophenyl)-propyl]-5-isoxazol-5-yl-2-thioxo-2,3-dihydro-1 H -imidazole-4-carboxyl Acid Methyl Ester], as a Noncompetitive and Orally Active Antagonist of the Human Chemokine Receptor CCR2

by Buntinx, Mieke, Hermans, Bart, Goossens, Jan, Moechars, Dieder, Gilissen, Ron A. H. J., Doyon, Julien, Boeckx, Staf, Coesemans, Erwin, Van Lommen, Guy, Van Wauwe, Jean P.
Published in The Journal of pharmacology and experimental therapeutics (01.10.2008)

Get full text

Journal Article

Design and Synthesis of a Series of Piperazine‐1‐carboxamidine Derivatives with Antifungal Activity Resulting from Accumulation of Endogenous Reactive Oxygen Species

Design and Synthesis of a Series of Piperazine‐1‐carboxamidine Derivatives with Antifungal Activity Resulting from Accumulation of Endogenous Reactive Oxygen Species

by François, Isabelle E., Thevissen, Karin, Pellens, Klaartje, Meert, Els M., Heeres, Jan, Freyne, Eddy, Coesemans, Erwin, Viellevoye, Marcel, Deroose, Frederik, Martinez Gonzalez, Sonia, Pastor, Joaquin, Corens, David, Meerpoel, Lieven, Borgers, Marcel, Ausma, Jannie, Dispersyn, Gerrit D., Cammue, Bruno P.
Published in ChemMedChem (05.10.2009)

Get full text

Journal Article

2-Mercaptoimidazoles, a new class of potent CCR2 antagonists

2-Mercaptoimidazoles, a new class of potent CCR2 antagonists

by Van Lommen, Guy, Doyon, Julien, Coesemans, Erwin, Boeckx, Staf, Cools, Marina, Buntinx, Mieke, Hermans, Bart, Jean VanWauwe
Published in Bioorganic & medicinal chemistry letters (01.02.2005)

Get full text

Journal Article

Discovery of Potent, Orally Bioavailable Small-Molecule Inhibitors of the Human CCR2 Receptor

Discovery of Potent, Orally Bioavailable Small-Molecule Inhibitors of the Human CCR2 Receptor

by Doyon, Julien, Coesemans, Erwin, Boeckx, Staf, Buntinx, Mieke, Hermans, Bart, Van Wauwe, Jean P., Gilissen, Ron A. H. J., De Groot, Alex H. J., Corens, David, Van Lommen, Guy
Published in ChemMedChem (14.04.2008)

Get full text

Journal Article

PROCESSES FOR THE PREPARATION OF (S)-2-(4-CHLORO-2-METHOXYPHENYL)-2-((3 -METHOXY-5-(M ETHYLSULFONYL)PHENYL)AMINO)-1 -(1H-INDOL-3-YL)ETHENONE DERIVATIVES

PROCESSES FOR THE PREPARATION OF (S)-2-(4-CHLORO-2-METHOXYPHENYL)-2-((3 -METHOXY-5-(M ETHYLSULFONYL)PHENYL)AMINO)-1 -(1H-INDOL-3-YL)ETHENONE DERIVATIVES

by Wu, Kai, Eriksson, Carl Arne Magnus, Oost, Rik, Schweitzer-Chaput, Bertrand, Coesemans, Erwin
Year of Publication 19.09.2024

Get full text

Patent

PROCESSES FOR THE PREPARATION OF (S)-2-(4-CHLORO-2-METHOXYPHENYL)-2-((3-METHOXY-5-(METHYLSULFONYL)PHENYL)AMINO)-1 -(1H-INDOL-3-YL)ETHENONE DERIVATIVES

PROCESSES FOR THE PREPARATION OF (S)-2-(4-CHLORO-2-METHOXYPHENYL)-2-((3-METHOXY-5-(METHYLSULFONYL)PHENYL)AMINO)-1 -(1H-INDOL-3-YL)ETHENONE DERIVATIVES

by COESEMANS, Erwin, SCHWEITZERAPUT, Bertrand, WU, Kai, ERIKSSON, Carl Arne Magnus, OOST, Rik
Year of Publication 08.05.2024

Get full text

Patent

PROCESSES FOR THE PREPARATION OF (S)-2-(4-CHLORO-2-METHOXYPHENYL)-2-((3-METHOXY-5-(METHYLSULFONYL)PHENYL)AMINO)-1 -(1H-INDOL-3-YL)ETHENONE DERIVATIVES

PROCESSES FOR THE PREPARATION OF (S)-2-(4-CHLORO-2-METHOXYPHENYL)-2-((3-METHOXY-5-(METHYLSULFONYL)PHENYL)AMINO)-1 -(1H-INDOL-3-YL)ETHENONE DERIVATIVES

by COESEMANS, Erwin, SCHWEITZERAPUT, Bertrand, WU, Kai, ERIKSSON, Carl Arne Magnus, OOST, Rik
Year of Publication 15.02.2024

Get full text

Patent

Processes for the preparation of (s)-2-(4-chloro-2-methoxyphenyl)-2-((3-methoxy-5-(methylsulfonyl)phenyl)amino)-1 -(1h-indol-3-yl)ethenone derivatives

Processes for the preparation of (s)-2-(4-chloro-2-methoxyphenyl)-2-((3-methoxy-5-(methylsulfonyl)phenyl)amino)-1 -(1h-indol-3-yl)ethenone derivatives

by COESEMANS Erwin, ERIKSSON Carl Arne Magnus, OOST Rik, SCHWEITZERAPUT Bertrand, WU Kai
Year of Publication 01.02.2024

Get full text

Patent

1
2
3
4
5
6
7
8
9
10
11
Next
[17]