Open saccharin-based secondary sulfonamides as potent and selective inhibitors of cancer-related carbonic anhydrase IX and XII isoforms
D'Ascenzio, Melissa, Guglielmi, Paolo, Carradori, Simone, Secci, Daniela, Florio, Rosalba, Mollica, Adriano, Ceruso, Mariangela, Akdemir, Atilla, Sobolev, Anatoly P., Supuran, Claudiu T.
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2017)
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2017)
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Journal Article
Inhibition studies of new ureido-substituted sulfonamides incorporating a GABA moiety against human carbonic anhydrase isoforms I–XIV
Ceruso, Mariangela, Antel, Sabrina, Vullo, Daniela, Scozzafava, Andrea, Supuran, Claudiu T.
Published in Bioorganic & medicinal chemistry (15.12.2014)
Published in Bioorganic & medicinal chemistry (15.12.2014)
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Journal Article
Inhibition of the α-carbonic anhydrase from Vibrio cholerae with amides and sulfonamides incorporating imidazole moieties
De Vita, Daniela, Angeli, Andrea, Pandolfi, Fabiana, Bortolami, Martina, Costi, Roberta, Di Santo, Roberto, Suffredini, Elisabetta, Ceruso, Mariangela, Del Prete, Sonia, Capasso, Clemente, Scipione, Luigi, Supuran, Claudiu T.
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2017)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2017)
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Journal Article
Aryl-4,5-dihydro-1H-pyrazole-1-carboxamide Derivatives Bearing a Sulfonamide Moiety Show Single-digit Nanomolar-to-Subnanomolar Inhibition Constants against the Tumor-associated Human Carbonic Anhydrases IX and XII
Hargunani, Priya, Tadge, Nikhil, Ceruso, Mariangela, Leitans, Janis, Kazaks, Andris, Tars, Kaspars, Gratteri, Paola, Supuran, Claudiu T., Nocentini, Alessio, Toraskar, Mrunmayee P.
Published in International journal of molecular sciences (01.04.2020)
Published in International journal of molecular sciences (01.04.2020)
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Journal Article
4-Functionalized 1,3-diarylpyrazoles bearing 6-aminosulfonylbenzothiazole moiety as potent inhibitors of carbonic anhydrase isoforms hCA I, II, IX and XII
SitaRam, Ceruso, Mariangela, Khloya, Poonam, Supuran, Claudiu T., Sharma, Pawan K.
Published in Bioorganic & medicinal chemistry (15.12.2014)
Published in Bioorganic & medicinal chemistry (15.12.2014)
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Journal Article
Inhibition studies of Brucella suis β-carbonic anhydrases with a series of 4-substituted pyridine-3-sulphonamides
Monti, Simona Maria, Meccariello, Angela, Ceruso, Mariangela, Szafrański, Krzysztof, Sławiński, Jarosław, Supuran, Claudiu T.
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2018)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2018)
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Journal Article
Click-tailed coumarins with potent and selective inhibitory action against the tumor-associated carbonic anhydrases IX and XII
Nocentini, Alessio, Carta, Fabrizio, Ceruso, Mariangela, Bartolucci, Gianluca, Supuran, Claudiu T.
Published in Bioorganic & medicinal chemistry (01.11.2015)
Published in Bioorganic & medicinal chemistry (01.11.2015)
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Journal Article
Benzenesulfonamides Incorporating Flexible Triazole Moieties Are Highly Effective Carbonic Anhydrase Inhibitors: Synthesis and Kinetic, Crystallographic, Computational, and Intraocular Pressure Lowering Investigations
Nocentini, Alessio, Ferraroni, Marta, Carta, Fabrizio, Ceruso, Mariangela, Gratteri, Paola, Lanzi, Cecilia, Masini, Emanuela, Supuran, Claudiu T
Published in Journal of medicinal chemistry (08.12.2016)
Published in Journal of medicinal chemistry (08.12.2016)
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Journal Article
Discovery of 4‑Hydroxy-3-(3-(phenylureido)benzenesulfonamides as SLC-0111 Analogues for the Treatment of Hypoxic Tumors Overexpressing Carbonic Anhydrase IX
Bozdag, Murat, Carta, Fabrizio, Ceruso, Mariangela, Ferraroni, Marta, McDonald, Paul C, Dedhar, Shoukat, Supuran, Claudiu T
Published in Journal of medicinal chemistry (26.07.2018)
Published in Journal of medicinal chemistry (26.07.2018)
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Journal Article
Geographical characterization by MAE-HPLC and NIR methodologies and carbonic anhydrase inhibition of Saffron components
Nescatelli, Riccardo, Carradori, Simone, Marini, Federico, Caponigro, Vicky, Bucci, Remo, De Monte, Celeste, Mollica, Adriano, Mannina, Luisa, Ceruso, Mariangela, Supuran, Claudiu T., Secci, Daniela
Published in Food chemistry (15.04.2017)
Published in Food chemistry (15.04.2017)
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Journal Article
Overexpression of the transmembrane carbonic anhydrase isoforms IX and XII in the inflamed synovium
Margheri, Francesca, Ceruso, Mariangela, Carta, Fabrizio, Laurenzana, Anna, Maggi, Laura, Lazzeri, Simone, Simonini, Gabriele, Annunziato, Francesco, Del Rosso, Mario, Supuran, Claudiu T., Cimaz, Rolando
Published in Journal of enzyme inhibition and medicinal chemistry (04.11.2016)
Published in Journal of enzyme inhibition and medicinal chemistry (04.11.2016)
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Journal Article
7-Aryl-triazolyl-substituted sulfocoumarins are potent, selective inhibitors of the tumor-associated carbonic anhydrase IX and XII
Nocentini, Alessio, Ceruso, Mariangela, Carta, Fabrizio, Supuran, Claudiu T.
Published in Journal of enzyme inhibition and medicinal chemistry (01.11.2016)
Published in Journal of enzyme inhibition and medicinal chemistry (01.11.2016)
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Journal Article
Synthesis of 4-sulfamoylphenyl-benzylamine derivatives with inhibitory activity against human carbonic anhydrase isoforms I, II, IX and XII
Durgun, Mustafa, Turkmen, Hasan, Ceruso, Mariangela, Supuran, Claudiu T.
Published in Bioorganic & medicinal chemistry (01.03.2016)
Published in Bioorganic & medicinal chemistry (01.03.2016)
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Journal Article
Synthesis of Schiff base derivatives of 4-(2-aminoethyl)-benzenesulfonamide with inhibitory activity against carbonic anhydrase isoforms I, II, IX and XII
Durgun, Mustafa, Turkmen, Hasan, Ceruso, Mariangela, Supuran, Claudiu T.
Published in Bioorganic & medicinal chemistry letters (01.06.2015)
Published in Bioorganic & medicinal chemistry letters (01.06.2015)
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Journal Article
Exploring new Probenecid-based carbonic anhydrase inhibitors: Synthesis, biological evaluation and docking studies
Mollica, Adriano, Costante, Roberto, Akdemir, Atilla, Carradori, Simone, Stefanucci, Azzurra, Macedonio, Giorgia, Ceruso, Mariangela, Supuran, Claudiu T.
Published in Bioorganic & medicinal chemistry (01.09.2015)
Published in Bioorganic & medicinal chemistry (01.09.2015)
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Journal Article
Design, synthesis and evaluation of N-substituted saccharin derivatives as selective inhibitors of tumor-associated carbonic anhydrase XII
D’Ascenzio, Melissa, Carradori, Simone, De Monte, Celeste, Secci, Daniela, Ceruso, Mariangela, Supuran, Claudiu T.
Published in Bioorganic & medicinal chemistry (15.03.2014)
Published in Bioorganic & medicinal chemistry (15.03.2014)
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Journal Article
Discovery of β‑Adrenergic Receptors Blocker–Carbonic Anhydrase Inhibitor Hybrids for Multitargeted Antiglaucoma Therapy
Nocentini, Alessio, Ceruso, Mariangela, Bua, Silvia, Lomelino, Carrie L, Andring, Jacob T, McKenna, Robert, Lanzi, Cecilia, Sgambellone, Silvia, Pecori, Riccardo, Matucci, Rosanna, Filippi, Luca, Gratteri, Paola, Carta, Fabrizio, Masini, Emanuela, Selleri, Silvia, Supuran, Claudiu T
Published in Journal of medicinal chemistry (28.06.2018)
Published in Journal of medicinal chemistry (28.06.2018)
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