Search Results - "Chodkowski, Andrzej" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Novel multi-target ligands of dopamine and serotonin receptors for the treatment of schizophrenia based on indazole and piperazine scaffolds-synthesis, biological activity, and structural evaluation

Novel multi-target ligands of dopamine and serotonin receptors for the treatment of schizophrenia based on indazole and piperazine scaffolds-synthesis, biological activity, and structural evaluation

by Stępnicki, Piotr, Wronikowska-Denysiuk, Olga, Zięba, Agata, Targowska-Duda, Katarzyna M., Bartyzel, Agata, Wróbel, Martyna Z., Wróbel, Tomasz M., Szałaj, Klaudia, Chodkowski, Andrzej, Mirecka, Karolina, Budzyńska, Barbara, Fornal, Emilia, Turło, Jadwiga, Castro, Marián, Kaczor, Agnieszka A.
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2023)

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Synthesis and anticonvulsant activity of novel 2,6-diketopiperazine derivatives. Part 1: Perhydropyrrole[1,2- a]pyrazines

Synthesis and anticonvulsant activity of novel 2,6-diketopiperazine derivatives. Part 1: Perhydropyrrole[1,2- a]pyrazines

by Dawidowski, Maciej, Herold, Franciszek, Chodkowski, Andrzej, Kleps, Jerzy, Szulczyk, Paweł, Wilczek, Marcin
Published in European journal of medicinal chemistry (01.10.2011)

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Design and Synthesis of Potential Multi-Target Antidepressants: Exploration of 1-pyrrolidine-2,5-dione Derivatives with Affinity for the Serotonin Transporter

Design and Synthesis of Potential Multi-Target Antidepressants: Exploration of 1-pyrrolidine-2,5-dione Derivatives with Affinity for the Serotonin Transporter

by Wróbel, Martyna Z, Chodkowski, Andrzej, Siwek, Agata, Satała, Grzegorz, Bojarski, Andrzej J, Dawidowski, Maciej
Published in International journal of molecular sciences (01.10.2024)

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Design and Synthesis of Potential Multi-Target Antidepressants: Exploration of 1-(4-(7-Azaindole)-3,6-dihydropyridin-1-yl)alkyl-3-(1 H -indol-3-yl)pyrrolidine-2,5-dione Derivatives with Affinity for the Serotonin Transporter

Design and Synthesis of Potential Multi-Target Antidepressants: Exploration of 1-(4-(7-Azaindole)-3,6-dihydropyridin-1-yl)alkyl-3-(1 H -indol-3-yl)pyrrolidine-2,5-dione Derivatives with Affinity for the Serotonin Transporter

by Wróbel, Martyna Z, Chodkowski, Andrzej, Siwek, Agata, Satała, Grzegorz, Bojarski, Andrzej J, Dawidowski, Maciej
Published in International journal of molecular sciences (20.10.2024)

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Understanding performance of 3D-printed sorbent in study of metabolic stability

Understanding performance of 3D-printed sorbent in study of metabolic stability

by Ulenberg, Szymon, Georgiev, Paweł, Belka, Mariusz, Ślifirski, Grzegorz, Wróbel, Martyna, Chodkowski, Andrzej, Król, Marek, Herold, Franciszek, Bączek, Tomasz
Published in Journal of Chromatography A (11.10.2020)

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Synthesis of new 4-butyl-arylpiperazine-3-(1H-indol-3-yl)pyrrolidine-2,5-dione derivatives and evaluation for their 5-HT1A and D-2 receptor affinity and serotonin transporter inhibition

Synthesis of new 4-butyl-arylpiperazine-3-(1H-indol-3-yl)pyrrolidine-2,5-dione derivatives and evaluation for their 5-HT1A and D-2 receptor affinity and serotonin transporter inhibition

by Wrobel, Martyna Z., Chodkowski, Andrzej, Marciniak, Monika, Dawidowski, Maciej, Maksymiuk, Anna, Siwek, Agata, Nowak, Gabriel, Turlo, Jadwiga
Published in Bioorganic chemistry (01.04.2020)

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Synthesis of new 4-butyl-arylpiperazine-3-(1H-indol-3-yl)pyrrolidine-2,5-dione derivatives and evaluation for their 5-HT1A and D2 receptor affinity and serotonin transporter inhibition

Synthesis of new 4-butyl-arylpiperazine-3-(1H-indol-3-yl)pyrrolidine-2,5-dione derivatives and evaluation for their 5-HT1A and D2 receptor affinity and serotonin transporter inhibition

by Wróbel, Martyna Z., Chodkowski, Andrzej, Marciniak, Monika, Dawidowski, Maciej, Maksymiuk, Anna, Siwek, Agata, Nowak, Gabriel, Turło, Jadwiga
Published in Bioorganic chemistry (01.04.2020)

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Synthesis and biological evaluation of new multi-target 3-(1H-indol-3-yl)pyrrolidine-2,5-dione derivatives with potential antidepressant effect

Synthesis and biological evaluation of new multi-target 3-(1H-indol-3-yl)pyrrolidine-2,5-dione derivatives with potential antidepressant effect

by Wróbel, Martyna Z., Chodkowski, Andrzej, Herold, Franciszek, Marciniak, Monika, Dawidowski, Maciej, Siwek, Agata, Starowicz, Gabriela, Stachowicz, Katarzyna, Szewczyk, Bernadeta, Nowak, Gabriel, Belka, Mariusz, Bączek, Tomasz, Satała, Grzegorz, Bojarski, Andrzej J., Turło, Jadwiga
Published in European journal of medicinal chemistry (01.12.2019)

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Synthesis and biological evaluation of novel 3-(5-substituted-1H-indol-3-yl)pyrrolidine-2,5-dione derivatives with a dual affinity for serotonin 5-HT1A receptor and SERT

Synthesis and biological evaluation of novel 3-(5-substituted-1H-indol-3-yl)pyrrolidine-2,5-dione derivatives with a dual affinity for serotonin 5-HT1A receptor and SERT

by Wróbel, Martyna Z., Chodkowski, Andrzej, Dawidowski, Maciej, Siwek, Agata, Stachowicz, Katarzyna, Szewczyk, Bernadeta, Nowak, Gabriel, Satała, Grzegorz, Bojarski, Andrzej J., Turło, Jadwiga
Published in Bioorganic chemistry (01.12.2023)

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Synthesis and anticonvulsant activity of novel 2,6-diketopiperazine derivatives. Part 2: Perhydropyrido[1,2- a]pyrazines

Synthesis and anticonvulsant activity of novel 2,6-diketopiperazine derivatives. Part 2: Perhydropyrido[1,2- a]pyrazines

by Dawidowski, Maciej, Herold, Franciszek, Chodkowski, Andrzej, Kleps, Jerzy
Published in European journal of medicinal chemistry (01.02.2012)

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Discovery of novel arylpiperazine-based DA/5-HT modulators as potential antipsychotic agents – Design, synthesis, structural studies and pharmacological profiling

Discovery of novel arylpiperazine-based DA/5-HT modulators as potential antipsychotic agents – Design, synthesis, structural studies and pharmacological profiling

by Stępnicki, Piotr, Targowska-Duda, Katarzyna M., Martínez, Antón L., Zięba, Agata, Wronikowska-Denysiuk, Olga, Wróbel, Martyna Z., Bartyzel, Agata, Trzpil, Alicja, Wróbel, Tomasz M., Chodkowski, Andrzej, Mirecka, Karolina, Karcz, Tadeusz, Szczepańska, Katarzyna, Loza, Maria I., Budzyńska, Barbara, Turło, Jadwiga, Handzlik, Jadwiga, Fornal, Emilia, Poleszak, Ewa, Castro, Marián, Kaczor, Agnieszka A.
Published in European journal of medicinal chemistry (05.04.2023)

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Synthesis of bicyclic 2,6-diketopiperazines via a three-step sequence involving an Ugi five-center, four-component reaction

Synthesis of bicyclic 2,6-diketopiperazines via a three-step sequence involving an Ugi five-center, four-component reaction

by Dawidowski, Maciej, Herold, Franciszek, Wilczek, Marcin, Turło, Jadwiga, Chodkowski, Andrzej, Gomółka, Anna, Kleps, Jerzy
Published in Tetrahedron (30.09.2012)

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Novel 4-aryl-pyrido[1,2-c]pyrimidines with dual SSRI and 5-HT1A activity. Part 4

Novel 4-aryl-pyrido[1,2-c]pyrimidines with dual SSRI and 5-HT1A activity. Part 4

by Chodkowski, Andrzej, Wróbel, Martyna Z., Turło, Jadwiga, Kleps, Jerzy, Siwek, Agata, Nowak, Gabriel, Belka, Mariusz, Bączek, Tomasz, Mazurek, Aleksander P., Herold, Franciszek
Published in European journal of medicinal chemistry (27.01.2015)

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Synthesis and biological evaluation of novel pyrrolidine-2,5-dione derivatives as potential antidepressant agents. Part 1

Synthesis and biological evaluation of novel pyrrolidine-2,5-dione derivatives as potential antidepressant agents. Part 1

by Wróbel, Martyna Z., Chodkowski, Andrzej, Herold, Franciszek, Gomółka, Anna, Kleps, Jerzy, Mazurek, Aleksander P., Pluciński, Franciszek, Mazurek, Andrzej, Nowak, Gabriel, Siwek, Agata, Stachowicz, Katarzyna, Sławińska, Anna, Wolak, Małgorzata, Szewczyk, Bernadeta, Satała, Grzegorz, Bojarski, Andrzej J., Turło, Jadwiga
Published in European journal of medicinal chemistry (01.05.2013)

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Novel 4-aryl-pyrido[1,2-c]pyrimidines with dual SSRI and 5-HT1A activity. Part 5

Novel 4-aryl-pyrido[1,2-c]pyrimidines with dual SSRI and 5-HT1A activity. Part 5

by Gomółka, Anna, Ciesielska, Agnieszka, Wróbel, Martyna Z., Chodkowski, Andrzej, Kleps, Jerzy, Dawidowski, Maciej, Siwek, Agata, Wolak, Małgorzata, Stachowicz, Katarzyna, Sławińska, Anna, Nowak, Gabriel, Satała, Grzegorz, Bojarski, Andrzej J., Belka, Mariusz, Ulenberg, Szymon, Bączek, Tomasz, Skowronek, Paweł, Turło, Jadwiga, Herold, Franciszek
Published in European journal of medicinal chemistry (15.06.2015)

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Structure-activity relationship and cardiac safety of 2-aryl-2-(pyridin-2-yl)acetamides as a new class of broad-spectrum anticonvulsants derived from Disopyramide

Structure-activity relationship and cardiac safety of 2-aryl-2-(pyridin-2-yl)acetamides as a new class of broad-spectrum anticonvulsants derived from Disopyramide

by Dawidowski, Maciej, Król, Marek, Szulczyk, Bartłomiej, Chodkowski, Andrzej, Podsadni, Piotr, Konopelski, Piotr, Ufnal, Marcin, Szuberski, Piotr, Wróbel, Martyna Zofia, Zhang, Yihong, El Harchi, Aziza, Hancox, Jules C., Jarkovska, Dagmar, Mistrova, Eliska, Sviglerova, Jitka, Štengl, Milan, Popowicz, Grzegorz M., Turło, Jadwiga
Published in Bioorganic chemistry (01.05.2020)

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Synthesis of new 4-butyl-arylpiperazine-3-(1H-indol-3-yl)pyrrolidine-2,5-dione derivatives and evaluation for their 5-HT 1A and D 2 receptor affinity and serotonin transporter inhibition

Synthesis of new 4-butyl-arylpiperazine-3-(1H-indol-3-yl)pyrrolidine-2,5-dione derivatives and evaluation for their 5-HT 1A and D 2 receptor affinity and serotonin transporter inhibition

by Wróbel, Martyna Z, Chodkowski, Andrzej, Marciniak, Monika, Dawidowski, Maciej, Maksymiuk, Anna, Siwek, Agata, Nowak, Gabriel, Turło, Jadwiga
Published in Bioorganic chemistry (01.04.2020)

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Novel 4-aryl-pyrido[1,2-c]pyrimidines with dual SSRI and 5-HT1A activity. part 3

Novel 4-aryl-pyrido[1,2-c]pyrimidines with dual SSRI and 5-HT1A activity. part 3

by Herold, Franciszek, Chodkowski, Andrzej, Izbicki, Łukasz, Turło, Jadwiga, Dawidowski, Maciej, Kleps, Jerzy, Nowak, Gabriel, Stachowicz, Katarzyna, Dybała, Małgorzata, Siwek, Agata, Mazurek, Aleksander P., Mazurek, Andrzej, Pluciński, Franciszek
Published in European journal of medicinal chemistry (01.01.2011)

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Novel 4-aryl-pyrido[1,2-c]pyrimidines with dual SSRI and 5-HT1A activity, Part 1

Novel 4-aryl-pyrido[1,2-c]pyrimidines with dual SSRI and 5-HT1A activity, Part 1

by Herold, Franciszek, Chodkowski, Andrzej, Izbicki, Lukasz, Krol, Marek, Kleps, Jerzy, Turlo, Jadwiga, Nowak, Gabriel, Stachowicz, Katarzyna, Dybala, Malgorzata, Siwek, Agata
Published in European journal of medicinal chemistry (01.04.2009)

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The synthesis of new diastereomers of (4 S,8a S)- and (4 R,8a S)-4-phenyl-perhydropyrrole[1,2- a]pyrazine-1,3-dione

The synthesis of new diastereomers of (4 S,8a S)- and (4 R,8a S)-4-phenyl-perhydropyrrole[1,2- a]pyrazine-1,3-dione

by Herold, Franciszek, Dawidowski, Maciej, Wolska, Irena, Chodkowski, Andrzej, Kleps, Jerzy, Turło, Jadwiga, Zimniak, Andrzej
Published in Tetrahedron: asymmetry (04.09.2007)

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