Discovery of a Potent and Orally Bioavailable Cyclophilin Inhibitor Derived from the Sanglifehrin Macrocycle
Mackman, Richard L, Steadman, Victoria A, Dean, David K, Jansa, Petr, Poullennec, Karine G, Appleby, Todd, Austin, Carol, Blakemore, Caroline A, Cai, Ruby, Cannizzaro, Carina, Chin, Gregory, Chiva, Jean-Yves C, Dunbar, Neil A, Fliri, Hans, Highton, Adrian J, Hui, Hon, Ji, Mingzhe, Jin, Haolun, Karki, Kapil, Keats, Andrew J, Lazarides, Linos, Lee, Yu-Jen, Liclican, Albert, Mish, Michael, Murray, Bernard, Pettit, Simon B, Pyun, Peter, Sangi, Michael, Santos, Rex, Sanvoisin, Jonathan, Schmitz, Uli, Schrier, Adam, Siegel, Dustin, Sperandio, David, Stepan, George, Tian, Yang, Watt, Gregory M, Yang, Hai, Schultz, Brian E
Published in Journal of medicinal chemistry (08.11.2018)
Published in Journal of medicinal chemistry (08.11.2018)
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Journal Article
The Discovery of Potent Nonstructural Protein 5A (NS5A) Inhibitors with a Unique Resistance Profile-Part 1
Tran, Thien Duc, Wakenhut, Florian, Pickford, Chris, Shaw, Stephen, Westby, Mike, Smith-Burchnell, Caroline, Watson, Lesa, Paradowski, Michael, Milbank, Jared, Brimage, Rebecca A., Halstead, Rebecca, Glen, Rebecca, Wilson, Craig P., Adam, Fiona, Hay, Duncan, Chiva, Jean-Yves, Nichols, Carly, Blakemore, David C., Gardner, Iain, Dayal, Satish, Pike, Andrew, Webster, Rob, Pryde, David C.
Published in ChemMedChem (01.07.2014)
Published in ChemMedChem (01.07.2014)
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The Discovery of Potent Nonstructural Protein 5A (NS5A) Inhibitors with a Unique Resistance Profile-Part 2
Wakenhut, Florian, Tran, Thien Duc, Pickford, Chris, Shaw, Stephen, Westby, Mike, Smith-Burchnell, Caroline, Watson, Lesa, Paradowski, Michael, Milbank, Jared, Stonehouse, David, Cheung, Kathy, Wybrow, Robert, Daverio, Felice, Crook, Samuel, Statham, Keith, Leese, David, Stead, Darren, Adam, Fiona, Hay, Duncan, Roberts, Lee R., Chiva, Jean-Yves, Nichols, Carly, Blakemore, David C., Goetz, Gilles H., Che, Ye, Gardner, Iain, Dayal, Satish, Pike, Andrew, Webster, Rob, Pryde, David C.
Published in ChemMedChem (01.07.2014)
Published in ChemMedChem (01.07.2014)
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1-Amido-1-phenyl-3-piperidinylbutanes – CCR5 antagonists for the treatment of HIV: Part 2
Barber, Christopher G., Blakemore, David C., Chiva, Jean-Yves, Eastwood, Rachel L., Middleton, Donald S., Paradowski, Kerry A.
Published in Bioorganic & medicinal chemistry letters (01.03.2009)
Published in Bioorganic & medicinal chemistry letters (01.03.2009)
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Journal Article
1-Amido-1-phenyl-3-piperidinylbutanes — CCR5 antagonists for the treatment of HIV. Part 1
Barber, Christopher G., Blakemore, David C., Chiva, Jean-Yves, Eastwood, Rachel L., Middleton, Donald S., Paradowski, Kerry A.
Published in Bioorganic & medicinal chemistry letters (15.02.2009)
Published in Bioorganic & medicinal chemistry letters (15.02.2009)
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Journal Article
Design and optimization of selective serotonin re-uptake inhibitors with high synthetic accessibility Part 1
Andrews, Mark, Brown, Alan, Chiva, Jean-Yves, Fradet, David, Gordon, David, Lansdell, Mark, MacKenny, Malcolm
Published in Bioorganic & medicinal chemistry letters (15.04.2009)
Published in Bioorganic & medicinal chemistry letters (15.04.2009)
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Journal Article
Design and optimisation of selective serotonin re-uptake inhibitors with high synthetic accessibility: Part 2
Andrews, Mark, Brown, Alan, Chiva, Jean-Yves, Fradet, David, Gordon, David, Lansdell, Mark, MacKenny, Malcolm
Published in Bioorganic & medicinal chemistry letters (15.10.2009)
Published in Bioorganic & medicinal chemistry letters (15.10.2009)
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Journal Article
A concise synthesis of HIV integrase inhibitors bearing the dipyridone acid motif
Platts, Michelle Y., Barber, Christopher G., Chiva, Jean-Yves, Eastwood, Rachel L., Fenwick, David R., Paradowski, Kerry A., Blakemore, David C.
Published in Tetrahedron letters (26.01.2011)
Published in Tetrahedron letters (26.01.2011)
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Journal Article
The Discovery of Potent Nonstructural Protein 5A (NS5A) Inhibitors with a Unique Resistance Profile--Part1
Tran, Thien Duc, Wakenhut, Florian, Pickford, Chris, Shaw, Stephen, Westby, Mike, Smith-Burchnell, Caroline, Watson, Lesa, Paradowski, Michael, Milbank, Jared, Brimage, Rebecca A, Halstead, Rebecca, Glen, Rebecca, Wilson, Craig P, Adam, Fiona, Hay, Duncan, Chiva, Jean-Yves, Nichols, Carly, Blakemore, David C, Gardner, Iain, Dayal, Satish, Pike, Andrew, Webster, Rob, Pryde, David C
Published in ChemMedChem (01.07.2014)
Published in ChemMedChem (01.07.2014)
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Journal Article
The Discovery of Potent Nonstructural Protein 5A (NS5A) Inhibitors with a Unique Resistance Profile--Part2
Wakenhut, Florian, Tran, Thien Duc, Pickford, Chris, Shaw, Stephen, Westby, Mike, Smith-Burchnell, Caroline, Watson, Lesa, Paradowski, Michael, Milbank, Jared, Stonehouse, David, Cheung, Kathy, Wybrow, Robert, Daverio, Felice, Crook, Samuel, Statham, Keith, Leese, David, Stead, Darren, Adam, Fiona, Hay, Duncan, Roberts, Lee R, Chiva, Jean-Yves, Nichols, Carly, Blakemore, David C, Goetz, Gilles H, Che, Ye, Gardner, Iain, Dayal, Satish, Pike, Andrew, Webster, Rob, Pryde, David C
Published in ChemMedChem (01.07.2014)
Published in ChemMedChem (01.07.2014)
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NOVEL DEPSIPEPTIDE AND USES THEREOF
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Year of Publication 14.08.2024
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Year of Publication 14.08.2024
Patent
NOVEL DEPSIPEPTIDE AND USES THEREOF
LING, Losee, Lucy, SPOERING, Amy, LEWIS, Kim, STEADMAN, Victoria, Alexandra, HUGHES, Dallas, EPSTEIN, Slava, NITTI, Anthony, PEOPLES, Aaron, J, MILLETT, William, POULLENNEC, Karine, Gaelle, CHIVA, Jean-Yves, Christophe, LAZARIDES, Linos, JONES, Michael Kenyon
Year of Publication 27.03.2024
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Year of Publication 27.03.2024
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Depsipeptide and uses thereof
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Year of Publication 26.12.2023
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Year of Publication 26.12.2023
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Novel depsipeptide and uses thereof
SPOERING, Amy, PEOPLES, Aaron J, LEWIS, Kim, MILLETT, William, HUGHES, Dallas, LING, Losee Lucy, STEADMAN, Victoria Alexandra, POULENEC, Karine Gaelle, LAZARIDES, Linos, CHIVA, Jean-Yves Christophe, JONES, Michael Kenyon, NITTI, Anthony
Year of Publication 11.05.2023
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Year of Publication 11.05.2023
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NOVEL DEPSIPEPTIDE AND USES THEREOF
Hughes, Dallas, Lewis, Kim, Nitti, Anthony, Chiva, Jean-Yves Christophe, Millett, William, Ling, Losee Lucy, Poullennec, Karine Gaelle, Steadman, Victoria Alexandra, Spoering, Amy, Jones, Michael Kenyon, Lazarides, Linos, Epstein, Slava, Peoples, Aaron J
Year of Publication 15.09.2022
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Year of Publication 15.09.2022
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NOVEL DEPSIPEPTIDE AND USES THEREOF
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Year of Publication 01.12.2021
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Year of Publication 01.12.2021
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Depsipeptide and uses thereof
Hughes, Dallas, Lewis, Kim, Nitti, Anthony, Chiva, Jean-Yves Christophe, Millett, William, Ling, Losee Lucy, Poullennec, Karine Gaelle, Steadman, Victoria Alexandra, Spoering, Amy, Jones, Michael Kenyon, Lazarides, Linos, Epstein, Slava, Peoples, Aaron J
Year of Publication 16.11.2021
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Year of Publication 16.11.2021
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MACROCYCLIC INHIBITORS OF FLAVIVIRIDAE VIRUSES
WATT, GREGORY, SCHRIER, ADAM JAMES, HIGHTON, ADRIAN JOHN, STEADMAN, VICTORIA ALEXANDRA, KEATS, ANDREW JOHN, CHIVA, JEAN YVES, LAZARIDES, LINOS, POULLENNEC, KARINE G, JANSA, PETR, DEAN, DAVID KENNETH, ACIRO, CAROLINE, MACKMAN, RICHARD, SIEGEL, DUSTIN SCOTT
Year of Publication 07.09.2021
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Year of Publication 07.09.2021
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MACROCYCLIC INHIBITORS OF FLAVIVIRIDAE VIRUSES
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Year of Publication 25.08.2021
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Year of Publication 25.08.2021
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Novel depsipeptide and uses thereof
SPOERING, Amy, PEOPLES, Aaron J, LEWIS, Kim, MILLETT, William, HUGHES, Dallas, LING, Losee Lucy, STEADMAN, Victoria Alexandra, POULENEC, Karine Gaelle, LAZARIDES, Linos, CHIVA, Jean-Yves Christophe, JONES, Michael Kenyon, NITTI, Anthony
Year of Publication 19.08.2021
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Year of Publication 19.08.2021
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