Small-molecule inhibitors of FABP4/5 ameliorate dyslipidemia but not insulin resistance in mice with diet-induced obesity
Lan, Hong, Cheng, Cliff C., Kowalski, Timothy J., Pang, Ling, Shan, Lixin, Chuang, Cheng-Chi, Jackson, James, Rojas-Triana, Alberto, Bober, Loretta, Liu, Li, Voigt, Johannes, Orth, Peter, Yang, Xianshu, Shipps, Jr. Gerald W., Hedrick, Joseph A.
Published in Journal of lipid research (01.04.2011)
Published in Journal of lipid research (01.04.2011)
Get full text
Journal Article
Application of affinity selection-mass spectrometry assays to purification and affinity-based screening of the chemokine receptor CXCR4
Whitehurst, Charles E, Yao, Zhiping, Murphy, Denise, Zhang, Mingxuan, Taremi, Shane, Wojcik, Lisa, Strizki, Julie M, Bracken, Jack D, Cheng, Cliff C, Yang, Xianshu, Shipps, Jr, Gerald W, Ziebell, Michael, Nickbarg, Elliott
Published in Combinatorial chemistry & high throughput screening (01.07.2012)
Published in Combinatorial chemistry & high throughput screening (01.07.2012)
Get more information
Journal Article
Structure-based design and optimization of 2-aminothiazole-4-carboxamide as a new class of CHK1 inhibitors
Huang, Xiaohua, Cheng, Cliff C., Fischmann, Thierry O., Duca, José S., Richards, Matthew, Tadikonda, Praveen K., Reddy, Panduranga Adulla, Zhao, Lianyun, Arshad Siddiqui, M., Parry, David, Davis, Nicole, Seghezzi, Wolfgang, Wiswell, Derek, Shipps, Gerald W.
Published in Bioorganic & medicinal chemistry letters (01.05.2013)
Published in Bioorganic & medicinal chemistry letters (01.05.2013)
Get full text
Journal Article
Discovery and optimization of antibacterial AccC inhibitors
Cheng, Cliff C., Shipps, Gerald W., Yang, Zhiwei, Sun, Binyuan, Kawahata, Noriyuki, Soucy, Kyle A., Soriano, Aileen, Orth, Peter, Xiao, Li, Mann, Paul, Black, Todd
Published in Bioorganic & medicinal chemistry letters (01.12.2009)
Published in Bioorganic & medicinal chemistry letters (01.12.2009)
Get full text
Journal Article
Inhibitors of hepatitis C virus polymerase: Synthesis and characterization of novel 2-oxy-6-fluoro- N-(( S)-1-hydroxy-3-phenylpropan-2-yl)-benzamides
Cheng, Cliff C., Shipps, Gerald W., Yang, Zhiwei, Kawahata, Noriyuki, Lesburg, Charles A., Duca, José S., Bandouveres, Jamie, Bracken, Jack D., Jiang, Chuan-kui, Agrawal, Sony, Ferrari, Eric, Huang, H.-C.
Published in Bioorganic & medicinal chemistry letters (01.04.2010)
Published in Bioorganic & medicinal chemistry letters (01.04.2010)
Get full text
Journal Article
Discovery and Hit-to-Lead Optimization of Non-ATP Competitive MK2 (MAPKAPK2) Inhibitors
Huang, Xiaohua, Shipps, Gerald W., Cheng, Cliff C., Spacciapoli, Peter, Zhang, Xingmin, McCoy, Mark A., Wyss, Daniel F., Yang, Xianshu, Achab, Abdelghani, Soucy, Kyle, Montavon, Donna K., Murphy, Denise M., Whitehurst, Charles E.
Published in ACS medicinal chemistry letters (11.08.2011)
Published in ACS medicinal chemistry letters (11.08.2011)
Get full text
Journal Article
Pyridine Carboxamides: Potent Palm Site Inhibitors of HCV NS5B Polymerase
Cheng, Cliff C, Huang, Xiaohua, Shipps, Gerald W, Wang, Yu-Sen, Wyss, Daniel F, Soucy, Kyle A, Jiang, Chuan-kui, Agrawal, Sony, Ferrari, Eric, He, Zhiqing, Huang, H.-C
Published in ACS medicinal chemistry letters (09.12.2010)
Published in ACS medicinal chemistry letters (09.12.2010)
Get full text
Journal Article
Inhibitors of the lipid phosphatase SHIP2 discovered by high-throughput affinity selection-mass spectrometry screening of combinatorial libraries
Annis, D Allen, Cheng, Cliff C, Chuang, Cheng-Chi, McCarter, John D, Nash, Huw M, Nazef, Naim, Rowe, Todd, Kurzeja, Robert J M, Shipps, Jr, Gerald W
Published in Combinatorial chemistry & high throughput screening (01.09.2009)
Published in Combinatorial chemistry & high throughput screening (01.09.2009)
Get more information
Journal Article
Discovery and characterization of orthosteric and allosteric muscarinic M2 acetylcholine receptor ligands by affinity selection-mass spectrometry
Whitehurst, Charles E, Nazef, Naim, Annis, D Allen, Hou, Yongmin, Murphy, Denise M, Spacciapoli, Peter, Yao, Zhiping, Ziebell, Michael R, Cheng, Cliff C, Shipps, Jr, Gerald W, Felsch, Jason S, Lau, David, Nash, Huw M
Published in Journal of biomolecular screening (01.03.2006)
Published in Journal of biomolecular screening (01.03.2006)
Get full text
Journal Article
2-AMINOTHIAZOLE-4-CARBOXYLIC AMIDES AS PROTEIN KINASE INHIBITORS
FISCHMANN THIERRY O, DUCA JOSE S, CHENG CLIFF C, RICHARDS MATTHEW, SHIPPS GERALD W. JR, HUANG XIAOHUA
Year of Publication 09.07.2009
Get full text
Year of Publication 09.07.2009
Patent
2-AMIN0THIAZ0LE-4-CARB0XYLIC AMIDES AS PROTEIN KINASE INHIBITORS
FISCHMANN THIERRY O, TADIKONDA PRAVEEN K, GUZI TIMOTHY J, ZENG HONGBO, REDDY PANDURANGA A, TANG SHUYI, ZHAO LIANYUN, HUANG XIAOHUA, TORRES LUIS E, DWYER MICHAEL P, DUCA JOSE S, SUN BINYUAN, CHENG CLIFF C, SIDDIQUI M. ARSHAD, RICHARDS MATTHEW, SHIPPS GERALD W. JR, KEERTIKAR KARTIK M, WONG TZU T
Year of Publication 30.07.2009
Get full text
Year of Publication 30.07.2009
Patent
ANILINOPIPERAZINE DERIVATIVES AND METHODS OF USE THEREOF
FISCHMANN THIERRY O, TADIKONDA PRAVEEN K, GUZI TIMOTHY J, ZENG HONGBO, REDDY PANDURANGA A, LABROLI MARC M, HUANG XIAOHUA, DUCA JOSE S, SUN BINYUAN, POKER CORY, CHENG CLIFF C, SIDDIQUI M. ARSHAD, RICHARDS MATTHEW, SHIPPS GERALD W. JR, WONG TZU T
Year of Publication 09.07.2009
Get full text
Year of Publication 09.07.2009
Patent
Inhibitors of hepatitis C virus polymerase: Synthesis and characterization of novel 2-oxy-6-fluoro-N-((S)-1-hydroxy-3-phenylpropan-2-yl)-benzam ides
Cheng, Cliff C, Shipps, Gerald W, Yang, Zhiwei, Kawahata, Noriyuki, Lesburg, Charles A, Duca, Jose S, Bandouveres, Jamie, Bracken, Jack D, Jiang, Chuan-Kui, Agrawal, Sony, Ferrari, Eric, Huang, H-C
Published in Bioorganic & medicinal chemistry letters (01.04.2010)
Published in Bioorganic & medicinal chemistry letters (01.04.2010)
Get full text
Journal Article
THIAZOLE CARBOXAMIDE DERIVATIVES AND THEIR USE TO TREAT CANCER
HUANG, Xiaohua, CHENG, Cliff, C, RICHARDS, Matthew, SHIPPS, Gerald, W., Jr
Year of Publication 06.09.2017
Get full text
Year of Publication 06.09.2017
Patent
PYRAZOLO[1, 5-A]PYRIMIDINE DERIVATIVES AS MTOR INHIBITORS
SIDDIQUI, M., Arshad, TANG, Shuyi, DENG, Yongqi, CHENG, Cliff, C, RICHARDS, Matthew, ZHAO, Lianyun, SHIPPS, Gerald, W., Jr, MCRINER, Andrew, PATEL, Mehul, F, EKLOV, Brian, M, LIU, Duan, MANDAL, Amit, K, WRONA, Iwona, E, ZENG, Hongbo, SUN, Binyuan, ZHAO, Yinyan, REDDY, Panduranga, Adulla, NAN, Yang, MENG, Zhaoyang
Year of Publication 27.11.2019
Get full text
Year of Publication 27.11.2019
Patent
ANILINOPIPERAZINE DERIVATIVES AND METHODS OF USE THEREOF
SIDDIQUI, M., Arshad, POKER, Cory, CHENG, Cliff, C, RICHARDS, Matthew, FISCHMANN, Thierry, O, SHIPPS, Gerald, W., Jr, REDDY, Panduranga, A, LABROLI, Marc, M, HUANG, Xiaohua, GUZI, Timothy, J, ZENG, Hongbo, SUN, Binyuan, DUCA, Jose, S, WONG, Tzu, T, TADIKONDA, Praveen, K
Year of Publication 08.03.2017
Get full text
Year of Publication 08.03.2017
Patent
INHIBITORS OF FATTY ACID BINDING PROTEIN (FABP)
ORTH, PETER, SHIPPS, JR., GERALD, W, SOUCY, KYLE, ANN, VOIGT, JOHANNES, H, CHENG, CLIFF, C, HUANG, XIAOHUA, ACHAB, ABDELGHANI, ABE
Year of Publication 06.01.2016
Get full text
Year of Publication 06.01.2016
Patent