New Caspase-1 inhibitor by scaffold hopping into bio-inspired 3D-fragment space
Brethon, Anne, Chantalat, Laurent, Christin, Olivier, Clary, Laurence, Fournier, Jean-François, Gastreich, Marcus, Harris, Craig S., Isabet, Tatiana, Pascau, Jonathan, Thoreau, Etienne, Roche, Didier, Rodeschini, Vincent
Published in Bioorganic & medicinal chemistry letters (15.12.2017)
Published in Bioorganic & medicinal chemistry letters (15.12.2017)
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Journal Article
A facile and rapid preparation of hydroxamic acids by hydroxylaminolysis using DBU as base
Beillard, Audrey, Bhurruth-Alcor, Yushma, Bouix-Peter, Claire, Bouquet, Karinne, Chambon, Sandrine, Clary, Laurence, Harris, Craig S., Millois, Corinne, Mouis, Grégoire, Ouvry, Gilles, Pierre, Romain, Reitz, Arnaud, Tomas, Loic
Published in Tetrahedron letters (18.05.2016)
Published in Tetrahedron letters (18.05.2016)
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Journal Article
An expedient synthesis of non-racemic N-alkylated pyrrolidin-2,5-diones and piperidin-2,6-diones as peptidomimetics
Brethon, Anne, Bouix-Peter, Claire, Clary, Laurence, Fournier, Jean-François, Harris, Craig S., Lardy, Claude, Roche, Didier, Rodeschini, Vincent, Talano, Sandrine
Published in Tetrahedron letters (28.12.2016)
Published in Tetrahedron letters (28.12.2016)
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Journal Article
An expedient synthesis of non-racemic N-alkylated pyrrolidin2,5-diones and piperidin-2,6-diones as peptidomimetics
Brethon, Anne, Bouix-Peter, Claire, Clary, Laurence, Fournier, Jean-Francois, Harris, Craig S., lardy, Claude, Roche, Didier, Rodeschini, Vincent, Talano, Sandrine
Published in Tetrahedron letters (28.12.2016)
Published in Tetrahedron letters (28.12.2016)
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Journal Article
Rational Drug Design of Topically Administered Caspase 1 Inhibitors for the Treatment of Inflammatory Acne
Fournier, Jean-François, Clary, Laurence, Chambon, Sandrine, Dumais, Laurence, Harris, Craig Steven, Millois, Corinne, Pierre, Romain, Talano, Sandrine, Thoreau, Étienne, Aubert, Jérome, Aurelly, Michèle, Bouix-Peter, Claire, Brethon, Anne, Chantalat, Laurent, Christin, Olivier, Comino, Catherine, El-Bazbouz, Ghizlane, Ghilini, Anne-Laurence, Isabet, Tatiana, Lardy, Claude, Luzy, Anne-Pascale, Mathieu, Céline, Mebrouk, Kenny, Orfila, Danielle, Pascau, Jonathan, Reverse, Kevin, Roche, Didier, Rodeschini, Vincent, Hennequin, Laurent François
Published in Journal of medicinal chemistry (10.05.2018)
Published in Journal of medicinal chemistry (10.05.2018)
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Journal Article
Synthesis and stability evaluation of novel peptidomimetic Caspase-1 inhibitors for topical application
Chambon, Sandrine, Talano, Sandrine, Millois, Corinne, Dumais, Laurence, Pierre, Romain, Tomas, Loic, Mathieu, Céline, Ghilini, Anne-Laurence, Vanthuyne, Nicolas, Reverse, Kevin, Brethon, Anne, Rodeschini, Vincent, Comino, Catherine, Mouis, Grégoire, El-Bazbouz, Ghizlane, Clary, Laurence, Fournier, Jean-François, Bouix-Peter, Claire, Harris, Craig S., Hennequin, Laurent F.
Published in Tetrahedron (13.09.2018)
Published in Tetrahedron (13.09.2018)
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Journal Article
N-3 alkylation of uracils with unprotected amino alcohols using the Mitsunobu reaction
Lafitte, Guillaume, Beillard, Audrey, Chambon, Sandrine, Soulet, Catherine, Dumais, Laurence, Mouis, Grégoire, Fournier, Jean-François, Clary, Laurence, Bouix-Peter, Claire, Tomas, Loic, Harris, Craig S.
Published in Tetrahedron letters (17.01.2018)
Published in Tetrahedron letters (17.01.2018)
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Journal Article
신규한 MTOR 저해제 화합물
OUVRY GILLES, THOREAU ETIENNE, CLARY LAURENCE, FOURNIER JEAN FRANCOIS, BHURRUTH ALCOR YUSHMA, TOMAS LOIC
Year of Publication 01.09.2020
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Year of Publication 01.09.2020
Patent
MTOR 저해제 화합물
OUVRY GILLES, THOREAU ETIENNE, CLARY LAURENCE, FOURNIER JEAN FRANCOIS, BHURRUTH ALCOR YUSHMA, TOMAS LOIC
Year of Publication 01.09.2020
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Year of Publication 01.09.2020
Patent
Impact of Minor Structural Modifications on Properties of a Series of mTOR Inhibitors
Ouvry, Gilles, Clary, Laurence, Tomas, Loïc, Aurelly, Michèle, Bonnary, Laetitia, Borde, Emilie, Bouix-Peter, Claire, Chantalat, Laurent, Defoin-Platel, Claire, Deret, Sophie, Forissier, Mathieu, Harris, Craig S, Isabet, Tatiana, Lamy, Laurent, Luzy, Anne-Pascale, Pascau, Jonathan, Soulet, Catherine, Taddei, Alessandro, Taquet, Nathalie, Thoreau, Etienne, Varvier, Emeric, Vial, Emmanuel, Hennequin, Laurent F
Published in ACS medicinal chemistry letters (14.11.2019)
Published in ACS medicinal chemistry letters (14.11.2019)
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Journal Article
An efficient multi-component synthesis of N-1-alkylated 5-nitrouracils from α-amino acids
Boiteau, Jean-Guy, Bouix-Peter, Claire, Chambon, Sandrine, Clary, Laurence, Daver, Sebastien, Dumais, Laurence, Fournier, Jean-François, Harris, Craig S., Mebrouk, Kenny, Millois, Corinne, Pierre, Romain, Rodeville, Nicolas, Talano, Sandrine, Tomas, Loïc
Published in Tetrahedron letters (01.06.2016)
Published in Tetrahedron letters (01.06.2016)
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Journal Article