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Safety, Pharmacokinetics, and Pharmacodynamics of Etavopivat (FT‐4202), an Allosteric Activator of Pyruvate Kinase‐R, in Healthy Adults: A Randomized, Placebo‐Controlled, Double‐Blind, First‐in‐Human Phase 1 Trial
Forsyth, Sanjeev, Schroeder, Patricia, Geib, James, Vrishabhendra, Leela, Konstantinidis, Diamantis G., LaSalvia, Kari, Ribadeneira, Maria D., Wu, Eric, Kelly, Patrick, Kalfa, Theodosia A.
Published in Clinical pharmacology in drug development (01.05.2022)
Published in Clinical pharmacology in drug development (01.05.2022)
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Single‐Dose Pharmacokinetics and Safety of Atogepant in Adults With Hepatic Impairment: Results From an Open‐Label, Phase 1 Trial
Boinpally, Ramesh, Jakate, Abhijeet, Butler, Matthew, Borbridge, Lisa, Periclou, Antonia
Published in Clinical pharmacology in drug development (01.07.2021)
Published in Clinical pharmacology in drug development (01.07.2021)
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A Phase 1 Randomized Study to Evaluate the Safety, Tolerability, and Pharmacokinetics of Single Escalating Oral Doses of Dordaviprone and the Effects of Food on the Bioavailability of Dordaviprone in Healthy Adult Subjects
Faison, Shamia L., Batonga, Joelle, Arumugham, Thangam, Bartkus, Angela, Morrison, Marion, Mullin, Mark J., Tippin, Tim, Naderer, Odin
Published in Clinical pharmacology in drug development (01.05.2025)
Published in Clinical pharmacology in drug development (01.05.2025)
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Bioequivalence and Relative Bioavailability Studies to Assess a New Acalabrutinib Formulation That Enables Coadministration With Proton‐Pump Inhibitors
Sharma, Shringi, Pepin, Xavier, Burri, Harini, Zheng, Lianqing, Kuptsova‐Clarkson, Nataliya, Jong, Anouk, Yu, Ting, MacArthur, Holly L., Majewski, Michal, Byrd, John C., Furman, Richard R., Ware, Joseph A., Mann, James, Ramies, David, Munugalavadla, Veerendra, Sheridan, Louise, Tomkinson, Helen
Published in Clinical pharmacology in drug development (01.11.2022)
Published in Clinical pharmacology in drug development (01.11.2022)
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Safety, Pharmacokinetics, and Pharmacodynamics of Etrasimod: Single and Multiple Ascending Dose Studies in Healthy Adults
Lee, Caroline A., Schreiber, Stefan, Bressler, Brian, Adams, John W., Oh, Dooman Alexander, Tang, Yong Q., Zhang, Jinkun, Komori, Heather Kiyomi, Grundy, John S.
Published in Clinical pharmacology in drug development (01.05.2024)
Published in Clinical pharmacology in drug development (01.05.2024)
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Evaluation of Potential Effects of CYP3A Inhibition and CYP3A Induction on the Pharmacokinetics of Fruquintinib in Healthy Subjects
Gonzalez, Martha, Yang, Zhao, Schelman, William R, Zhou, Xiaofei, Gupta, Neeraj, Chien, Caly
Published in Clinical pharmacology in drug development (01.08.2025)
Published in Clinical pharmacology in drug development (01.08.2025)
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Pharmacokinetic Drug‐Drug Interaction With Coadministration of Cannabidiol and Everolimus in a Phase 1 Healthy Volunteer Trial
Wray, Louise, Berwaerts, Joris, Critchley, David, Hyland, Kerry, Chen, Cuiping, Thai, Ching, Tayo, Bola
Published in Clinical pharmacology in drug development (01.09.2023)
Published in Clinical pharmacology in drug development (01.09.2023)
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A Phase 1 Study to Evaluate the Absorption, Metabolism, and Disposition of Dordaviprone in Healthy Adult Participants
Teffera, Yohannes, Tippin, Tim, Bartkus, Angela, de Castro, Francine A, Faison, Shamia L, Morrison, Marion, Mullin, Mark J, Naderer, Odin
Published in Clinical pharmacology in drug development (01.07.2025)
Published in Clinical pharmacology in drug development (01.07.2025)
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Disposition and Mass Balance of Etrasimod in Healthy Subjects and In Vitro Determination of the Enzymes Responsible for Its Oxidative Metabolism
Lee, Caroline A., Oh, D. Alexander, Tang, Yong, Yi, Ping, Bashir, Mohammad, English, Stephen, Croft, Marie, Blackburn, Anthony, Bloom, Steve, Gilder, Kye, Grundy, John S.
Published in Clinical pharmacology in drug development (01.06.2023)
Published in Clinical pharmacology in drug development (01.06.2023)
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Phase 1 Clinical Trial of PPMX‐T003, a Novel Human Monoclonal Antibody Specific for Transferrin Receptor 1, to Evaluate Its Safety, Pharmacokinetics, and Pharmacodynamics
Ogama, Yoichiro, Kumagai, Yuji, Komatsu, Norio, Araki, Marito, Masubuchi, Nami, Akiyoshi, Hiroko, Matsuura, Tadashi, Kirisako, Hiromi, Kyoya, Akiko, Nomura, Fumiko, Ohira, Yuta, Yokokawa, Takuya, Yamamoto, Yukiya
Published in Clinical pharmacology in drug development (01.06.2023)
Published in Clinical pharmacology in drug development (01.06.2023)
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Enhanced Bioavailability and Reduced Variability of Dasatinib and Sorafenib with a Novel Amorphous Solid Dispersion Technology Platform
Lennernäs, Hans, Brisander, Magnus, Liljebris, Charlotta, Jesson, Gérald, Andersson, Per
Published in Clinical pharmacology in drug development (01.09.2024)
Published in Clinical pharmacology in drug development (01.09.2024)
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Single‐Dose Pharmacokinetics of Oral Cannabidiol Following Administration of PTL101: A New Formulation Based on Gelatin Matrix Pellets Technology
Atsmon, Jacob, Heffetz, Daphna, Deutsch, Lisa, Deutsch, Frederic, Sacks, Hagit
Published in Clinical pharmacology in drug development (01.09.2018)
Published in Clinical pharmacology in drug development (01.09.2018)
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A Phase 1 Open‐Label, Fixed‐Sequence Pharmacokinetic Drug Interaction Trial to Investigate the Effect of Cannabidiol on the CYP1A2 Probe Caffeine in Healthy Subjects
Thai, Ching, Tayo, Bola, Critchley, David
Published in Clinical pharmacology in drug development (01.11.2021)
Published in Clinical pharmacology in drug development (01.11.2021)
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A Randomized Phase 1 Study Evaluating Pharmacokinetics, Safety, and Tolerability of a High‐Concentration, Long‐Acting Cabotegravir Formulation in Adults Without HIV
Han, Kelong, Benn, Paul, Sievers, Jörg, Dorey, David, Warwick‐Sanders, Michael, Hareedy, Randa, Harkness, Louise, Leemereise, Claudia, Offenbecker, Kjersten, Donatti, Christina, Brimhall, Darin B., Schwabe, Christian, Boyle, Craig, Hassman, Michael A., Knowles, Steve, D'Amico, Ronald, Spreen, William R.
Published in Clinical pharmacology in drug development (01.07.2025)
Published in Clinical pharmacology in drug development (01.07.2025)
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New Ustekinumab Biosimilar Candidate FYB202: Pharmacokinetic Equivalence Demonstrated in a Randomized, Double‐Blind, Parallel‐Group, Single‐Dose Trial in Healthy Subjects
Balser, Sigrid, Nopora, Katrin, Körner, Juliane, Wedemeyer, Ralph‐Steven, Anschütz, Maria, Schug, Barbara
Published in Clinical pharmacology in drug development (01.12.2024)
Published in Clinical pharmacology in drug development (01.12.2024)
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Pharmacokinetics of the Akt Serine/Threonine Protein Kinase Inhibitor, Capivasertib, Administered to Healthy Volunteers in the Presence and Absence of the CYP3A4 Inhibitor Itraconazole
Miller, Claire, Sommavilla, Roberto, Barry, Simon T., Eberlein, Cath, Morris, Thomas, Wadsworth, Ian, Cullberg, Marie
Published in Clinical pharmacology in drug development (01.09.2023)
Published in Clinical pharmacology in drug development (01.09.2023)
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Safety, Tolerability, and Pharmacokinetics of IMU‐935, a Novel Inverse Agonist of Retinoic Acid Receptor–Related Orphan Nuclear Receptor γt: Results From a Double‐Blind, Placebo‐Controlled, First‐in‐Human Phase 1 Study
Polasek, Thomas M., Leelasena, Indika, Betscheider, Irina, Marolt, Marija, Kohlhof, Hella, Vitt, Daniel, Fliegert, Frank, Muehler, Andreas R.
Published in Clinical pharmacology in drug development (01.05.2023)
Published in Clinical pharmacology in drug development (01.05.2023)
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