Pharmacological properties of S1RA, a new sigma‐1 receptor antagonist that inhibits neuropathic pain and activity‐induced spinal sensitization
Romero, L, Zamanillo, D, Nadal, X, Sánchez‐Arroyos, R, Rivera‐Arconada, I, Dordal, A, Montero, A, Muro, A, Bura, A, Segalés, C, Laloya, M, Hernández, E, Portillo‐Salido, E, Escriche, M, Codony, X, Encina, G, Burgueño, J, Merlos, M, Baeyens, JM, Giraldo, J, López‐García, JA, Maldonado, R, Plata‐Salamán, CR, Vela, JM
Published in British journal of pharmacology (01.08.2012)
Published in British journal of pharmacology (01.08.2012)
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Selective 5-HT6 receptor ligands: progress in the development of a novel pharmacological approach to the treatment of obesity and related metabolic disorders
Heal, D J, Smith, S L, Fisas, A, Codony, X, Buschmann, H
Published in Pharmacology & therapeutics (Oxford) (01.02.2008)
Published in Pharmacology & therapeutics (Oxford) (01.02.2008)
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Chronic 5‐HT6 receptor modulation by E‐6837 induces hypophagia and sustained weight loss in diet‐induced obese rats
Fisas, A, Codony, X, Romero, G, Dordal, A, Giraldo, J, Mercé, R, Holenz, J, Vrang, N, Sørensen, R V, Heal, D, Buschmann, H, Pauwels, P J
Published in British journal of pharmacology (01.06.2007)
Published in British journal of pharmacology (01.06.2007)
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Administration of a co-crystal of tramadol and celecoxib in a 1:1 molecular ratio produces synergistic antinociceptive effects in a postoperative pain model in rats
Merlos, Manuel, Portillo-Salido, Enrique, Brenchat, Alex, Aubel, Bertrand, Buxens, Jordi, Fisas, Angels, Codony, Xavier, Romero, Luz, Zamanillo, Daniel, Vela, José Miguel
Published in European journal of pharmacology (15.08.2018)
Published in European journal of pharmacology (15.08.2018)
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Sigma-1 receptor antagonism as opioid adjuvant strategy: Enhancement of opioid antinociception without increasing adverse effects
Vidal-Torres, Alba, de la Puente, Beatriz, Rocasalbas, Maria, Touriño, Clara, Andreea Bura, Simona, Fernández-Pastor, Begoña, Romero, Luz, Codony, Xavier, Zamanillo, Daniel, Buschmann, Helmut, Merlos, Manuel, Manuel Baeyens, José, Maldonado, Rafael, Vela, José Miguel
Published in European journal of pharmacology (05.07.2013)
Published in European journal of pharmacology (05.07.2013)
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P033 DSS-induced colitis is attenuated in sigma-1 receptor knockout mice
Lόpez-Estévez, S., Aguilera, M., Gris, G., de la Puente, B., Codony, X., Zamanillo, D., Martínez, V.
Published in Journal of Crohn's and colitis (01.02.2017)
Published in Journal of Crohn's and colitis (01.02.2017)
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DOP088 Somatic and visceral hypersensitivity associated to acute intestinal inflammation are absent in sigma 1 receptor knockout mice
Lόpez-Estévez, S., Gris, G., de la Puente, B., Codony, X., Merlos, M., Martínez, V.
Published in Journal of Crohn's and colitis (01.02.2017)
Published in Journal of Crohn's and colitis (01.02.2017)
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Generation and phenotypic analysis of sigma receptor type I (σ1) knockout mice
Langa, Francina, Codony, Xavier, Tovar, Victoria, Lavado, Alfonso, Giménez, Estela, Cozar, Patricia, Cantero, Marta, Dordal, Albert, Hernández, Enric, Pérez, Raquel, Monroy, Xavier, Zamanillo, Daniel, Guitart, Xavier, Montoliu, Lluís
Published in The European journal of neuroscience (01.10.2003)
Published in The European journal of neuroscience (01.10.2003)
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Journal Article
Medicinal chemistry strategies to 5-HT sub(6) receptor ligands as potential cognitive enhancers and antiobesity agents
Holenz, J, Pauwels, P J, Diaz, J L, Merce, R, Codony, X, Buschmann, H
Published in Drug discovery today (01.04.2006)
Published in Drug discovery today (01.04.2006)
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Journal Article
E‐5842: A New Potent and Preferential Sigma Ligand. Preclinical Pharmacological Profile
Guitart, X., Codony, X., Ballarín, M., Dordal, A., Farré, A. J.
Published in CNS drug reviews (01.09.1998)
Published in CNS drug reviews (01.09.1998)
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Journal Article
Promising Novel 5-HT6 Receptor Ligands to Treat Obesity
P. J. Pauwels, A. Fisas, X. Codony, H. Buschmann
Published in Journal of Pharmacological Sciences (2006)
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Published in Journal of Pharmacological Sciences (2006)
Journal Article
Medicinal Chemistry approaches toward novel, selective 5-HT6 receptor ligands
J. Holenz, P. J. Pauwels, J. L. Diaz, R. Merce, X. Codony, H. Buschmann
Published in Journal of Pharmacological Sciences (2006)
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Published in Journal of Pharmacological Sciences (2006)
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Effect of E-6006 citrate upon schedule-induced polydipsia (SIP)
Fisas, M.A., Codony, X., Laloya, M., Farré, A.J., Guitart, X.
Published in European neuropsychopharmacology (01.10.2002)
Published in European neuropsychopharmacology (01.10.2002)
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Journal Article
Medicinal Chemistry Driven Approaches Toward Novel and Selective Serotonin 5-HT sub(6) Receptor Ligands
Holenz, J, Merce, R, Diaz, J L, Guitart, X, Codony, X, Dordal, A, Romero, G, Torrens, A, Mas, J, Andaluz, B, Hernandez, S, Monroy, X, Sanchez, E, Hernandez, E
Published in Journal of medicinal chemistry (24.03.2005)
Published in Journal of medicinal chemistry (24.03.2005)
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