Crystal Structures of Human Factor Xa Complexed with Potent Inhibitors
Maignan, Sébastien, Guilloteau, Jean-Pierre, Pouzieux, Stéphanie, Choi-Sledeski, Yong Mi, Becker, Michael R, Klein, Scott I, Ewing, William R, Pauls, Henry W, Spada, Alfred P, Mikol, Vincent
Published in Journal of medicinal chemistry (24.08.2000)
Published in Journal of medicinal chemistry (24.08.2000)
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Aminoisoquinolines: Design and synthesis of an orally active benzamidine isostere for the inhibition of factor XA
Choi-Sledeski, Y.M., Becker, M.R., Green, D.M., Davis, R., Ewing, W.R., Mason, H.J., Ly, C., Spada, A., Liang, G., Cheney, D., Barton, J., Chu, V., Brown, K., Colussi, D., Bentley, R., Leadley, R., Dunwiddie, C., Pauls, H.W.
Published in Bioorganic & medicinal chemistry letters (06.09.1999)
Published in Bioorganic & medicinal chemistry letters (06.09.1999)
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Design and Structure−Activity Relationships of Potent and Selective Inhibitors of Blood Coagulation Factor Xa
Ewing, William R, Becker, Michael R, Manetta, Vincent E, Davis, Roderick S, Pauls, Henry W, Mason, Helen, Choi-Sledeski, Yong Mi, Green, Daniel, Cha, Don, Spada, Alfred P, Cheney, Daniel L, Mason, Jonathan S, Maignan, Sebastien, Guilloteau, Jean-Pierre, Brown, Karen, Colussi, Dennis, Bentley, Ross, Bostwick, Jeff, Kasiewski, Charles J, Morgan, Suzanne R, Leadley, Robert J, Dunwiddie, Christopher T, Perrone, Mark H, Chu, Valeria
Published in Journal of medicinal chemistry (09.09.1999)
Published in Journal of medicinal chemistry (09.09.1999)
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Synthesis, SAR and in vivo activity of novel thienopyridine sulfonamide pyrrolidinones as factor Xa inhibitors
Becker, Michael R., Ewing, William R., Davis, Roderick S., Pauls, Henry W., Ly, Cuong, Li, Aiwen, Mason, Helen J., Choi-Sledeski, Yong Mi, Spada, Alfred P., Chu, Valeria, Brown, Karen D., Colussi, Dennis J., Leadley, Robert J., Bentley, Ross, Bostwick, Jeff, Kasiewski, Charles, Morgan, Suzanne
Published in Bioorganic & medicinal chemistry letters (20.09.1999)
Published in Bioorganic & medicinal chemistry letters (20.09.1999)
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Solid-phase parallel synthesis of azarene pyrrolidinones as factor Xa inhibitors
Gong, Y, Becker, M, Choi-Sledeski, Y M, Davis, R S, Salvino, J M, Chu, V, Brown, K D, Pauls, H W
Published in Bioorganic & medicinal chemistry letters (15.05.2000)
Published in Bioorganic & medicinal chemistry letters (15.05.2000)
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Synthesis of Functionalized Aromatic Oligomers from a Versatile Diphenylmethane Template
Bruno, J. G, Chang, M. N, Choi-Sledeski, Y. M, Green, D. M, McGarry, D. G, Regan, J. R, Volz, F. A
Published in Journal of organic chemistry (25.07.1997)
Published in Journal of organic chemistry (25.07.1997)
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Discovery of an orally efficacious inhibitor of coagulation factor Xa which incorporates a neutral P-1 ligand
Choi-Sledeski, YM, Kearney, R, Poli, G, Pauls, H, Gardner, C, Gong, Y, Becker, M, Davis, R, Spada, A, Liang, G, Chu, Brown, K, Collussi, D, Leadley, R, Rebello, S, Moxey, P, Morgan, S, Bentley, R, Kasiewski, C, Maignan, S, Guilloteau, JP, Mikol
Published in Journal of medicinal chemistry (27.02.2003)
Published in Journal of medicinal chemistry (27.02.2003)
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Sulfonamidopyrrolidinone Factor Xa Inhibitors: Potency and Selectivity Enhancements via P-1 and P-4 Optimization
Choi-Sledeski, Yong Mi, McGarry, Daniel G, Green, Daniel M, Mason, Helen J, Becker, Michael R, Davis, Roderick S, Ewing, William R, Dankulich, William P, Manetta, Vincent E, Morris, Robert L, Spada, Alfred P, Cheney, Daniel L, Brown, Karen D, Colussi, Dennis J, Chu, Valeria, Heran, Christopher L, Morgan, Suzanne R, Bentley, Ross G, Leadley, Robert J, Maignan, Sebastien, Guilloteau, Jean-Pierre, Dunwiddie, Christopher T, Pauls, Henry W
Published in Journal of medicinal chemistry (09.09.1999)
Published in Journal of medicinal chemistry (09.09.1999)
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