Discovery of I‑BRD9, a Selective Cell Active Chemical Probe for Bromodomain Containing Protein 9 Inhibition
Theodoulou, Natalie H, Bamborough, Paul, Bannister, Andrew J, Becher, Isabelle, Bit, Rino A, Che, Ka Hing, Chung, Chun-wa, Dittmann, Antje, Drewes, Gerard, Drewry, David H, Gordon, Laurie, Grandi, Paola, Leveridge, Melanie, Lindon, Matthew, Michon, Anne-Marie, Molnar, Judit, Robson, Samuel C, Tomkinson, Nicholas C. O, Kouzarides, Tony, Prinjha, Rab K, Humphreys, Philip G
Published in Journal of medicinal chemistry (25.02.2016)
Published in Journal of medicinal chemistry (25.02.2016)
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A Chemical Probe for the ATAD2 Bromodomain
Bamborough, Paul, Chung, Chun-wa, Demont, Emmanuel H., Furze, Rebecca C., Bannister, Andrew J., Che, Ka Hing, Diallo, Hawa, Douault, Clement, Grandi, Paola, Kouzarides, Tony, Michon, Anne-Marie, Mitchell, Darren J., Prinjha, Rab K., Rau, Christina, Robson, Samuel, Sheppard, Robert J., Upton, Richard, Watson, Robert J.
Published in Angewandte Chemie (International ed.) (12.09.2016)
Published in Angewandte Chemie (International ed.) (12.09.2016)
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A Selective Inhibitor and Probe of the Cellular Functions of Jumonji C Domain-Containing Histone Demethylases
Luo, Xuelai, Liu, Yongxiang, Kubicek, Stefan, Myllyharju, Johanna, Tumber, Anthony, Ng, Stanley, Che, Ka Hing, Podoll, Jessica, Heightman, Tom D, Oppermann, Udo, Schreiber, Stuart L, Wang, Xiang
Published in Journal of the American Chemical Society (22.06.2011)
Published in Journal of the American Chemical Society (22.06.2011)
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Linking of 2-Oxoglutarate and Substrate Binding Sites Enables Potent and Highly Selective Inhibition of JmjC Histone Demethylases
Woon, Esther C. Y., Tumber, Anthony, Kawamura, Akane, Hillringhaus, Lars, Ge, Wei, Rose, Nathan R., Ma, Jerome H. Y., Chan, Mun Chiang, Walport, Louise J., Che, Ka Hing, Ng, Stanley S., Marsden, Brian D., Oppermann, Udo, McDonough, Michael A., Schofield, Christopher J.
Published in Angewandte Chemie (International ed.) (13.02.2012)
Published in Angewandte Chemie (International ed.) (13.02.2012)
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canSAR: update to the cancer translational research and drug discovery knowledgebase
Mitsopoulos, Costas, Di Micco, Patrizio, Fernandez, Eloy Villasclaras, Dolciami, Daniela, Holt, Esty, Mica, Ioan L, Coker, Elizabeth A, Tym, Joseph E, Campbell, James, Che, Ka Hing, Ozer, Bugra, Kannas, Christos, Antolin, Albert A, Workman, Paul, Al-Lazikani, Bissan
Published in Nucleic Acids Research (08.01.2021)
Published in Nucleic Acids Research (08.01.2021)
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Imperfect interface of Beclin1 coiled-coil domain regulates homodimer and heterodimer formation with Atg14L and UVRAG
Li, Xiaohua, He, Liqiang, Che, Ka Hing, Funderburk, Sarah F, Pan, Lifeng, Pan, Nina, Zhang, Mingjie, Yue, Zhenyu, Zhao, Yanxiang
Published in Nature communications (07.02.2012)
Published in Nature communications (07.02.2012)
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Generation of a Selective Small Molecule Inhibitor of the CBP/p300 Bromodomain for Leukemia Therapy
Picaud, Sarah, Fedorov, Oleg, Thanasopoulou, Angeliki, Leonards, Katharina, Jones, Katherine, Meier, Julia, Olzscha, Heidi, Monteiro, Octovia, Martin, Sarah, Philpott, Martin, Tumber, Anthony, Filippakopoulos, Panagis, Yapp, Clarence, Wells, Christopher, Che, Ka Hing, Bannister, Andrew, Robson, Samuel, Kumar, Umesh, Parr, Nigel, Lee, Kevin, Lugo, Dave, Jeffrey, Philip, Taylor, Simon, Vecellio, Matteo L, Bountra, Chas, Brennan, Paul E, O'Mahony, Alison, Velichko, Sharlene, Müller, Susanne, Hay, Duncan, Daniels, Danette L, Urh, Marjeta, La Thangue, Nicholas B, Kouzarides, Tony, Prinjha, Rab, Schwaller, Jürg, Knapp, Stefan
Published in Cancer research (Chicago, Ill.) (01.12.2015)
Published in Cancer research (Chicago, Ill.) (01.12.2015)
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The roles of Jumonji-type oxygenases in human disease
Johansson, Catrine, Tumber, Anthony, Che, KaHing, Cain, Peter, Nowak, Rados aw, Gileadi, Carina, Oppermann, Udo
Published in Epigenomics (01.02.2014)
Published in Epigenomics (01.02.2014)
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Advances and challenges in understanding histone demethylase biology
Nowak, Radoslaw P, Tumber, Anthony, Johansson, Catrine, Che, Ka Hing, Brennan, Paul, Owen, Dafydd, Oppermann, Udo
Published in Current opinion in chemical biology (01.08.2016)
Published in Current opinion in chemical biology (01.08.2016)
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Journal Article
5-Carboxy-8-hydroxyquinoline is a Broad Spectrum 2-Oxoglutarate Oxygenase Inhibitor which Causes Iron Translocation
Hopkinson, Richard J, Tumber, Anthony, Yapp, Clarence, Chowdhury, Rasheduzzaman, Aik, WeiShen, Che, Ka Hing, Li, Xuan Shirley, Kristensen, Jan B L, King, Oliver N F, Chan, Mun Chiang, Yeoh, Kar Kheng, Choi, Hwanho, Walport, Louise J, Thinnes, Cyrille C, Bush, Jacob T, Lejeune, Clarisse, Rydzik, Anna M, Rose, Nathan R, Bagg, Eleanor A, McDonough, Michael A, Krojer, Tobias, Yue, Wyatt W, Ng, Stanley S, Olsen, Lars, Brennan, Paul E, Oppermann, Udo, Muller-Knapp, Susanne, Klose, Robert J, Ratcliffe, Peter J, Schofield, Christopher J, Kawamura, Akane
Published in Chemical science (Cambridge) (01.08.2013)
Published in Chemical science (Cambridge) (01.08.2013)
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Journal Article
Plant Growth Regulator Daminozide Is a Selective Inhibitor of Human KDM2/7 Histone Demethylases
Rose, Nathan R, Woon, Esther C. Y, Tumber, Anthony, Walport, Louise J, Chowdhury, Rasheduzzaman, Li, Xuan Shirley, King, Oliver N. F, Lejeune, Clarisse, Ng, Stanley S, Krojer, Tobias, Chan, Mun Chiang, Rydzik, Anna M, Hopkinson, Richard J, Che, Ka Hing, Daniel, Michelle, Strain-Damerell, Claire, Gileadi, Carina, Kochan, Grazyna, Leung, Ivanhoe K. H, Dunford, James, Yeoh, Kar Kheng, Ratcliffe, Peter J, Burgess-Brown, Nicola, von Delft, Frank, Muller, Susanne, Marsden, Brian, Brennan, Paul E, McDonough, Michael A, Oppermann, Udo, Klose, Robert J, Schofield, Christopher J, Kawamura, Akane
Published in Journal of medicinal chemistry (26.07.2012)
Published in Journal of medicinal chemistry (26.07.2012)
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Kruidenier et al. reply
Kruidenier, Laurens, Chung, Chun-wa, Cheng, Zhongjun, Liddle, John, Che, KaHing, Joberty, Gerard, Bantscheff, Marcus, Bountra, Chas, Bridges, Angela, Diallo, Hawa, Eberhard, Dirk, Hutchinson, Sue, Jones, Emma, Katso, Roy, Leveridge, Melanie, Mander, Palwinder K, Mosley, Julie, Ramirez-Molina, Cesar, Rowland, Paul, Schofield, Christopher J, Sheppard, Robert J, Smith, Julia E, Swales, Catherine, Tanner, Robert, Thomas, Pamela, Tumber, Anthony, Drewes, Gerard, Oppermann, Udo, Patel, Dinshaw J, Lee, Kevin, Wilson, David M
Published in Nature (London) (02.10.2014)
Published in Nature (London) (02.10.2014)
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Journal Article
A Chemical Probe for the ATAD2 Bromodomain
Bamborough, Paul, Chung, Chun-wa, Demont, Emmanuel H., Furze, Rebecca C., Bannister, Andrew J., Che, Ka Hing, Diallo, Hawa, Douault, Clement, Grandi, Paola, Kouzarides, Tony, Michon, Anne-Marie, Mitchell, Darren J., Prinjha, Rab K., Rau, Christina, Robson, Samuel, Sheppard, Robert J., Upton, Richard, Watson, Robert J.
Published in Angewandte Chemie (12.09.2016)
Published in Angewandte Chemie (12.09.2016)
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Journal Article
Linking of 2-Oxoglutarate and Substrate Binding Sites Enables Potent and Highly Selective Inhibition of JmjC Histone Demethylases
Woon, Esther C. Y., Tumber, Anthony, Kawamura, Akane, Hillringhaus, Lars, Ge, Wei, Rose, Nathan R., Ma, Jerome H. Y., Chan, Mun Chiang, Walport, Louise J., Che, Ka Hing, Ng, Stanley S., Marsden, Brian D., Oppermann, Udo, McDonough, Michael A., Schofield, Christopher J.
Published in Angewandte Chemie (13.02.2012)
Published in Angewandte Chemie (13.02.2012)
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Journal Article
Linking of 2‐Oxoglutarate and Substrate Binding Sites Enables Potent and Highly Selective Inhibition of JmjC Histone Demethylases
Woon, Esther C. Y., Tumber, Anthony, Kawamura, Akane, Hillringhaus, Lars, Ge, Wei, Rose, Nathan R., Ma, Jerome H. Y., Chan, Mun Chiang, Walport, Louise J., Che, Ka Hing, Ng, Stanley S., Marsden, Brian D., Oppermann, Udo, McDonough, Michael A., Schofield, Christopher J.
Published in Angewandte Chemie (13.02.2012)
Published in Angewandte Chemie (13.02.2012)
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