Reconstitution of the Ataxia-Telangiectasia Cellular Phenotype With Lentiviral Vectors
Carranza, Diana, Torres-Rusillo, Sara, Ceballos-Pérez, Gloria, Blanco-Jimenez, Eva, Muñoz-López, Martin, García-Pérez, José L, Molina, Ignacio J
Published in Frontiers in immunology (20.11.2018)
Published in Frontiers in immunology (20.11.2018)
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Journal Article
Pharmacophore Identification and Structure–Activity Relationship Analysis of a Series of Substituted Azaindoles as Inhibitors of Trypanosoma brucei
Ferrins, Lori, Diaz, Rosario, Cordon-Obras, Carlos, Rojas-Barros, Domingo, Quotadamo, Antonio, Oehme, Daniel P., Ceballos-Pérez, Gloria, Swaminathan, Uma, Pérez-Moreno, Guiomar, Bosch-Navarrete, Cristina, García-Hernández, Raquel, Gomez-Liñan, Claudia, Saura, Andreu, Ruiz-Perez, Luis Miguel, Gamarro, Francisco, Martinez-Martinez, Maria Santos, Manzano, Pilar, González-Pacanowska, Dolores, Navarro, Miguel, Pollastri, Michael P.
Published in Journal of medicinal chemistry (22.08.2024)
Published in Journal of medicinal chemistry (22.08.2024)
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Journal Article
Selectivity and Physicochemical Optimization of Repurposed Pyrazolo[1,5‑b]pyridazines for the Treatment of Human African Trypanosomiasis
Tear, Westley F, Bag, Seema, Diaz-Gonzalez, Rosario, Ceballos-Pérez, Gloria, Rojas-Barros, Domingo I, Cordon-Obras, Carlos, Pérez-Moreno, Guiomar, García-Hernández, Raquel, Martinez-Martinez, Maria Santos, Ruiz-Perez, Luis Miguel, Gamarro, Francisco, Gonzalez Pacanowska, Dolores, Caffrey, Conor R, Ferrins, Lori, Manzano, Pilar, Navarro, Miguel, Pollastri, Michael P
Published in Journal of medicinal chemistry (23.01.2020)
Published in Journal of medicinal chemistry (23.01.2020)
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Journal Article
Lead Optimization of 3,5-Disubstituted-7-Azaindoles for the Treatment of Human African Trypanosomiasis
Klug, Dana M, Mavrogiannaki, Eftychia M, Forbes, Katherine C, Silva, Lisseth, Diaz-Gonzalez, Rosario, Pérez-Moreno, Guiomar, Ceballos-Pérez, Gloria, Garcia-Hernández, Raquel, Bosch-Navarrete, Cristina, Cordón-Obras, Carlos, Gómez-Liñán, Claudia, Saura, Andreu, Momper, Jeremiah D, Martinez-Martinez, Maria Santos, Manzano, Pilar, Syed, Ali, El-Sakkary, Nelly, Caffrey, Conor R, Gamarro, Francisco, Ruiz-Perez, Luis Miguel, Gonzalez Pacanowska, Dolores, Ferrins, Lori, Navarro, Miguel, Pollastri, Michael P
Published in Journal of medicinal chemistry (08.07.2021)
Published in Journal of medicinal chemistry (08.07.2021)
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Journal Article
Evaluation of a class of isatinoids identified from a high-throughput screen of human kinase inhibitors as anti-Sleeping Sickness agents
Klug, Dana M, Diaz-Gonzalez, Rosario, Pérez-Moreno, Guiomar, Ceballos-Pérez, Gloria, García-Hernández, Raquel, Gomez-Pérez, Veronica, Ruiz-Pérez, Luis Miguel, Rojas-Barros, Domingo I, Gamarro, Francisco, González-Pacanowska, Dolores, Martínez-Martínez, María S, Manzano, Pilar, Ferrins, Lori, Caffrey, Conor R, Navarro, Miguel, Pollastri, Michael P
Published in PLoS neglected tropical diseases (01.02.2019)
Published in PLoS neglected tropical diseases (01.02.2019)
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Journal Article
Novel 1,2-dihydroquinazolin-2-ones: Design, synthesis, and biological evaluation against Trypanosoma brucei
Pham, ThanhTruc, Walden, Madeline, Butler, Christopher, Diaz-Gonzalez, Rosario, Pérez-Moreno, Guiomar, Ceballos-Pérez, Gloria, Gomez-Pérez, Veronica, García-Hernández, Raquel, Zecca, Henry, Krakoff, Emma, Kopec, Brian, Ichire, Ogar, Mackenzie, Caden, Pitot, Marika, Ruiz, Luis Miguel, Gamarro, Francisco, González-Pacanowska, Dolores, Navarro, Miguel, Dounay, Amy B.
Published in Bioorganic & medicinal chemistry letters (15.08.2017)
Published in Bioorganic & medicinal chemistry letters (15.08.2017)
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Journal Article
Structure-property studies of an imidazoquinoline chemotype with antitrypanosomal activity
Klug, Dana M, Diaz-Gonzalez, Rosario, DeLano, Travis J, Mavrogiannaki, Eftychia M, Buskes, Melissa J, Dalton, Raeann M, Fisher, John K, Schneider, Katherine M, Hilborne, Vivian, Fritsche, Melanie G, Simpson, Quillon J, Tear, Westley F, Devine, William G, Pérez-Moreno, Guiomar, Ceballos-Pérez, Gloria, García-Hernández, Raquel, Bosch-Navarrete, Cristina, Ruiz-Pérez, Luis Miguel, Gamarro, Francisco, González-Pacanowska, Dolores, Martinez-Martinez, Maria Santos, Manzano-Chinchon, Pilar, Navarro, Miguel, Pollastri, Michael P, Ferrins, Lori
Published in MedChemComm (01.08.2020)
Published in MedChemComm (01.08.2020)
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Journal Article
Medicinal chemistry optimization of a diaminopurine chemotype: Towards a lead for Trypanosoma brucei inhibitors
Singh, Baljinder, Diaz-Gonzalez, Rosario, Ceballos-Perez, Gloria, Rojas-Barros, Domingo I., Gunaganti, Naresh, Gillingwater, Kirsten, Martinez-Martinez, Maria Santos, Manzano, Pilar, Navarro, Miguel, Pollastri, Michael P.
Published in Journal of medicinal chemistry (13.08.2020)
Published in Journal of medicinal chemistry (13.08.2020)
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Journal Article
Medicinal Chemistry Optimization of a Diaminopurine Chemotype: Toward a Lead for Trypanosoma brucei Inhibitors
Singh, Baljinder, Diaz-Gonzalez, Rosario, Ceballos-Perez, Gloria, Rojas-Barros, Domingo I, Gunaganti, Naresh, Gillingwater, Kirsten, Martinez-Martinez, Maria Santos, Manzano, Pilar, Navarro, Miguel, Pollastri, Michael P
Published in Journal of medicinal chemistry (10.09.2020)
Published in Journal of medicinal chemistry (10.09.2020)
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Journal Article
Identification of novel anti-amoebic pharmacophores from kinase inhibitor chemotypes
Ferrins, Lori, Buskes, Melissa J, Kapteyn, Madison M, Engels, Hannah N, Enos, Suzanne E, Lu, Chenyang, Klug, Dana M, Singh, Baljinder, Quotadamo, Antonio, Bachovchin, Kelly, Tear, Westley F, Spaulding, Andrew E, Forbes, Katherine C, Bag, Seema, Rivers, Mitch, LeBlanc, Catherine, Burchfield, Erin, Armand, Jeremy R, Diaz-Gonzalez, Rosario, Ceballos-Perez, Gloria, García-Hernández, Raquel, Pérez-Moreno, Guiomar, Bosch-Navarrete, Cristina, Ruiz-Pérez, Luis Miguel, Gamarro, Francisco, González-Pacanowska, Dolores, Navarro, Miguel, Mensa-Wilmot, Kojo, Pollastri, Michael P, Kyle, Dennis E, Rice, Christopher A
Published in Frontiers in microbiology (10.05.2023)
Published in Frontiers in microbiology (10.05.2023)
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Journal Article
Corrigendum: Identification of novel anti-amoebic pharmacophores from kinase inhibitor chemotypes
Ferrins, Lori, Buskes, Melissa J., Kapteyn, Madison M., Engels, Hannah N., Enos, Suzanne E., Lu, Chenyang, Klug, Dana M., Singh, Baljinder, Quotadamo, Antonio, Bachovchin, Kelly, Tear, Westley F., Spaulding, Andrew E., Forbes, Katherine C., Bag, Seema, Rivers, Mitch, LeBlanc, Catherine, Burchfield, Erin, Armand, Jeremy R., Diaz-Gonzalez, Rosario, Ceballos-Perez, Gloria, García-Hernández, Raquel, Pérez-Moreno, Guiomar, Bosch-Navarrete, Cristina, Gómez-Liñán, Claudia, Ruiz-Pérez, Luis Miguel, Gamarro, Francisco, González-Pacanowska, Dolores, Navarro, Miguel, Mensa-Wilmot, Kojo, Pollastri, Michael P., Kyle, Dennis E., Rice, Christopher A.
Published in Frontiers in microbiology (25.10.2023)
Published in Frontiers in microbiology (25.10.2023)
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Journal Article
From Cells to Mice to Target: Characterization of NEU-1053 (SB-443342) and Its Analogues for Treatment of Human African Trypanosomiasis
Devine, William G, Diaz-Gonzalez, Rosario, Ceballos-Perez, Gloria, Rojas, Domingo, Satoh, Takashi, Tear, Westley, Ranade, Ranae M, Barros-Álvarez, Ximena, Hol, Wim G. J, Buckner, Frederick S, Navarro, Miguel, Pollastri, Michael P
Published in ACS infectious diseases (10.03.2017)
Published in ACS infectious diseases (10.03.2017)
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Journal Article
Structure–property studies of an imidazoquinoline chemotype with antitrypanosomal activity† †Electronic supplementary information (ESI) available. See DOI: 10.1039/d0md00103a
Klug, Dana M., Diaz-Gonzalez, Rosario, DeLano, Travis J., Mavrogiannaki, Eftychia M., Buskes, Melissa J., Dalton, Raeann M., Fisher, John K., Schneider, Katherine M., Hilborne, Vivian, Fritsche, Melanie G., Simpson, Quillon J., Tear, Westley F., Devine, William G., Pérez-Moreno, Guiomar, Ceballos-Pérez, Gloria, García-Hernández, Raquel, Bosch-Navarrete, Cristina, Ruiz-Pérez, Luis Miguel, Gamarro, Francisco, González-Pacanowska, Dolores, Martinez-Martinez, Maria Santos, Manzano-Chinchon, Pilar, Navarro, Miguel, Pollastri, Michael P., Ferrins, Lori
Published in RSC medicinal chemistry (10.07.2020)
Published in RSC medicinal chemistry (10.07.2020)
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Journal Article