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A Phase 1, Open‐Label, Pharmacokinetic Trial to Investigate Possible Drug‐Drug Interactions Between Clobazam, Stiripentol, or Valproate and Cannabidiol in Healthy Subjects
Morrison, Gilmour, Crockett, Julie, Blakey, Graham, Sommerville, Kenneth
Published in Clinical pharmacology in drug development (01.11.2019)
Published in Clinical pharmacology in drug development (01.11.2019)
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Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of the Oral NLRP3 Inflammasome Inhibitor ZYIL1: First‐in‐Human Phase 1 Studies (Single Ascending Dose and Multiple Ascending Dose)
Parmar, Deven V., Kansagra, Kevinkumar A., Momin, Taufik, Patel, Hardik B., Jansari, Gaurav A., Bhavsar, Jay, Shah, Chintan, Patel, Jayesh M., Ghoghari, Ashok, Barot, Ajay, Sharma, Bhavesh, Viswanathan, Kasinath, Patel, Harilal V., Jain, Mukul R.
Published in Clinical pharmacology in drug development (01.02.2023)
Published in Clinical pharmacology in drug development (01.02.2023)
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Pharmacokinetics, Pharmacodynamics, Safety, and Tolerability of Oral Venglustat in Healthy Volunteers
Peterschmitt, M. Judith, Crawford, Nigel P. S., Gaemers, Sebastiaan J. M., Ji, Allena J., Sharma, Jyoti, Pham, Theresa T.
Published in Clinical pharmacology in drug development (01.01.2021)
Published in Clinical pharmacology in drug development (01.01.2021)
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Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of the Novel Non–Bile Acid FXR Agonist Tropifexor (LJN452) in Healthy Volunteers
Badman, Michael K., Chen, Jin, Desai, Sachin, Vaidya, Soniya, Neelakantham, Srikanth, Zhang, Jie, Gan, Lu, Danis, Kate, Laffitte, Bryan, Klickstein, Lloyd B.
Published in Clinical pharmacology in drug development (01.04.2020)
Published in Clinical pharmacology in drug development (01.04.2020)
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A Phase 1 Randomized, Double‐Blind, Placebo‐Controlled Trial to Assess the Safety, Tolerability, and Pharmacokinetics of a Respiratory Syncytial Virus Neutralizing Monoclonal Antibody MK‐1654 in Healthy Adults
Aliprantis, Antonios O., Wolford, Dennis, Caro, Luzelena, Maas, Brian M., Ma, Hua, Montgomery, Diana L., Sterling, Laura M., Hunt, Allen, Cox, Kara S., Vora, Kalpit A., Roadcap, Brad A., Railkar, Radha A., Lee, Andrew W., Stoch, S. Aubrey, Lai, Eseng
Published in Clinical pharmacology in drug development (01.05.2021)
Published in Clinical pharmacology in drug development (01.05.2021)
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Safety, Tolerability, and Pharmacokinetics of Single Ascending Doses of ELX‐02, a Potential Treatment for Genetic Disorders Caused by Nonsense Mutations, in Healthy Volunteers
Leubitz, Andi, Frydman‐Marom, Anat, Sharpe, Neal, Duzer, John, Campbell, Kathleen C.M., Vanhoutte, Frédéric
Published in Clinical pharmacology in drug development (01.11.2019)
Published in Clinical pharmacology in drug development (01.11.2019)
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Pharmacokinetics, Pharmacodynamics, Safety, and Tolerability of Dupilumab in Healthy Adult Subjects
Li, Zhaoyang, Radin, Allen, Li, Meng, Hamilton, Jennifer D., Kajiwara, Miyuki, Davis, John D., Takahashi, Yoshinori, Hasegawa, Setsuo, Ming, Jeffrey E., DiCioccio, A. Thomas, Li, Yongtao, Kovalenko, Pavel, Lu, Qiang, Ortemann‐Renon, Catherine, Ardeleanu, Marius, Swanson, Brian N.
Published in Clinical pharmacology in drug development (01.08.2020)
Published in Clinical pharmacology in drug development (01.08.2020)
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Pharmacokinetic Assessment of Drug‐Drug Interactions of Isavuconazole With the Immunosuppressants Cyclosporine, Mycophenolic Acid, Prednisolone, Sirolimus, and Tacrolimus in Healthy Adults
Groll, Andreas H., Desai, Amit, Han, David, Howieson, Corrie, Kato, Kota, Akhtar, Shahzad, Kowalski, Donna, Lademacher, Christopher, Lewis, William, Pearlman, Helene, Mandarino, Debra, Yamazaki, Takao, Townsend, Robert
Published in Clinical pharmacology in drug development (01.01.2017)
Published in Clinical pharmacology in drug development (01.01.2017)
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Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of a Liver‐Targeting Acetyl‐CoA Carboxylase Inhibitor (PF‐05221304): A Three‐Part Randomized Phase 1 Study
Bergman, Arthur, Carvajal‐Gonzalez, Santos, Tarabar, Sanela, Saxena, Aditi R., Esler, William P., Amin, Neeta B.
Published in Clinical pharmacology in drug development (01.05.2020)
Published in Clinical pharmacology in drug development (01.05.2020)
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Pharmacokinetics and Safety of Letermovir Coadministered With Cyclosporine A or Tacrolimus in Healthy Subjects
Kropeit, Dirk, Richter, Oliver, Stobernack, Hans‐Peter, Rübsamen‐Schaeff, Helga, Zimmermann, Holger
Published in Clinical pharmacology in drug development (01.01.2018)
Published in Clinical pharmacology in drug development (01.01.2018)
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Pharmacokinetics, Pharmacodynamics, and Safety of the Dual Orexin Receptor Antagonist Lemborexant: Findings From Single‐Dose and Multiple‐Ascending‐Dose Phase 1 Studies in Healthy Adults
Landry, Ishani, Nakai, Kenya, Ferry, Jim, Aluri, Jagadeesh, Hall, Nancy, Lalovic, Bojan, Moline, Margaret L.
Published in Clinical pharmacology in drug development (01.02.2021)
Published in Clinical pharmacology in drug development (01.02.2021)
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Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of ZY‐IL1 in Three Patients with Cryopyrin‐Associated Periodic Syndromes
Hissaria, Pravin, Kansagra, Kevinkumar, Patel, Hardik, Momin, Taufik, Ghoghari, Ashok, Patel, Harilal, Sharma, Bhavesh
Published in Clinical pharmacology in drug development (01.02.2024)
Published in Clinical pharmacology in drug development (01.02.2024)
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Pharmacokinetic Similarity of ABP 654, an Ustekinumab Biosimilar Candidate: Results from a Randomized, Double‐blind Study in Healthy Subjects
Chow, Vincent, Mytych, Daniel T., Das, Shyamal, Franklin, Janet
Published in Clinical pharmacology in drug development (01.09.2023)
Published in Clinical pharmacology in drug development (01.09.2023)
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Safety, Tolerability, and Pharmacokinetics of ARC‐520 Injection, an RNA Interference‐Based Therapeutic for the Treatment of Chronic Hepatitis B Virus Infection, in Healthy Volunteers
Schluep, Thomas, Lickliter, Jason, Hamilton, James, Lewis, David L., Lai, Ching‐Lung, Lau, Johnson YN, Locarnini, Stephen A., Gish, Robert G., Given, Bruce D.
Published in Clinical pharmacology in drug development (01.07.2017)
Published in Clinical pharmacology in drug development (01.07.2017)
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Pharmacokinetic Evaluation of CYP3A4‐Mediated Drug‐Drug Interactions of Isavuconazole With Rifampin, Ketoconazole, Midazolam, and Ethinyl Estradiol/Norethindrone in Healthy Adults
Townsend, Robert, Dietz, Albert, Hale, Christine, Akhtar, Shahzad, Kowalski, Donna, Lademacher, Christopher, Lasseter, Kenneth, Pearlman, Helene, Rammelsberg, Diane, Schmitt‐Hoffmann, Anne, Yamazaki, Takao, Desai, Amit
Published in Clinical pharmacology in drug development (01.01.2017)
Published in Clinical pharmacology in drug development (01.01.2017)
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First‐in‐Human Study of AG10, a Novel, Oral, Specific, Selective, and Potent Transthyretin Stabilizer for the Treatment of Transthyretin Amyloidosis: A Phase 1 Safety, Tolerability, Pharmacokinetic, and Pharmacodynamic Study in Healthy Adult Volunteers
Fox, Jonathan C., Hellawell, Jennifer L., Rao, Satish, O'Reilly, Terry, Lumpkin, Rick, Jernelius, Jesper, Gretler, Daniel, Sinha, Uma
Published in Clinical pharmacology in drug development (01.01.2020)
Published in Clinical pharmacology in drug development (01.01.2020)
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