Senolytics reduce coronavirus-related mortality in old mice
Camell, Christina D., Yousefzadeh, Matthew J., Zhu, Yi, Prata, Larissa G. P. Langhi, Huggins, Matthew A., Pierson, Mark, Zhang, Lei, O’Kelly, Ryan D., Pirtskhalava, Tamar, Xun, Pengcheng, Ejima, Keisuke, Xue, Ailing, Tripathi, Utkarsh, Espindola-Netto, Jair Machado, Giorgadze, Nino, Atkinson, Elizabeth J., Inman, Christina L., Johnson, Kurt O., Cholensky, Stephanie H., Carlson, Timothy W., LeBrasseur, Nathan K., Khosla, Sundeep, O’Sullivan, M. Gerard, Allison, David B., Jameson, Stephen C., Meves, Alexander, Li, Ming, Prakash, Y. S., Chiarella, Sergio E., Hamilton, Sara E., Tchkonia, Tamara, Niedernhofer, Laura J., Kirkland, James L., Robbins, Paul D.
Published in Science (16.07.2021)
Published in Science (16.07.2021)
Get full text
Journal Article
Web Resource
Degradation of Polycomb Repressive Complex 2 with an EED-Targeted Bivalent Chemical Degrader
Potjewyd, Frances, Turner, Anne-Marie W., Beri, Joshua, Rectenwald, Justin M., Norris-Drouin, Jacqueline L., Cholensky, Stephanie H., Margolis, David M., Pearce, Kenneth H., Herring, Laura E., James, Lindsey I.
Published in Cell chemical biology (16.01.2020)
Published in Cell chemical biology (16.01.2020)
Get full text
Journal Article
A cellular chemical probe targeting the chromodomains of Polycomb repressive complex 1
Stuckey, Jacob I, Dickson, Bradley M, Cheng, Nancy, Liu, Yanli, Norris, Jacqueline L, Cholensky, Stephanie H, Tempel, Wolfram, Qin, Su, Huber, Katherine G, Sagum, Cari, Black, Karynne, Li, Fengling, Huang, Xi-Ping, Roth, Bryan L, Baughman, Brandi M, Senisterra, Guillermo, Pattenden, Samantha G, Vedadi, Masoud, Brown, Peter J, Bedford, Mark T, Min, Jinrong, Arrowsmith, Cheryl H, James, Lindsey I, Frye, Stephen V
Published in Nature chemical biology (01.03.2016)
Published in Nature chemical biology (01.03.2016)
Get full text
Journal Article
Discovery and Characterization of a Cellular Potent Positive Allosteric Modulator of the Polycomb Repressive Complex 1 Chromodomain, CBX7
Lamb, Kelsey N, Bsteh, Daniel, Dishman, Sarah N, Moussa, Hagar F, Fan, Huitao, Stuckey, Jacob I, Norris, Jacqueline L, Cholensky, Stephanie H, Li, Dongxu, Wang, Jingkui, Sagum, Cari, Stanton, Benjamin Z, Bedford, Mark T, Pearce, Kenneth H, Kenakin, Terry P, Kireev, Dmitri B, Wang, Gang Greg, James, Lindsey I, Bell, Oliver, Frye, Stephen V
Published in Cell chemical biology (17.10.2019)
Published in Cell chemical biology (17.10.2019)
Get full text
Journal Article
Discovery of an H3K36me3-Derived Peptidomimetic Ligand with Enhanced Affinity for Plant Homeodomain Finger Protein 1 (PHF1)
Engelberg, Isabelle A, Liu, Jiuyang, Norris-Drouin, Jacqueline L, Cholensky, Stephanie H, Ottavi, Samantha A, Frye, Stephen V, Kutateladze, Tatiana G, James, Lindsey I
Published in Journal of medicinal chemistry (24.06.2021)
Published in Journal of medicinal chemistry (24.06.2021)
Get full text
Journal Article
Age-associated accumulation of B cells promotes macrophage inflammation and inhibits lipolysis in adipose tissue during sepsis
Carey, Anna, Nguyen, Katie, Kandikonda, Pranathi, Kruglov, Victor, Bradley, Claire, Dahlquist, Korbyn J.V., Cholensky, Stephanie, Swanson, Whitney, Badovinac, Vladimir P., Griffith, Thomas S., Camell, Christina D.
Published in Cell reports (Cambridge) (26.03.2024)
Published in Cell reports (Cambridge) (26.03.2024)
Get full text
Journal Article
Structure–Activity Relationships and Kinetic Studies of Peptidic Antagonists of CBX Chromodomains
Stuckey, Jacob I, Simpson, Catherine, Norris-Drouin, Jacqueline L, Cholensky, Stephanie H, Lee, Junghyun, Pasca, Ryan, Cheng, Nancy, Dickson, Bradley M, Pearce, Kenneth H, Frye, Stephen V, James, Lindsey I
Published in Journal of medicinal chemistry (13.10.2016)
Published in Journal of medicinal chemistry (13.10.2016)
Get full text
Journal Article
PROTAC Linkerology Leads to an Optimized Bivalent Chemical Degrader of Polycomb Repressive Complex 2 (PRC2) Components
Bashore, Frances M., Foley, Caroline A., Ong, Han Wee, Rectenwald, Justin M., Hanley, Ronan P., Norris-Drouin, Jacqueline L., Cholensky, Stephanie H., Mills, Christine A., Pearce, Kenneth H., Herring, Laura E., Kireev, Dmitri, Frye, Stephen V., James, Lindsey I.
Published in ACS chemical biology (17.03.2023)
Published in ACS chemical biology (17.03.2023)
Get full text
Journal Article
Reprogramming CBX8-PRC1 function with a positive allosteric modulator
Suh, Junghyun L., Bsteh, Daniel, Hart, Bryce, Si, Yibo, Weaver, Tyler M., Pribitzer, Carina, Lau, Roy, Soni, Shivani, Ogana, Heather, Rectenwald, Justin M., Norris, Jacqueline L., Cholensky, Stephanie H., Sagum, Cari, Umana, Jessica D., Li, Dongxu, Hardy, Brian, Bedford, Mark T., Mumenthaler, Shannon M., Lenz, Heinz-Josef, Kim, Yong-Mi, Wang, Gang Greg, Pearce, Ken H., James, Lindsey I., Kireev, Dmitri B., Musselman, Catherine A., Frye, Stephen V., Bell, Oliver
Published in Cell chemical biology (21.04.2022)
Published in Cell chemical biology (21.04.2022)
Get full text
Journal Article
Chromodomain Ligand Optimization via Target-Class Directed Combinatorial Repurposing
Barnash, Kimberly D, Lamb, Kelsey N, Stuckey, Jacob I, Norris, Jacqueline L, Cholensky, Stephanie H, Kireev, Dmitri B, Frye, Stephen V, James, Lindsey I
Published in ACS chemical biology (16.09.2016)
Published in ACS chemical biology (16.09.2016)
Get full text
Journal Article
Design and Construction of a Focused DNA-Encoded Library for Multivalent Chromatin Reader Proteins
Rectenwald, Justin M, Guduru, Shiva Krishna Reddy, Dang, Zhao, Collins, Leonard B, Liao, Yi-En, Norris-Drouin, Jacqueline L, Cholensky, Stephanie H, Kaufmann, Kyle W, Hammond, Scott M, Kireev, Dmitri B, Frye, Stephen V, Pearce, Kenneth H
Published in Molecules (Basel, Switzerland) (22.02.2020)
Published in Molecules (Basel, Switzerland) (22.02.2020)
Get full text
Journal Article
Discovery of Peptidomimetic Ligands of EED as Allosteric Inhibitors of PRC2
Barnash, Kimberly D, The, Juliana, Norris-Drouin, Jacqueline L, Cholensky, Stephanie H, Worley, Beau M, Li, Fengling, Stuckey, Jacob I, Brown, Peter J, Vedadi, Masoud, Arrowsmith, Cheryl H, Frye, Stephen V, James, Lindsey I
Published in ACS combinatorial science (13.03.2017)
Published in ACS combinatorial science (13.03.2017)
Get full text
Journal Article
A Peptidomimetic Ligand Targeting the Chromodomain of MPP8 Reveals HRP2’s Association with the HUSH Complex
Waybright, Jarod M, Clinkscales, Sarah E, Barnash, Kimberly D, Budziszewski, Gabrielle R, Rectenwald, Justin M, Chiarella, Anna M, Norris-Drouin, Jacqueline L, Cholensky, Stephanie H, Pearce, Kenneth H, Herring, Laura E, McGinty, Robert K, Hathaway, Nathaniel A, James, Lindsey I
Published in ACS chemical biology (17.09.2021)
Published in ACS chemical biology (17.09.2021)
Get full text
Journal Article
A General TR-FRET Assay Platform for High-Throughput Screening and Characterizing Inhibitors of Methyl-Lysine Reader Proteins
Rectenwald, Justin M., Hardy, P. Brian, Norris-Drouin, Jacqueline L., Cholensky, Stephanie H., James, Lindsey I., Frye, Stephen V., Pearce, Kenneth H.
Published in SLAS discovery (01.07.2019)
Published in SLAS discovery (01.07.2019)
Get full text
Journal Article
Discovery and Characterization of Peptide Inhibitors for Calcium and Integrin Binding Protein 1
Puhl, Ana C, Bogart, Jonathan W, Haberman, Victoria A, Larson, Jacob E, Godoy, Andre S, Norris-Drouin, Jacqueline L, Cholensky, Stephanie H, Leisner, Tina M, Frye, Stephen V, Parise, Leslie V, Bowers, Albert A, Pearce, Kenneth H
Published in ACS chemical biology (19.06.2020)
Published in ACS chemical biology (19.06.2020)
Get full text
Journal Article
Quantitative Characterization of Bivalent Probes for a Dual Bromodomain Protein, Transcription Initiation Factor TFIID Subunit 1
Suh, Junghyun L, Watts, Brian, Stuckey, Jacob I, Norris-Drouin, Jacqueline L, Cholensky, Stephanie H, Dickson, Bradley M, An, Yi, Mathea, Sebastian, Salah, Eidarus, Knapp, Stefan, Khan, Abid, Adams, Alexander T, Strahl, Brian D, Sagum, Cari A, Bedford, Mark T, James, Lindsey I, Kireev, Dmitri B, Frye, Stephen V
Published in Biochemistry (Easton) (10.04.2018)
Published in Biochemistry (Easton) (10.04.2018)
Get full text
Journal Article
PD1 blockade improves survival and CD8 + cytotoxic capacity, without increasing inflammation, during normal microbial experience in old mice
Dahlquist, Korbyn J V, Huggins, Matthew A, Yousefzadeh, Matthew J, Soto-Palma, Carolina, Cholensky, Stephanie H, Pierson, Mark, Smith, Declan M, Hamilton, Sara E, Camell, Christina D
Published in Nature aging (01.07.2024)
Published in Nature aging (01.07.2024)
Get more information
Journal Article
Correction to “Quantitative Characterization of Bivalent Probes for a Dual Bromodomain Protein, Transcription Initiation Factor TFIID subunit 1”
Suh, Junghyun L, Watts, Brian, Stuckey, Jacob I, Norris-Drouin, Jacqueline L, Cholensky, Stephanie H, Dickson, Bradley M, An, Yi, Mathea, Sebastian, Salah, Eidarus, Knapp, Stefan, Khan, Abid, Adams, Alexander T, Strahl, Brian D, Sagum, Cari A, Bedford, Mark T, James, Lindsey I, Kireev, Dmitri B, Frye, Stephen V
Published in Biochemistry (Easton) (11.12.2018)
Published in Biochemistry (Easton) (11.12.2018)
Get full text
Journal Article
Discovery of Potent Peptidomimetic Antagonists for Heterochromatin Protein 1 Family Proteins
Lamb, Kelsey N, Dishman, Sarah N, Waybright, Jarod M, Engelberg, Isabelle A, Rectenwald, Justin M, Norris-Drouin, Jacqueline L, Cholensky, Stephanie H, Pearce, Kenneth H, James, Lindsey I, Frye, Stephen V
Published in ACS omega (11.01.2022)
Published in ACS omega (11.01.2022)
Get full text
Journal Article