Synthesis and antimalarial activity of E-2-quinolinylbenzocycloalkanones
Charris, JE, Dominguez, JN, Gamboa, N, Rodrigues, Angel, JE
Published in European journal of medicinal chemistry (01.09.2005)
Published in European journal of medicinal chemistry (01.09.2005)
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Journal Article
Synthesis of quinolinyl chalcones and evaluation of their antimalarial activity
Domı́nguez, José N, Charris, Jaime E, Lobo, Gricela, Gamboa de Domı́nguez, Neira, Moreno, Marı́a M, Riggione, Flavia, Sanchez, Erlinda, Olson, Jed, Rosenthal, Philip J
Published in European journal of medicinal chemistry (01.06.2001)
Published in European journal of medicinal chemistry (01.06.2001)
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Journal Article
Synthesis and theoretical study of 2-amino-2,3,3a,4,5,6-hexahydro-1H-phenalene and its biological evaluation on central dopaminergic system
Angel-Guio, JE, Charris, JE, Perez, J, de Perez, ZD, Compagnone, R, Israel, A, Orfila, L, de Angel, BM, Lopez, SE, Rodriguez, L, Caldera, J, de Baez, EM
Published in Farmaco (Società chimica italiana : 1989) (01.09.2000)
Published in Farmaco (Società chimica italiana : 1989) (01.09.2000)
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Journal Article
Synthesis and inhibitory activity of dimethylamino-chalcone derivatives on the induction of nitric oxide synthase
Rojas, Javier, Domı́nguez, José N, Charris, Jaime E, Lobo, Gricela, Payá, Miguel, Ferrándiz, M.Luisa
Published in European journal of medicinal chemistry (01.08.2002)
Published in European journal of medicinal chemistry (01.08.2002)
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Journal Article
4-dimethylamino-3′,4′-dimethoxychalcone downregulates iNOS expression and exerts anti-inflammatory effects
Herencia, Felipe, Ferrándiz, Maria Luisa, Ubeda, Amalia, Guillén, Isabel, Dominguez, José N, Charris, Jaime E, Lobo, Gricela M, Alcaraz, Maria José
Published in Free radical biology & medicine (2001)
Published in Free radical biology & medicine (2001)
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Journal Article
Novel anti-inflammatory chalcone derivatives inhibit the induction of nitric oxide synthase and cyclooxygenase-2 in mouse peritoneal macrophages
Herencia, Felipe, Ferrándiz, M.Luisa, Ubeda, Amalia, Guillén, Isabel, Dominguez, José N., Charris, Jaime E., Lobo, Gricela M., Alcaraz, M.José
Published in FEBS letters (18.06.1999)
Published in FEBS letters (18.06.1999)
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Journal Article
H-1 and C-13 NMR spectral characterization of some antimalarial in vitro 2,4-diamino-10-methylpyrimido[4,5-b]-5-quinolone derivatives
Charris, JE, Dominguez, JN, Gamboa, N, Angel, J, Pina, N, Guerra, M, Michelena, E, Lopez, SE
Published in Magnetic resonance in chemistry (01.07.2002)
Published in Magnetic resonance in chemistry (01.07.2002)
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Journal Article
H-1 and C-13 NMR spectral characterization of some antimalarial in vitro - 3-amino-9-methyl-1H-pyrazolo[3,4-b]-4-quinolones
Charris, JE, Dominguez, JN, Lobo, G, Cordero, MI, Lopez, SE, Mendez, B, Pekerar, S, Riggione, F
Published in Magnetic resonance in chemistry (01.12.2000)
Published in Magnetic resonance in chemistry (01.12.2000)
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Journal Article
Crystal structure of 3-hydroxy-4-cyano-5-methylthiopyrazole, C5H5N3OS
Capparelli, M. V., Avila, R., Charris, J. E., Domínguez, J. N.
Published in Zeitschrift für Kristallographie. New crystal structures (01.03.2003)
Published in Zeitschrift für Kristallographie. New crystal structures (01.03.2003)
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Journal Article
Perfil Dopaminérgico del compuesto 2-aminoindano N-aralquíl sustituido
Angel-Guío, JE, Charris, JE, Israel, Migliore de Angel, Suárez-Roca, Garrido, MR, López, SE, Díaz, Ferrer, Michelena de Báez, Rodríguez, LJ, Silva, Moronta, Espinoza, Quintero
Published in Archivos venezolanos de farmacología y terapéutica (01.07.2004)
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Published in Archivos venezolanos de farmacología y terapéutica (01.07.2004)
Journal Article
Synthesis and antimalarial activity of substituted pyrazole derivatives
Dominguez, JN, Charris, JE, Caparelli, M, Riggione, F
Published in Arzneimittel-Forschung (01.01.2002)
Published in Arzneimittel-Forschung (01.01.2002)
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Conformational theoretical study of substituted and non-substituted N-aralkyl-2-aminoindans and its relation with dopaminergic activity
Rodrı́guez, Leonardo J, Medina, Yolibeth, Suárez-Roca, Heberto, de Angel, Biagina Migliore, Israel, Anita, Charris, Jaime E, E. López, Simón, Caldera, José A, Angel-Guio, Jorge E
Published in Journal of molecular structure. Theochem (30.09.2003)
Published in Journal of molecular structure. Theochem (30.09.2003)
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Journal Article
N-aralkyl substitution of 2-aminoindans - Synthesis and their inotropic and chronotropic activity in isolated guinea pig atria
Perez, JA, Dominguez, JN, Angel, JE, de Perez, ZD, Salazar-Bookaman, MM, Acosta, H, Charris, JE
Published in Arzneimittel-Forschung (01.11.1997)
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Published in Arzneimittel-Forschung (01.11.1997)
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