Time-Trajectories in Efficiency Maps as Effective Guides for Drug Discovery Efforts
Christmann-Franck, Serge, Cravo, Daniel, Abad-Zapatero, Cele
Published in Molecular informatics (14.03.2011)
Published in Molecular informatics (14.03.2011)
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Journal Article
Correction: Time-Trajectories in Efficiency Maps as Effective Guides for Drug Discovery Efforts
Christmann-Franck, Serge, Cravo, Daniel, Abad-Zapatero, Cele
Published in Molecular informatics (14.03.2011)
Published in Molecular informatics (14.03.2011)
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Journal Article
Unprecedently Large-Scale Kinase Inhibitor Set Enabling the Accurate Prediction of Compound–Kinase Activities: A Way toward Selective Promiscuity by Design?
Christmann-Franck, Serge, van Westen, Gerard J. P, Papadatos, George, Beltran Escudie, Fanny, Roberts, Alexander, Overington, John P, Domine, Daniel
Published in Journal of chemical information and modeling (26.09.2016)
Published in Journal of chemical information and modeling (26.09.2016)
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Journal Article
BENZOFURANE, BENZOTHIOPHENE, BENZOTHIAZOL DERIVATIVES AS FXR MODULATORS
KOBER INGO, VENKATESHWAR RAO GUMMADI, SENGUPTA SAUMITRA, ROCHE DIDIER, CHRISTMANN FRANCK SERGE, MAUTINO GISELE, CONTARD FRANCIS, SISTLA RAMESH
Year of Publication 07.01.2011
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Year of Publication 07.01.2011
Patent
Structure-based design of 7-azaindole-pyrrolidine amides as inhibitors of 11β-hydroxysteroid dehydrogenase type I
Valeur, Eric, Christmann-Franck, Serge, Lepifre, Franck, Carniato, Denis, Cravo, Daniel, Charon, Christine, Bozec, Sophie, Musil, Djordje, Hillertz, Per, Doare, Liliane, Schmidlin, Fabien, Lecomte, Marc, Schultz, Melanie, Roche, Didier
Published in Bioorganic & medicinal chemistry letters (15.09.2012)
Published in Bioorganic & medicinal chemistry letters (15.09.2012)
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Journal Article
Discovery and structure-guided drug design of inhibitors of 11β-hydroxysteroid-dehydrogenase type I based on a spiro-carboxamide scaffold
Lepifre, Franck, Christmann-Franck, Serge, Roche, Didier, Leriche, Caroline, Carniato, Denis, Charon, Christine, Bozec, Sophie, Doare, Liliane, Schmidlin, Fabien, Lecomte, Marc, Valeur, Eric
Published in Bioorganic & medicinal chemistry letters (01.07.2009)
Published in Bioorganic & medicinal chemistry letters (01.07.2009)
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Journal Article
Correction: Time-Trajectories in Efficiency Maps as Effective Guides for Drug Discovery Efforts
Christmann-Franck, Serge, Cravo, Daniel, Abad-Zapatero, Cele
Published in Molecular informatics (14.03.2011)
Published in Molecular informatics (14.03.2011)
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Journal Article
Discovery and structure–activity relationships of pentanedioic acid diamides as potent inhibitors of 11β-hydroxysteroid dehydrogenase type I
Roche, Didier, Carniato, Denis, Leriche, Caroline, Lepifre, Franck, Christmann-Franck, Serge, Graedler, Ulrich, Charon, Christine, Bozec, Sophie, Doare, Liliane, Schmidlin, Fabien, Lecomte, Marc, Valeur, Eric
Published in Bioorganic & medicinal chemistry letters (15.05.2009)
Published in Bioorganic & medicinal chemistry letters (15.05.2009)
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Journal Article
Structure-based design of 7-azaindole-pyrrolidine amides as inhibitors of 11[beta]-hydroxysteroid dehydrogenase type I
Valeur, Eric, Christmann-Franck, Serge, Lepifre, Franck, Carniato, Denis, Cravo, Daniel, Charon, Christine, Bozec, Sophie, Musil, Djordje, Hillertz, Per, Doare, Liliane, Schmidlin, Fabien, Lecomte, Marc, Schultz, Melanie, Roche, Didier
Published in Bioorganic & medicinal chemistry letters (15.09.2012)
Published in Bioorganic & medicinal chemistry letters (15.09.2012)
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Journal Article
Structure-Based Virtual Screening: An Application to Human Topoisomerase II α
Christmann-Franck, Serge, Bertrand, Hugues-Olivier, Goupil-Lamy, Anne, der Garabedian, P. Arsène, Mauffret, Olivier, Hoffmann, Rémy, Fermandjian, Serge
Published in Journal of medicinal chemistry (30.12.2004)
Published in Journal of medicinal chemistry (30.12.2004)
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Journal Article
Pyridoxal 5′-phosphate inactivates DNA topoisomerase IB by modifying the lysine general acid
Vermeersch, Jacqueline J., Christmann-Franck, Serge, Karabashyan, Leon V., Fermandjian, Serge, Mirambeau, Gilles, Der Garabedian, P. Arsène
Published in Nucleic acids research (01.01.2004)
Published in Nucleic acids research (01.01.2004)
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Journal Article
MACROCYCLIC PYRIDAZINONE DERIVATIVES
JORAND-LEBRUN, CATHERINE, KULKARNI, SANTOSH, CHRISTMANN-FRANCK, SERGE
Year of Publication 21.09.2021
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Year of Publication 21.09.2021
Patent
Discovery and structure-guided drug design of inhibitors of 11beta-hydroxysteroid-dehydrogenase type I based on a spiro-carboxamide scaffold
Lepifre, Franck, Christmann-Franck, Serge, Roche, Didier, Leriche, Caroline, Carniato, Denis, Charon, Christine, Bozec, Sophie, Doare, Liliane, Schmidlin, Fabien, Lecomte, Marc, Valeur, Eric
Published in Bioorganic & medicinal chemistry letters (01.07.2009)
Published in Bioorganic & medicinal chemistry letters (01.07.2009)
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Journal Article
Discovery and structure-activity relationships of pentanedioic acid diamides as potent inhibitors of 11beta-hydroxysteroid dehydrogenase type I
Roche, Didier, Carniato, Denis, Leriche, Caroline, Lepifre, Franck, Christmann-Franck, Serge, Graedler, Ulrich, Charon, Christine, Bozec, Sophie, Doare, Liliane, Schmidlin, Fabien, Lecomte, Marc, Valeur, Eric
Published in Bioorganic & medicinal chemistry letters (15.05.2009)
Published in Bioorganic & medicinal chemistry letters (15.05.2009)
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Journal Article
Macrocyclic pyridazinone derivatives
Christmann-Franck, Serge, Kulkarni, Santosh, Jorand-Lebrun, Catherine
Year of Publication 04.09.2018
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Year of Publication 04.09.2018
Patent
MACROCYCLIC PYRIDAZINONE DERIVATIVES
KULKARNI, Santosh, JORAND-LEBRUN, Catherine, CHRISTMANN-FRANCK, Serge
Year of Publication 28.05.2018
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Year of Publication 28.05.2018
Patent