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Published in EMBO molecular medicine (01.12.2010)
Published in EMBO molecular medicine (01.12.2010)
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Large-Scale Assessment of Binding Free Energy Calculations in Active Drug Discovery Projects
Schindler, Christina E. M, Baumann, Hannah, Blum, Andreas, Böse, Dietrich, Buchstaller, Hans-Peter, Burgdorf, Lars, Cappel, Daniel, Chekler, Eugene, Czodrowski, Paul, Dorsch, Dieter, Eguida, Merveille K. I, Follows, Bruce, Fuchß, Thomas, Grädler, Ulrich, Gunera, Jakub, Johnson, Theresa, Jorand Lebrun, Catherine, Karra, Srinivasa, Klein, Markus, Knehans, Tim, Koetzner, Lisa, Krier, Mireille, Leiendecker, Matthias, Leuthner, Birgitta, Li, Liwei, Mochalkin, Igor, Musil, Djordje, Neagu, Constantin, Rippmann, Friedrich, Schiemann, Kai, Schulz, Robert, Steinbrecher, Thomas, Tanzer, Eva-Maria, Unzue Lopez, Andrea, Viacava Follis, Ariele, Wegener, Ansgar, Kuhn, Daniel
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Pudelko, Linda, Jaehrling, Frank, Reusch, Christof, Viteri, Santiago, Stroh, Christopher, Linde, Nina, Sanderson, Michael P., Musch, Doreen, Lebrun, Catherine Jorand, Keil, Marina, Esdar, Christina, Blaukat, Andree, Rosell, Rafael, Schumacher, Karl Maria, Karachaliou, Niki
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Published in iScience (18.12.2020)
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Optimization of the Central Core of Indolinone–Acetic Acid-Based CRTH2 (DP2) Receptor Antagonists
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Published in ACS medicinal chemistry letters (11.08.2011)
Published in ACS medicinal chemistry letters (11.08.2011)
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Crosignani, Stefano, Prêtre, Adeline, Jorand-Lebrun, Catherine, Fraboulet, Gaële, Seenisamy, Jeyaprakashnarayanan, Augustine, John Kallikat, Missotten, Marc, Humbert, Yves, Cleva, Christophe, Abla, Nada, Daff, Hamina, Schott, Olivier, Schneider, Manfred, Burgat-Charvillon, Fabienne, Rivron, Delphine, Hamernig, Ingrid, Arrighi, Jean-François, Gaudet, Marilène, Zimmerli, Simone C, Juillard, Pierre, Johnson, Zoe
Published in Journal of medicinal chemistry (27.10.2011)
Published in Journal of medicinal chemistry (27.10.2011)
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Convergent Functional Genomics of Oligodendrocyte Differentiation Identifies Multiple Autoinhibitory Signaling Circuits
Pescini Gobert, Rosanna, Joubert, Lara, Curchod, Marie-Laure, Salvat, Catherine, Foucault, Isabelle, Jorand-Lebrun, Catherine, Lamarine, Marc, Peixoto, Hélène, Vignaud, Chloé, Frémaux, Christèle, Jomotte, Thérèse, Françon, Bernard, Alliod, Chantal, Bernasconi, Lilia, Abderrahim, Hadi, Perrin, Dominique, Bombrun, Agnes, Zanoguera, Francisca, Rommel, Christian, van Huijsduijnen, Rob Hooft
Published in Molecular and Cellular Biology (01.03.2009)
Published in Molecular and Cellular Biology (01.03.2009)
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OLIVER POHL, ANNA QUATTROPANI, VINCENT POMEL, ERNEST LOUMAYE, JEAN-PIERRE GOTTELAND, MATTHIAS SCHWARZ, CATHERINE JORAND-LEBRUN, PATRICK NAXOS PAGE
Year of Publication 30.01.2024
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Year of Publication 30.01.2024
Patent
Discovery of novel Cyclophilin D inhibitors starting from three dimensional fragments with millimolar potencies
Grädler, Ulrich, Schwarz, Daniel, Blaesse, Michael, Leuthner, Birgitta, Johnson, Theresa L., Bernard, Frederic, Jiang, Xuliang, Marx, Andreas, Gilardone, Marine, Lemoine, Hugues, Roche, Didier, Jorand-Lebrun, Catherine
Published in Bioorganic & medicinal chemistry letters (01.12.2019)
Published in Bioorganic & medicinal chemistry letters (01.12.2019)
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Abstract ND09: M3913 induces the maladaptive unfolded protein response through a novel mechanism resulting in strong anti-tumor activity
Czauderna, Frank, Schneider, Richard, Ramaswamy, Shivapriya, Brandstetter, Susanne, Drouin, Elise, Bogatyrova, Olga, Mazur, Johanna, Sun, Qing, Jorand-Lebrun, Catherine, Sherbetjian, Eva, Nachtigall, Jonny, Wing, Carolyn, Hildebrand, Christian, Ellinghaus, Peter, Lemoine, Isabelle, Johnson, Mac, Hoover, Russell, Clark, Michael, Lindemann, Ralph
Published in Cancer research (Chicago, Ill.) (29.05.2023)
Published in Cancer research (Chicago, Ill.) (29.05.2023)
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Identification, synthesis, and biological evaluation of novel pyrazoles as low molecular weight luteinizing hormone receptor agonists
Jorand-Lebrun, Catherine, Brondyk, Bill, Lin, Jing, Magar, Sharad, Murray, Robert, Reddy, Adulla, Shroff, Hitesh, Wands, Greg, Weiser, Weishui, Xu, Qihong, McKenna, Sean, Brugger, Nadia
Published in Bioorganic & medicinal chemistry letters (01.04.2007)
Published in Bioorganic & medicinal chemistry letters (01.04.2007)
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GLEPP1/Protein-tyrosine Phosphatase ϕ Inhibitors Block Chemotaxis in Vitro and in Vivo and Improve Murine Ulcerative Colitis
Gobert, Rosanna Pescini, van den Eijnden, Monique, Szyndralewiez, Cedric, Jorand-Lebrun, Catherine, Swinnen, Dominique, Chen, Linfeng, Gillieron, Corine, Pixley, Fiona, Juillard, Pierre, Gerber, Patrick, Johnson-Léger, Caroline, Halazy, Serge, Camps, Montserrat, Bombrun, Agnes, Shipp, Margaret, Vitte, Pierre-Alain, Ardissone, Vittoria, Ferrandi, Chiara, Perrin, Dominique, Rommel, Christian, van Huijsduijnen, Rob Hooft
Published in The Journal of biological chemistry (24.04.2009)
Published in The Journal of biological chemistry (24.04.2009)
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