Synthesis and Evaluation of Efavirenz (Sustiva TM) Analogues as HIV-1 Reverse Transcriptase Inhibitors: Replacement of the Cyclopropylacetylene Side Chain
Cocuzza, Anthony J., Chidester, Dennis R., Cordova, Beverly C., Jeffrey, Susan, Parsons, Rodney L., Bacheler, Lee T., Erickson-Viitanen, Susan, Trainor, George L., Ko, Soo S.
Published in Bioorganic & medicinal chemistry letters (07.05.2001)
Published in Bioorganic & medicinal chemistry letters (07.05.2001)
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Use of the suzuki reaction for the synthesis of aryl-substituted heterocycles as corticotropin-releasing hormone (CRH) antagonists
Cocuzza, Anthony J., Chidester, Dennis R., Culp, Steven, Fitzgerald, Lawrence, Gilligan, Paul
Published in Bioorganic & medicinal chemistry letters (05.04.1999)
Published in Bioorganic & medicinal chemistry letters (05.04.1999)
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Journal Article
4,1-Benzoxazepinone analogues of efavirenz (Sustiva™) as HIV-1 reverse transcriptase inhibitors
Cocuzza, Anthony J., Chidester, Dennis R., Cordova, Beverly C., Klabe, Ronald M., Jeffrey, Susan, Diamond, Sharon, Weigelt, Carolyn A., Ko, Soo S., Bacheler, Lee T., Erickson-Viitanen, Susan K., Rodgers, James D.
Published in Bioorganic & medicinal chemistry letters (04.06.2001)
Published in Bioorganic & medicinal chemistry letters (04.06.2001)
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The discovery of 4-(3-pentylamino)-2,7-dimethyl-8-(2-methyl-4-methoxyphenyl)-pyrazolo-[1 ,5-a]-pyrimidine: a corticotropin-releasing factor (hCRF1) antagonist
Gilligan, P J, Baldauf, C, Cocuzza, A, Chidester, D, Zaczek, R, Fitzgerald, L W, McElroy, J, Smith, M A, Shen, H S, Saye, J A, Christ, D, Trainor, G, Robertson, D W, Hartig, P
Published in Bioorganic & medicinal chemistry (01.01.2000)
Published in Bioorganic & medicinal chemistry (01.01.2000)
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Non-Peptide Corticotropin-Releasing Hormone Antagonists: Syntheses and Structure−Activity Relationships of 2-Anilinopyrimidines and -triazines
Arvanitis, Argyrios G, Gilligan, Paul J, Chorvat, Robert J, Cheeseman, Robert S, Christos, Thomas E, Bakthavatchalam, Rajagopal, Beck, James P, Cocuzza, Anthony J, Hobbs, Frank W, Wilde, Richard G, Arnold, Charles, Chidester, Dennis, Curry, Matthew, He, Liqi, Hollis, Andrea, Klaczkiewicz, John, Krenitsky, Paul J, Rescinito, Joseph P, Scholfield, Everett, Culp, Steven, De Souza, Errol B, Fitzgerald, Lawrence, Grigoriadis, Dimitri, Tam, S. William, Wong, Y. Nancy, Huang, Shiew-Mei, Shen, Helen L
Published in Journal of medicinal chemistry (11.03.1999)
Published in Journal of medicinal chemistry (11.03.1999)
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Synthesis, Corticotropin-Releasing Factor Receptor Binding Affinity, and Pharmacokinetic Properties of Triazolo-, Imidazo-, and Pyrrolopyrimidines and -pyridines
Chorvat, Robert J, Bakthavatchalam, Rajagopal, Beck, James P, Gilligan, Paul J, Wilde, Richard G, Cocuzza, Anthony J, Hobbs, Frank W, Cheeseman, Robert S, Curry, Matthew, Rescinito, Joseph P, Krenitsky, Paul, Chidester, Dennis, Yarem, Jerry A, Klaczkiewicz, John D, Hodge, C. Nicholas, Aldrich, Paul E, Wasserman, Zelda R, Fernandez, Christine H, Zaczek, Robert, Fitzgerald, Lawrence W, Huang, Shiew-Mei, Shen, Helen L, Wong, Y. Nancy, Chien, Ben M, Quon, Check Y, Arvanitis, Argyrios
Published in Journal of medicinal chemistry (11.03.1999)
Published in Journal of medicinal chemistry (11.03.1999)
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Journal Article
4-Aryl-2-anilinopyrimidines as corticotropin-releasing hormone (CRH) antagonists
Cocuzza, Anthony J., Hobbs, Frank W., Arnold, Charles R., Chidester, Dennis R., Yarem, Jerry A., Culp, Steven, Fitzgerald, Lawrence, Gilligan, Paul J.
Published in Bioorganic & medicinal chemistry letters (05.04.1999)
Published in Bioorganic & medicinal chemistry letters (05.04.1999)
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Journal Article