Search Results - "Classon, Bjorn" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Selective Cathepsin S Inhibition with MIV-247 Attenuates Mechanical Allodynia and Enhances the Antiallodynic Effects of Gabapentin and Pregabalin in a Mouse Model of Neuropathic Pain

Selective Cathepsin S Inhibition with MIV-247 Attenuates Mechanical Allodynia and Enhances the Antiallodynic Effects of Gabapentin and Pregabalin in a Mouse Model of Neuropathic Pain

by Hewitt, Ellen, Pitcher, Thomas, Rizoska, Biljana, Tunblad, Karin, Henderson, Ian, Sahlberg, Britt-Louise, Grabowska, Urszula, Classon, Björn, Edenius, Charlotte, Malcangio, Marzia, Lindström, Erik
Published in The Journal of pharmacology and experimental therapeutics (01.09.2016)

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A one-pot, solid-phase synthesis of secondary amines from reactive alkyl halides and an alkyl azide

A one-pot, solid-phase synthesis of secondary amines from reactive alkyl halides and an alkyl azide

by Ayesa, Susana, Samuelsson, Bertil, Classon, Bjorn
Published in Synlett (03.01.2008)

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Solid-phase parallel synthesis and SAR of 4-amidofuran-3-one inhibitors of cathepsin S: Effect of sulfonamides P3 substituents on potency and selectivity

Solid-phase parallel synthesis and SAR of 4-amidofuran-3-one inhibitors of cathepsin S: Effect of sulfonamides P3 substituents on potency and selectivity

by Ayesa, Susana, Lindquist, Charlotta, Agback, Tatiana, Benkestock, Kurt, Classon, Björn, Henderson, Ian, Hewitt, Ellen, Jansson, Katarina, Kallin, Anders, Sheppard, Dave, Samuelsson, Bertil
Published in Bioorganic & medicinal chemistry (01.02.2009)

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Discovery of novel, potent and bioavailable proline-urea based macrocyclic HCV NS3/4A protease inhibitors

Discovery of novel, potent and bioavailable proline-urea based macrocyclic HCV NS3/4A protease inhibitors

by VENDEVILLE, Sandrine, NILSSON, Magnus, ENEROTH, Anders, WIKSTROM, Kristina, VRANG, Lotta, EDLUND, Michael, LINDSTRÖM, Stefan, VAN DE VREKEN, Wim, MCGOWAN, David, TAHRI, Abdellah, LILI HU, LENZ, Oliver, DE KOCK, Herman, DELOUVROY, Frederic, VAN DOOREN, Marleen, KINDERMANS, Natalie, SURLERAUX, Dominique, WIGERINCK, Piet, ROSENQUIST, Asa, SAMUELSSON, Bertil, SIMMENA, Kenneth, RABOISSON, Pierre, LINA, Tse-I, ANTONOV, Dmitry, CLASSON, Björn, AYESA, Susana, IVANOV, Vladimir, JOHANSSON, Per-Ola, KAHNBERG, Pia
Published in Bioorganic & medicinal chemistry (01.12.2008)

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Characterization of a set of HIV-1 protease inhibitors using binding kinetics data from a biosensor-based screen

Characterization of a set of HIV-1 protease inhibitors using binding kinetics data from a biosensor-based screen

by Hämäläinen, M D, Markgren, P O, Schaal, W, Karlén, A, Classon, B, Vrang, L, Samuelsson, B, Hallberg, A, Danielson, U H
Published in Journal of biomolecular screening (01.10.2000)

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Synthesis of carbocyclic 2′3′-dideoxy-2′-fluoro-3′-C-hydroxymethyl nucleoside analogues as potential inhibitors of HIV and HSV

Synthesis of carbocyclic 2′3′-dideoxy-2′-fluoro-3′-C-hydroxymethyl nucleoside analogues as potential inhibitors of HIV and HSV

by Wachtmeister, Johanna, Björn, Classon, Bertil, Samuelsson, Kvarnström, Ingemar
Published in Tetrahedron (03.02.1997)

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Impact of the Central Hydroxyl Groups on the Activity of Symmetrical HIV-1 Protease Inhibitors Derived From l-Mannaric Acid

Impact of the Central Hydroxyl Groups on the Activity of Symmetrical HIV-1 Protease Inhibitors Derived From l-Mannaric Acid

by Wachtmeister, Johanna, Mühlman, Anna, Classon, Björn, Kvarnström, Ingemar, Hallberg, Anders, Samuelsson, Bertil
Published in Tetrahedron (12.05.2000)

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Synthesis of [4,5-Bis(hydroxymethyl)-1,3-dioxolan-2-yl]nucleosides as Potential Inhibitors of HIV

Synthesis of [4,5-Bis(hydroxymethyl)-1,3-dioxolan-2-yl]nucleosides as Potential Inhibitors of HIV

by Brånalt, Jonas, Kvarnström, Ingemar, Classon, Björn, Samuelsson, Bertil
Published in Journal of organic chemistry (31.05.1996)

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Abstract 5101: Defining exposure-PD and efficacy relationships with the novel liver-targeting nucleotide prodrug MIV-818 for the treatment of liver cancers

Abstract 5101: Defining exposure-PD and efficacy relationships with the novel liver-targeting nucleotide prodrug MIV-818 for the treatment of liver cancers

by Albertella, Mark, Rizoska, Biljana, Kyle, Alastair, Minchinton, Andrew, Linqvist, Annelie, Juric, Sanja, Sedig, Susanne, Tunblad, Karin, Öberg, Fredrik, Classon, Björn, Eneroth, Anders, Öhd, John, Bethell, Richard
Published in Cancer research (Chicago, Ill.) (01.07.2017)

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Design and Synthesis of Potent C2-Symmetric Diol-Based HIV-1 Protease Inhibitors: Effects of Fluoro Substitution

Design and Synthesis of Potent C2-Symmetric Diol-Based HIV-1 Protease Inhibitors: Effects of Fluoro Substitution

by PYRING, David, LINDBERG, Jimmy, ROSENQUIST, Åsa, ZUCCARELLO, Guido, KVARNSTRöM, Ingemar, ZHANG, Hong, VRANG, Lotta, UNGE, Torsten, CLASSON, Bjorn, HALLBERG, Anders, SAMUELSSON, Bertil
Published in Journal of medicinal chemistry (13.09.2001)

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Design and Synthesis of Potent C 2-Symmetric Diol-Based HIV-1 Protease Inhibitors: Effects of Fluoro Substitution

Design and Synthesis of Potent C 2-Symmetric Diol-Based HIV-1 Protease Inhibitors: Effects of Fluoro Substitution

by Pyring, David, Lindberg, Jimmy, Rosenquist, Åsa, Zuccarello, Guido, Kvarnström, Ingemar, Zhang, Hong, Vrang, Lotta, Unge, Torsten, Classon, Bjorn, Hallberg, Anders, Samuelsson, Bertil
Published in Journal of medicinal chemistry (13.09.2001)

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Symmetric fluoro‐substituted diol‐based HIV protease inhibitors

Symmetric fluoro‐substituted diol‐based HIV protease inhibitors

by Lindberg, Jimmy, Pyring, David, Löwgren, Seved, Rosenquist, Åsa, Zuccarello, Guido, Kvarnström, Ingemar, Zhang, Hong, Vrang, Lotta, Classon, Björn, Hallberg, Anders, Samuelsson, Bertil, Unge, Torsten
Published in European journal of biochemistry (01.11.2004)

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Solid phase assisted synthesis of HIV-1 protease inhibitors. Expedient entry to unsymmetrical substitution of a C(2) symmetric template

Solid phase assisted synthesis of HIV-1 protease inhibitors. Expedient entry to unsymmetrical substitution of a C(2) symmetric template

by Oscarsson, Karin, Classon, Bjorn, Kvarnstrom, Ingemar, Hallberg, Anders, Samuelsson, Bertil
Published in Canadian journal of chemistry (01.06.2000)

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A novel route to olefins from vicinal diols

A novel route to olefins from vicinal diols

by Liu, Zhengchun, Classon, Bjoern, Samuelsson, Bertil
Published in Journal of organic chemistry (01.07.1990)

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Novel potent macrocyclic inhibitors of the hepatitis C virus NS3 protease: Use of cyclopentane and cyclopentene P2-motifs

Novel potent macrocyclic inhibitors of the hepatitis C virus NS3 protease: Use of cyclopentane and cyclopentene P2-motifs

by Bäck, Marcus, Johansson, Per-Ola, Wångsell, Fredrik, Thorstensson, Fredrik, Kvarnström, Ingemar, Ayesa, Susana, Wähling, Horst, Pelcman, Mikael, Jansson, Katarina, Lindström, Stefan, Wallberg, Hans, Classon, Björn, Rydergård, Christina, Vrang, Lotta, Hamelink, Elizabeth, Hallberg, Anders, Rosenquist, Åsa, Samuelsson, Bertil
Published in Bioorganic & medicinal chemistry (15.11.2007)

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Synthesis and Comparative Molecular Field Analysis (CoMFA) of Symmetric and Nonsymmetric Cyclic Sulfamide HIV-1 Protease Inhibitors

Synthesis and Comparative Molecular Field Analysis (CoMFA) of Symmetric and Nonsymmetric Cyclic Sulfamide HIV-1 Protease Inhibitors

by Schaal, Wesley, Karlsson, Anna, Ahlsén, Göran, Lindberg, Jimmy, Andersson, Hans O, Danielson, U. Helena, Classon, Björn, Unge, Torsten, Samuelsson, Bertil, Hultén, Johan, Hallberg, Anders, Karlén, Anders
Published in Journal of medicinal chemistry (18.01.2001)

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Cyclic HIV-1 Protease Inhibitors Derived from Mannitol: Synthesis, Inhibitory Potencies, and Computational Predictions of Binding Affinities

Cyclic HIV-1 Protease Inhibitors Derived from Mannitol: Synthesis, Inhibitory Potencies, and Computational Predictions of Binding Affinities

by Hultén, Johan, Bonham, Nicholas M, Nillroth, Ulrika, Hansson, Tomas, Zuccarello, Guido, Bouzide, Abderrahim, Åqvist, Johan, Classon, Björn, Danielson, U. Helena, Karlén, Anders, Kvarnström, Ingemar, Samuelsson, Bertil, Hallberg, Anders
Published in Journal of medicinal chemistry (14.03.1997)

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Design and Fast Synthesis of C-Terminal Duplicated Potent C2-Symmetric P1/P1‘-Modified HIV-1 Protease Inhibitors

Design and Fast Synthesis of C-Terminal Duplicated Potent C2-Symmetric P1/P1‘-Modified HIV-1 Protease Inhibitors

by ALTERMAN, Mathias, ANDERSSON, Hans O., GARG, Neeraj, AHLSéN, Göran, LöVGREN, Seved, CLASSON, Björn, DANIELSON, U. Helena, KVARNSTRöM, Ingmar, VRANG, Lotta, UNGE, Torsten, SAMUELSSON, Bertil, HALLBERG, Anders
Published in Journal of medicinal chemistry (23.09.1999)

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Design and Fast Synthesis of C-Terminal Duplicated Potent C 2-Symmetric P1/P1‘-Modified HIV-1 Protease Inhibitors

Design and Fast Synthesis of C-Terminal Duplicated Potent C 2-Symmetric P1/P1‘-Modified HIV-1 Protease Inhibitors

by Alterman, Mathias, Andersson, Hans O, Garg, Neeraj, Ahlsén, Göran, Lövgren, Seved, Classon, Björn, Danielson, U. Helena, Kvarnström, Ingmar, Vrang, Lotta, Unge, Torsten, Samuelsson, Bertil, Hallberg, Anders
Published in Journal of medicinal chemistry (23.09.1999)

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Synthesis of Potent C 2-Symmetric, Diol-Based HIV-1 Protease Inhibitors. Investigation of Thioalkyl and Thioaryl P1/P1‘ Substituents

Synthesis of Potent C 2-Symmetric, Diol-Based HIV-1 Protease Inhibitors. Investigation of Thioalkyl and Thioaryl P1/P1‘ Substituents

by Mühlman, Anna, Classon, Björn, Hallberg, Anders, Samuelsson, Bertil
Published in Journal of medicinal chemistry (11.10.2001)

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