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Just, Stefan, Chenard, Bertrand L, Ceci, Angelo, Strassmaier, Timothy, Chong, Jayhong A, Blair, Nathaniel T, Gallaschun, Randall J, Del Camino, Donato, Cantin, Susan, D'Amours, Marc, Eickmeier, Christian, Fanger, Christopher M, Hecker, Carsten, Hessler, David P, Hengerer, Bastian, Kroker, Katja S, Malekiani, Sam, Mihalek, Robert, McLaughlin, Joseph, Rast, Georg, Witek, JoAnn, Sauer, Achim, Pryce, Christopher R, Moran, Magdalene M
Published in PloS one (31.01.2018)
Published in PloS one (31.01.2018)
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Discovery of Novel 6,6-Heterocycles as Transient Receptor Potential Vanilloid (TRPV1) Antagonists
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Published in Journal of medicinal chemistry (22.04.2010)
Published in Journal of medicinal chemistry (22.04.2010)
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Atropisomeric quinazolin-4-one derivatives are potent noncompetitive α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptor antagonists
WELCH, W. M, EWING, F. E, CRITCHETT, D, LAZZARO, J, GANONG, A. H, DEVRIES, K. M, STAIGERS, T. L, CHENARD, B. L, HUANG, J, MENNITI, F. S, PAGNOZZI, M. J, KELLY, K, SEYMOUR, P. A, GUANOWSKY, V, GUHAN, S, GUINN, M. R
Published in Bioorganic & medicinal chemistry letters (22.01.2001)
Published in Bioorganic & medicinal chemistry letters (22.01.2001)
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Quinazolin-4-one α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptor Antagonists: Structure−Activity Relationship of the C-2 Side Chain Tether
Chenard, Bertrand L, Welch, Willard M, Blake, James F, Butler, Todd W, Reinhold, Anthony, Ewing, Frank E, Menniti, Frank S, Pagnozzi, Martin J
Published in Journal of medicinal chemistry (24.05.2001)
Published in Journal of medicinal chemistry (24.05.2001)
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Equilibration of the Oxidative Addition Product of Tetrakis(triphenylphosphine)palladium and Electron-Rich Aryl Halides Leads to Product Scrambling in the Stille Reaction
Segelstein, B. E, Butler, T. W, Chenard, B. L
Published in Journal of organic chemistry (01.01.1995)
Published in Journal of organic chemistry (01.01.1995)
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CP-101,606, an NR2B subunit selective NMDA receptor antagonist, inhibits NMDA and injury induced c-fos expression and cortical spreading depression in rodents
Menniti, Frank S, Pagnozzi, Martin J, Butler, Paul, Chenard, Bertrand L, Jaw-Tsai, Sarah S, Frost White, W
Published in Neuropharmacology (01.06.2000)
Published in Neuropharmacology (01.06.2000)
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Molecular Characterization of the Gerbil C5a Receptor and Identification of a Transmembrane Domain V Amino Acid That Is Crucial for Small Molecule Antagonist Interaction
Waters, Stephen M., Brodbeck, Robbin M., Steflik, Jeremy, Yu, Jianying, Baltazar, Carolyn, Peck, Amy E., Severance, Daniel, Zhang, Lu Yan, Currie, Kevin, Chenard, Bertrand L., Hutchison, Alan J., Maynard, George, Krause, James E.
Published in The Journal of biological chemistry (09.12.2005)
Published in The Journal of biological chemistry (09.12.2005)
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Functional characterization of CP-465,022, a selective, noncompetitive AMPA receptor antagonist
Lazzaro, J.T., Paternain, A.V., Lerma, J., Chenard, B.L., Ewing, F.E., Huang, J., Welch, W.M., Ganong, A.H., Menniti, F.S.
Published in Neuropharmacology (01.02.2002)
Published in Neuropharmacology (01.02.2002)
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Pyrido[2,3-b]pyrazines, discovery of TRPV1 antagonists with reduced potential for the formation of reactive metabolites
Hodgetts, Kevin J., Blum, Charles A., Caldwell, Timothy, Bakthavatchalam, Rajagopal, Zheng, Xiaozhang, Capitosti, Scott, Krause, James E., Cortright, Daniel, Crandall, Marci, Murphy, Beth Ann, Boyce, Susan, Brian Jones, A., Chenard, Bertrand L.
Published in Bioorganic & medicinal chemistry letters (01.08.2010)
Published in Bioorganic & medicinal chemistry letters (01.08.2010)
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(1S,2S)-1-(4-Hydroxyphenyl)-2-(4-hydroxy-4-phenylpiperidino)-1-propanol: A Potent New Neuroprotectant Which Blocks N-Methyl-D-Aspartate Responses
Chenard, B. L, Bordner, J, Butler, T. W, Chambers, L. K, Collins, M. A, De Costa, D. L, Ducat, M. F, Dumont, M. L, Fox, C. B
Published in Journal of medicinal chemistry (01.08.1995)
Published in Journal of medicinal chemistry (01.08.1995)
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CP-465,022, a selective noncompetitive AMPA receptor antagonist, blocks AMPA receptors but is not neuroprotective in vivo
MENNITI, Frank S, BUCHAN, Alistair M, CHENARD, Bertrand L, CRITCHETT, Donald J, GANONG, Alan H, GUANOWSKY, Victor, SEYMOUR, Patricia A, WELCH, Willard M
Published in Stroke (1970) (2003)
Published in Stroke (1970) (2003)
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C-reactive protein or erythrocyte sedimentation rate results reliably exclude invasive bacterial infections
Paydar-Darian, Niloufar, Kimia, Amir A., Monuteaux, Michael C., Michelson, Kenneth A., Landschaft, Assaf, Maulden, Alexandra B., Chenard, Rachel L., Nigrovic, Lise E.
Published in The American journal of emergency medicine (01.08.2019)
Published in The American journal of emergency medicine (01.08.2019)
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Methaqualone derivatives are potent noncompetitive AMPA receptor antagonists
CHENARD, B. L, MENNITI, F. S, PAGNOZZI, M. J, SHENK, K. D, EWING, F. E, WELCH, W. M
Published in Bioorganic & medicinal chemistry letters (05.06.2000)
Published in Bioorganic & medicinal chemistry letters (05.06.2000)
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Characterization of the binding site for a novel class of noncompetitive alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptor antagonists
Menniti, F S, Chenard, B L, Collins, M B, Ducat, M F, Elliott, M L, Ewing, F E, Huang, J I, Kelly, K A, Lazzaro, J T, Pagnozzi, M J, Weeks, J L, Welch, W M, White, W F
Published in Molecular pharmacology (01.12.2000)
Published in Molecular pharmacology (01.12.2000)
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Neuroprotective effects of the N-methyl-D-aspartate receptor antagonists ifenprodil and SL-82,0715 on hippocampal cells in culture
SHALABY, I. A, CHENARD, B. L, PROCHNIAK, M. A, BUTLER, T. W
Published in The Journal of pharmacology and experimental therapeutics (01.02.1992)
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Published in The Journal of pharmacology and experimental therapeutics (01.02.1992)
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Water intake and wastage at nipple drinkers by growing-finishing pigs
Li, Y. Z, Chénard, L, Lemay, S. P, Gonyou, H. W
Published in Journal of animal science (01.06.2005)
Published in Journal of animal science (01.06.2005)
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(3R,4S)-3-[4-(4-Fluorophenyl)-4-hydroxypiperidin-1-yl]chroman-4,7-diol: A Conformationally Restricted Analogue of the NR2B Subtype-Selective NMDA Antagonist (1S,2S)-1-(4-Hydroxyphenyl)-2- (4-hydroxy-4-phenylpiperidino)-1-propanol
Butler, Todd W, Blake, James F, Bordner, Jon, Butler, Paul, Chenard, Bertrand L, Collins, Mary A, DeCosta, Debra, Ducat, Mary J, Eisenhard, Michael E, Menniti, Frank S, Pagnozzi, Martin J, Sands, Steven B, Segelstein, Barbara E, Volberg, Walter, White, W. Frost, Zhao, Dayao
Published in Journal of medicinal chemistry (26.03.1998)
Published in Journal of medicinal chemistry (26.03.1998)
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