Mapping, Structure and Modulation of PPI
Martino, Elisa, Chiarugi, Sara, Margheriti, Francesco, Garau, Gianpiero
Published in Frontiers in chemistry (07.10.2021)
Published in Frontiers in chemistry (07.10.2021)
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Journal Article
Crosslinked Chitosan Nanoparticles with Muco-Adhesive Potential for Intranasal Delivery Applications
Gagliardi, Mariacristina, Chiarugi, Sara, De Cesari, Chiara, Di Gregorio, Giulia, Diodati, Alessandra, Baroncelli, Laura, Cecchini, Marco, Tonazzini, Ilaria
Published in International journal of molecular sciences (01.04.2023)
Published in International journal of molecular sciences (01.04.2023)
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Journal Article
Development of potent dual PDK1/AurA kinase inhibitors for cancer therapy: Lead-optimization, structural insights, and ADME-Tox profile
Sestito, Simona, Bacci, Andrea, Chiarugi, Sara, Runfola, Massimiliano, Gado, Francesca, Margheritis, Eleonora, Gul, Sheraz, Riveiro, Maria E., Vazquez, Ramiro, Huguet, Samuel, Manera, Clementina, Rezai, Keyvan, Garau, Gianpiero, Rapposelli, Simona
Published in European journal of medicinal chemistry (15.12.2021)
Published in European journal of medicinal chemistry (15.12.2021)
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Journal Article
Hit-to-Lead Optimization of Mouse Trace Amine Associated Receptor 1 (mTAAR1) Agonists with a Diphenylmethane-Scaffold: Design, Synthesis, and Biological Study
Chiellini, Grazia, Nesi, Giulia, Sestito, Simona, Chiarugi, Sara, Runfola, Massimiliano, Espinoza, Stefano, Sabatini, Martina, Bellusci, Lorenza, Laurino, Annunziatina, Cichero, Elena, Gainetdinov, Raul R, Fossa, Paola, Raimondi, Laura, Zucchi, Riccardo, Rapposelli, Simona
Published in Journal of medicinal chemistry (10.11.2016)
Published in Journal of medicinal chemistry (10.11.2016)
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Journal Article
Novel Dual PDK1/AurK-A Inhibitors for Cancer Therapy: Med Chem Evolution and Crystallographic Investigation
Simona Sestito, Sara Chiarugi, Eleonora Margheritis, Massimiliano Runfola, Simone Bertini, Gianpiero Garau, Simona Rapposelli
Published in Proceedings (01.08.2019)
Published in Proceedings (01.08.2019)
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