Search Results - "Clausen, Rasmus P" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

α4βδ GABAA receptors are high-affinity targets for γ-hydroxybutyric acid (GHB)

α4βδ GABAA receptors are high-affinity targets for γ-hydroxybutyric acid (GHB)

by Absalom, Nathan, Eghorn, Laura F, Villumsen, Inge S, Karim, Nasiara, Bay, Tina, Olsen, Jesper V, Knudsen, Gitte M, Bräuner-Osborne, Hans, Frølund, Bente, Clausen, Rasmus P, Chebib, Mary, Wellendorph, Petrine
Published in Proceedings of the National Academy of Sciences - PNAS (14.08.2012)

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Pharmacological Characterization of a Betaine/GABA Transporter 1 (BGT1) Inhibitor Displaying an Unusual Biphasic Inhibition Profile and Anti-seizure Effects

by Lie, Maria E. K., Kickinger, Stefanie, Skovgaard-Petersen, Jonas, Ecker, Gerhard F., Clausen, Rasmus P., Schousboe, Arne, White, H. Steve, Wellendorph, Petrine
Published in Neurochemical research (01.07.2020)

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Synaptic and extrasynaptic GABA transporters as targets for anti-epileptic drugs

Synaptic and extrasynaptic GABA transporters as targets for anti-epileptic drugs

by Madsen, Karsten K, Clausen, Rasmus P, Larsson, Orla M, Krogsgaard-Larsen, Povl, Schousboe, Arne, Steve White, H
Published in Journal of neurochemistry (01.05.2009)

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In Vitro and In Vivo Evidence for Active Brain Uptake of the GHB Analog HOCPCA by the Monocarboxylate Transporter Subtype 1

In Vitro and In Vivo Evidence for Active Brain Uptake of the GHB Analog HOCPCA by the Monocarboxylate Transporter Subtype 1

by Thiesen, Louise, Kehler, Jan, Clausen, Rasmus P, Frølund, Bente, Bundgaard, Christoffer, Wellendorph, Petrine
Published in The Journal of pharmacology and experimental therapeutics (01.08.2015)

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Structure activity relationship of selective GABA uptake inhibitors

Structure activity relationship of selective GABA uptake inhibitors

by Vogensen, Stine B., Jørgensen, Lars, Madsen, Karsten K., Jurik, Andreas, Borkar, Nrupa, Rosatelli, Emiliano, Nielsen, Birgitte, Ecker, Gerhard F., Schousboe, Arne, Clausen, Rasmus P.
Published in Bioorganic & medicinal chemistry (15.05.2015)

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Inhibition of GABA transporters fails to afford significant protection following focal cerebral ischemia

Inhibition of GABA transporters fails to afford significant protection following focal cerebral ischemia

by Lie, Maria EK, Gowing, Emma K, Clausen, Rasmus P, Wellendorph, Petrine, Clarkson, Andrew N
Published in Journal of cerebral blood flow and metabolism (01.01.2018)

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Pharmacology and Structural Analysis of Ligand Binding to the Orthosteric Site of Glutamate-Like GluD2 Receptors

Pharmacology and Structural Analysis of Ligand Binding to the Orthosteric Site of Glutamate-Like GluD2 Receptors

by Kristensen, Anders S, Hansen, Kasper B, Naur, Peter, Olsen, Lars, Kurtkaya, Natalie L, Dravid, Shashank M, Kvist, Trine, Yi, Feng, Pøhlsgaard, Jacob, Clausen, Rasmus P, Gajhede, Michael, Kastrup, Jette S, Traynelis, Stephen F
Published in Molecular pharmacology (01.02.2016)

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Discovery of ( R )-2-amino-3-triazolpropanoic acid derivatives as NMDA receptor glycine site agonists with GluN2 subunit-specific activity

Discovery of ( R )-2-amino-3-triazolpropanoic acid derivatives as NMDA receptor glycine site agonists with GluN2 subunit-specific activity

by Zhao, Fabao, Mazis, Georgios, Yi, Feng, Lotti, James S, Layeux, Michael S, Schultz, Eric P, Bunch, Lennart, Hansen, Kasper B, Clausen, Rasmus P
Published in Frontiers in chemistry (17.11.2022)

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Does increasing the ratio of AMPA-to-NMDA receptor mediated neurotransmission engender antidepressant action? Studies in the mouse forced swim and tail suspension tests

Does increasing the ratio of AMPA-to-NMDA receptor mediated neurotransmission engender antidepressant action? Studies in the mouse forced swim and tail suspension tests

by Andreasen, Jesper T., Gynther, Mikko, Rygaard, Allan, Bøgelund, Trine, Nielsen, Simon D., Clausen, Rasmus P., Mogensen, Jesper, Pickering, Darryl S.
Published in Neuroscience letters (24.06.2013)

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Subunit-Specific Agonist Activity at NR2A-, NR2B-, NR2C-, and NR2D-Containing N-Methyl-d-aspartate Glutamate Receptors

Subunit-Specific Agonist Activity at NR2A-, NR2B-, NR2C-, and NR2D-Containing N-Methyl-d-aspartate Glutamate Receptors

by Erreger, Kevin, Geballe, Matthew T, Kristensen, Anders, Chen, Philip E, Hansen, Kasper B, Lee, C Justin, Yuan, Hongjie, Le, Phuong, Lyuboslavsky, Polina N, Micale, Nicola, Jørgensen, Lars, Clausen, Rasmus P, Wyllie, David J A, Snyder, James P, Traynelis, Stephen F
Published in Molecular pharmacology (01.10.2007)

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Substrate- and Cofactor-independent Inhibition of Histone Demethylase KDM4C

Substrate- and Cofactor-independent Inhibition of Histone Demethylase KDM4C

by Leurs, Ulrike, Lohse, Brian, Rand, Kasper D, Ming, Shonoi, Riise, Erik S, Cole, Philip A, Kristensen, Jesper L, Clausen, Rasmus P
Published in ACS chemical biology (19.09.2014)

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Astrocytic GABA Transporters: Pharmacological Properties and Targets for Antiepileptic Drugs

Astrocytic GABA Transporters: Pharmacological Properties and Targets for Antiepileptic Drugs

by Schousboe, Arne, Wellendorph, Petrine, Frølund, Bente, Clausen, Rasmus P., Krogsgaard-Larsen, Povl
Published in Advances in neurobiology (01.01.2017)

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Book Chapter Journal Article

Targeting Histone Lysine Demethylases by Truncating the Histone 3 Tail to Obtain Selective Substrate-Based Inhibitors

Targeting Histone Lysine Demethylases by Truncating the Histone 3 Tail to Obtain Selective Substrate-Based Inhibitors

by Lohse, Brian, Nielsen, Anders L., Kristensen, Jan B. L., Helgstrand, Charlotte, Cloos, Paul A. C., Olsen, Lars, Gajhede, Michael, Clausen, Rasmus P., Kristensen, Jesper L.
Published in Angewandte Chemie (International ed.) (19.09.2011)

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Posttranslational modifications of the histone 3 tail and their impact on the activity of histone lysine demethylases in vitro

Posttranslational modifications of the histone 3 tail and their impact on the activity of histone lysine demethylases in vitro

by Lohse, Brian, Helgstrand, Charlotte, Kristensen, Jan B L, Leurs, Ulrike, Cloos, Paul A C, Kristensen, Jesper L, Clausen, Rasmus P
Published in PloS one (02.07.2013)

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Identification of the First Highly Subtype-Selective Inhibitor of Human GABA Transporter GAT3

Identification of the First Highly Subtype-Selective Inhibitor of Human GABA Transporter GAT3

by Damgaard, Maria, Al-Khawaja, Anas, Vogensen, Stine B, Jurik, Andreas, Sijm, Maarten, Lie, Maria E. K, Bæk, Mathias I, Rosenthal, Emil, Jensen, Anders A, Ecker, Gerhard F, Frølund, Bente, Wellendorph, Petrine, Clausen, Rasmus P
Published in ACS chemical neuroscience (16.09.2015)

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Journal Article

Synthesis and Characterisation of Substrate-Based Peptides as Inhibitors of Histone Demethylase KDM4C

Synthesis and Characterisation of Substrate-Based Peptides as Inhibitors of Histone Demethylase KDM4C

by Nielsen, Simon D, Leurs, Ulrike, Bergner, Magnus, Barris, Silvia A, Devkota, Kanchan, Meyer, Kamilla, Iaria, Daniella, McCaughan, Jack, Lohse, Brian, Kristensen, Jesper L, Clausen, Rasmus P
Published in Protein and peptide letters (01.01.2016)

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Journal Article

Derivatives of (R)‑3-(5-Furanyl)carboxamido-2-aminopropanoic Acid as Potent NMDA Receptor Glycine Site Agonists with GluN2 Subunit-Specific Activity

Derivatives of (R)‑3-(5-Furanyl)carboxamido-2-aminopropanoic Acid as Potent NMDA Receptor Glycine Site Agonists with GluN2 Subunit-Specific Activity

by Zhao, Fabao, Atxabal, Unai, Mariottini, Sofia, Yi, Feng, Lotti, James S, Rouzbeh, Nirvan, Liu, Na, Bunch, Lennart, Hansen, Kasper B, Clausen, Rasmus P
Published in Journal of medicinal chemistry (13.01.2022)

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In vitro ADME characterization of a very potent 3-acylamino-2-aminopropionic acid-derived GluN2C-NMDA receptor agonist and its ester prodrugs

In vitro ADME characterization of a very potent 3-acylamino-2-aminopropionic acid-derived GluN2C-NMDA receptor agonist and its ester prodrugs

by Bechthold, Elena, Grey, Lucie, Diamant, Emil, Schmidt, Judith, Steigerwald, Ruben, Zhao, Fabao, Hansen, Kasper B., Bunch, Lennart, Clausen, Rasmus P., Wünsch, Bernhard
Published in Biological chemistry (28.03.2023)

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Journal Article

Inhibition of the betaine-GABA transporter (mGAT2/BGT-1) modulates spontaneous electrographic bursting in the medial entorhinal cortex (mEC)

Inhibition of the betaine-GABA transporter (mGAT2/BGT-1) modulates spontaneous electrographic bursting in the medial entorhinal cortex (mEC)

by Smith, Misty D, Saunders, Gerald W, Clausen, Rasmus P, Frǿlund, Bente, Krogsgaard-Larsen, Povl, Larsson, Orla M, Schousboe, Arne, Wilcox, Karen S, White, H. Steve
Published in Epilepsy research (01.03.2008)

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Identification of AICP as a GluN2C-Selective N -Methyl-d-Aspartate Receptor Superagonist at the GluN1 Glycine Site

Identification of AICP as a GluN2C-Selective N -Methyl-d-Aspartate Receptor Superagonist at the GluN1 Glycine Site

by Jessen, Maja, Frederiksen, Kristen, Yi, Feng, Clausen, Rasmus P, Hansen, Kasper B, Bräuner-Osborne, Hans, Kilburn, Paul, Damholt, Anders
Published in Molecular pharmacology (01.08.2017)

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