Corticotropin-Releasing Hormone Receptor Antagonists: Framework Design and Synthesis Guided by Ligand Conformational Studies
Hodge, C. Nicholas, Aldrich, Paul E, Wasserman, Zelda R, Fernandez, Christina H, Nemeth, Gregory A, Arvanitis, Argyrios, Cheeseman, Robert S, Chorvat, Robert J, Ciganek, Engelbert, Christos, Thomas E, Gilligan, Paul J, Krenitsky, Paul, Scholfield, Everett, Strucely, Philip
Published in Journal of medicinal chemistry (11.03.1999)
Published in Journal of medicinal chemistry (11.03.1999)
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Studies on New Acidic Azoles as Glucose-Lowering Agents in Obese, Diabetic db/db Mice
Kees, Kenneth L, Caggiano, Thomas J, Steiner, Kurt E, Fitzgerald, John J, Kates, Michael J, Christos, Thomas E, Kulishoff, John M, Moore, Robin D, McCaleb, Michael L
Published in Journal of medicinal chemistry (01.02.1995)
Published in Journal of medicinal chemistry (01.02.1995)
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Synthesis of (−)-Fumagillin
Taber, Douglass F, Christos, Thomas E
Published in Journal of the American Chemical Society (16.06.1999)
Published in Journal of the American Chemical Society (16.06.1999)
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Non-Peptide Corticotropin-Releasing Hormone Antagonists: Syntheses and Structure−Activity Relationships of 2-Anilinopyrimidines and -triazines
Arvanitis, Argyrios G, Gilligan, Paul J, Chorvat, Robert J, Cheeseman, Robert S, Christos, Thomas E, Bakthavatchalam, Rajagopal, Beck, James P, Cocuzza, Anthony J, Hobbs, Frank W, Wilde, Richard G, Arnold, Charles, Chidester, Dennis, Curry, Matthew, He, Liqi, Hollis, Andrea, Klaczkiewicz, John, Krenitsky, Paul J, Rescinito, Joseph P, Scholfield, Everett, Culp, Steven, De Souza, Errol B, Fitzgerald, Lawrence, Grigoriadis, Dimitri, Tam, S. William, Wong, Y. Nancy, Huang, Shiew-Mei, Shen, Helen L
Published in Journal of medicinal chemistry (11.03.1999)
Published in Journal of medicinal chemistry (11.03.1999)
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Journal Article
Cyclization of 1,1-Disubstituted Alkenes to Cyclopentenes
Taber, Douglass F, Christos, Thomas E, Neubert, Timothy D, Batra, Dolly
Published in Journal of organic chemistry (24.12.1999)
Published in Journal of organic chemistry (24.12.1999)
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A Convenient Chiron for Substituted Cyclohexanones
Taber, Douglass F, Christos, Thomas E, Rahimizadeh, Mohammed, Chen, Bei
Published in Journal of organic chemistry (24.08.2001)
Published in Journal of organic chemistry (24.08.2001)
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Cyclohexenone Annelation by Alkylidene C−H Insertion: Synthesis of Oxo-T-cadinol
Taber, Douglass F, Christos, Thomas E, Hodge, C. Nicholas
Published in Journal of organic chemistry (22.03.1996)
Published in Journal of organic chemistry (22.03.1996)
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Novel piperidine .sigma. receptor ligands as potential antipsychotic drugs
Gilligan, Paul J, Cain, Gary A, Christos, Thomas E, Cook, Leonard, Drummond, Spencer, Johnson, Alexander L, Kergaye, Ahmed A, McElroy, John F, Rohrbach, Kenneth W
Published in Journal of medicinal chemistry (01.11.1992)
Published in Journal of medicinal chemistry (01.11.1992)
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Stable isosteres of neurotensin c-terminal pentapeptides derived by modification of the amide function
Christos, Thomas E., Arvanitis, Argyrios, Cain, Gary A., Johnson, Alexander L., Pottorf, Richard S., Tam, S.William, Schmidt, William K.
Published in Bioorganic & medicinal chemistry letters (01.06.1993)
Published in Bioorganic & medicinal chemistry letters (01.06.1993)
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Journal Article
Perfluorocarbon-based antidiabetic agents
Kees, Kenneth L, Smith, Ted M, McCaleb, Michael L, Prozialeck, Dorothy H, Cheeseman, Robert S, Christos, Thomas E, Patt, William C, Steiner, Kurt E
Published in Journal of medicinal chemistry (01.03.1992)
Published in Journal of medicinal chemistry (01.03.1992)
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Journal Article
Identification of simpler analogs of neurotensin(9–13) which retain antinociceptive activity
Cain, Gary A., Christos, Thomas E., Johnson, Alexander L., Pottorf, Richard S., Tam, S.William, Schmidt, William K.
Published in Bioorganic & medicinal chemistry letters (01.08.1993)
Published in Bioorganic & medicinal chemistry letters (01.08.1993)
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Journal Article
Neurotensin receptor binding and antinociceptive activity for lipophilic N α-amido neurotensin(9–13) analogs
Cain, Gary A., Christos, Thomas E., Johnson, Alexander L., Pottorf, Richard S., Confalone, Pat N., William Tam, S., Schmidt, William K.
Published in Bioorganic & medicinal chemistry letters (01.10.1993)
Published in Bioorganic & medicinal chemistry letters (01.10.1993)
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Journal Article
Novel conformationally restricted aromatic piperidines as selective sigma receptor ligands
Cain, Gary A., Christos, Thomas E., Eyermann, Charles J., Gilligan, Paul J., Grigoriadis, Dimitri E., Johnson, Alexander L., Tam, S.William
Published in Bioorganic & medicinal chemistry letters (20.01.1994)
Published in Bioorganic & medicinal chemistry letters (20.01.1994)
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