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Published in PLoS pathogens (02.12.2020)
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PI(4,5)P2 controls plasma membrane PI4P and PS levels via ORP5/8 recruitment to ER–PM contact sites
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Published in The Journal of cell biology (07.05.2018)
Published in The Journal of cell biology (07.05.2018)
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Published in Nature communications (20.04.2023)
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Structure-based design and modular synthesis of novel PI4K class II inhibitors bearing a 4-aminoquinazoline scaffold
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Published in Bioorganic & medicinal chemistry letters (15.11.2022)
Published in Bioorganic & medicinal chemistry letters (15.11.2022)
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Design, synthesis and evaluation of novel thieno[2,3d]pyrimidine derivatives as potent and specific RIPK2 inhibitors
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Published in Bioorganic & medicinal chemistry letters (01.01.2024)
Published in Bioorganic & medicinal chemistry letters (01.01.2024)
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Phosphatidylinositol 4-kinase IIIβ (PI4KB) forms highly flexible heterocomplexes that include ACBD3, 14-3-3, and Rab11 proteins
Chalupska, Dominika, Różycki, Bartosz, Humpolickova, Jana, Faltova, Lenka, Klima, Martin, Boura, Evzen
Published in Scientific reports (24.01.2019)
Published in Scientific reports (24.01.2019)
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Exploring positions 6 and 7 of a quinazoline-based scaffold leads to changes in selectivity and potency towards RIPK2/3 kinases
Misehe, Mbilo, Matoušová, Marika, Dvořáková, Alexandra, Hercík, Kamil, Škach, Kryštof, Chalupská, Dominika, Dejmek, Milan, Šála, Michal, Hájek, Miroslav, Boura, Evzen, Mertlíková-Kaiserová, Helena, Nencka, Radim
Published in European journal of medicinal chemistry (15.11.2023)
Published in European journal of medicinal chemistry (15.11.2023)
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Antiviral Properties of the NSAID Drug Naproxen Targeting the Nucleoprotein of SARS-CoV-2 Coronavirus
Terrier, Olivier, Dilly, Sébastien, Pizzorno, Andrés, Chalupska, Dominika, Humpolickova, Jana, Bouřa, Evžen, Berenbaum, Francis, Quideau, Stéphane, Lina, Bruno, Fève, Bruno, Adnet, Frédéric, Sabbah, Michèle, Rosa-Calatrava, Manuel, Maréchal, Vincent, Henri, Julien, Slama-Schwok, Anny
Published in Molecules (Basel, Switzerland) (29.04.2021)
Published in Molecules (Basel, Switzerland) (29.04.2021)
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Structural insights and in vitro reconstitution of membrane targeting and activation of human PI4KB by the ACBD3 protein
Klima, Martin, Tóth, Dániel J, Hexnerova, Rozalie, Baumlova, Adriana, Chalupska, Dominika, Tykvart, Jan, Rezabkova, Lenka, Sengupta, Nivedita, Man, Petr, Dubankova, Anna, Humpolickova, Jana, Nencka, Radim, Veverka, Vaclav, Balla, Tamas, Boura, Evzen
Published in Scientific reports (24.03.2016)
Published in Scientific reports (24.03.2016)
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Localization of SARS-CoV-2 Capping Enzymes Revealed by an Antibody against the nsp10 Subunit
Horova, Vladimira, Landova, Barbora, Hodek, Jan, Chalupsky, Karel, Krafcikova, Petra, Chalupska, Dominika, Duchoslav, Vojtech, Weber, Jan, Boura, Evzen, Klima, Martin
Published in Viruses (29.07.2021)
Published in Viruses (29.07.2021)
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Convergent evolution in the mechanisms of ACBD3 recruitment to picornavirus replication sites
Horova, Vladimira, Lyoo, Heyrhyoung, Różycki, Bartosz, Chalupska, Dominika, Smola, Miroslav, Humpolickova, Jana, Strating, Jeroen R P M, van Kuppeveld, Frank J M, Boura, Evzen, Klima, Martin
Published in PLoS pathogens (05.08.2019)
Published in PLoS pathogens (05.08.2019)
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A large scale high-throughput screen identifies chemical inhibitors of phosphatidylinositol 4-kinase type II alpha[S]
Sengupta, Nivedita, Jović, Marko, Barnaeva, Elena, Kim, David W., Hu, Xin, Southall, Noel, Dejmek, Milan, Mejdrova, Ivana, Nencka, Radim, Baumlova, Adriana, Chalupska, Dominika, Boura, Evzen, Ferrer, Marc, Marugan, Juan, Balla, Tamas
Published in Journal of lipid research (01.03.2019)
Published in Journal of lipid research (01.03.2019)
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Adaptation of an L-proline adenylation domain to use 4-propyl-L-proline in the evolution of lincosamide biosynthesis
Kadlčík, Stanislav, Kučera, Tomáš, Chalupská, Dominika, Gažák, Radek, Koběrská, Markéta, Ulanová, Dana, Kopecký, Jan, Kutejová, Eva, Najmanová, Lucie, Janata, Jiří
Published in PloS one (27.12.2013)
Published in PloS one (27.12.2013)
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Single-site mutations in the carboxyltransferase domain of plastid acetyl-CoA carboxylase confer resistance to grass-specific herbicides
Liu, Wenjie, Harrison, Dion K, Chalupska, Dominika, Gornicki, Piotr, O'Donnell, Chris C, Adkins, Steve W, Haselkorn, Robert, Williams, Richard R
Published in Proceedings of the National Academy of Sciences - PNAS (27.02.2007)
Published in Proceedings of the National Academy of Sciences - PNAS (27.02.2007)
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Discovery of highly potent SARS-CoV-2 nsp14 methyltransferase inhibitors based on adenosine 5′-carboxamides
Kocek, Hugo, Chalupská, Dominika, Dejmek, Milan, Dvořáková, Alexandra, Zgarbová, Michala, Šála, Michal, Chalupský, Karel, Krafčíková, Petra, Otava, Tomáš, Drexler, Matúš, Procházková, Eliška, Klepetářová, Blanka, Štefek, Milan, Kozic, Ján, Mertlíková-Kaiserová, Helena, Boura, Evzen, Weber, Jan, Nencka, Radim
Published in RSC medicinal chemistry (01.08.2024)
Published in RSC medicinal chemistry (01.08.2024)
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Norbornane-based nucleoside and nucleotide analogues locked in North conformation
Dejmek, Milan, Šála, Michal, Hřebabecký, Hubert, Dračínský, Martin, Procházková, Eliška, Chalupská, Dominika, Klíma, Martin, Plačková, Pavla, Hájek, Miroslav, Andrei, Graciela, Naesens, Lieve, Leyssen, Pieter, Neyts, Johan, Balzarini, Jan, Boura, Evzen, Nencka, Radim
Published in Bioorganic & medicinal chemistry (01.01.2015)
Published in Bioorganic & medicinal chemistry (01.01.2015)
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Recombinant yeast screen for new inhibitors of human acetyl-CoA carboxylase 2 identifies potential drugs to treat obesity
Marjanovic, Jasmina, Chalupska, Dominika, Patenode, Caroline, Coster, Adam, Arnold, Evan, Ye, Alice, Anesi, George, Lu, Ying, Okun, Ilya, Tkachenko, Sergey, Haselkorn, Robert, Gornicki, Piotr
Published in Proceedings of the National Academy of Sciences - PNAS (18.05.2010)
Published in Proceedings of the National Academy of Sciences - PNAS (18.05.2010)
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Rational Design of Novel Highly Potent and Selective Phosphatidylinositol 4‑Kinase IIIβ (PI4KB) Inhibitors as Broad-Spectrum Antiviral Agents and Tools for Chemical Biology
Mejdrová, Ivana, Chalupská, Dominika, Plačková, Pavla, Müller, Christin, Šála, Michal, Klíma, Martin, Baumlová, Adriana, Hřebabecký, Hubert, Procházková, Eliška, Dejmek, Milan, Strunin, Dmytro, Weber, Jan, Lee, Gary, Matoušová, Marika, Mertlíková-Kaiserová, Helena, Ziebuhr, John, Birkus, Gabriel, Boura, Evzen, Nencka, Radim
Published in Journal of medicinal chemistry (12.01.2017)
Published in Journal of medicinal chemistry (12.01.2017)
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Highly Selective Phosphatidylinositol 4‑Kinase IIIβ Inhibitors and Structural Insight into Their Mode of Action
Mejdrová, Ivana, Chalupská, Dominika, Kögler, Martin, Šála, Michal, Plačková, Pavla, Baumlová, Adriana, Hřebabecký, Hubert, Procházková, Eliška, Dejmek, Milan, Guillon, Rémi, Strunin, Dmytro, Weber, Jan, Lee, Gary, Birkus, Gabriel, Mertlíková-Kaiserová, Helena, Boura, Evzen, Nencka, Radim
Published in Journal of medicinal chemistry (14.05.2015)
Published in Journal of medicinal chemistry (14.05.2015)
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Structural and functional insights in flavivirus NS5 proteins gained by the structure of Ntaya virus polymerase and methyltransferase
Krejčová, Kateřina, Krafcikova, Petra, Klima, Martin, Chalupska, Dominika, Chalupsky, Karel, Zilecka, Eva, Boura, Evzen
Published in Structure (London) (08.08.2024)
Published in Structure (London) (08.08.2024)
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