Structure−Activity Relationships of Novel 2-Substituted Quinazoline Antibacterial Agents
Kung, Pei-Pei, Casper, Martin D, Cook, Kimberley L, Wilson-Lingardo, Laura, Risen, Lisa M, Vickers, Timothy A, Ranken, Ray, Blyn, Lawrence B, Wyatt, Jacqueline R, Cook, P. Dan, Ecker, David J
Published in Journal of medicinal chemistry (04.11.1999)
Published in Journal of medicinal chemistry (04.11.1999)
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Discovery and Structure−Activity Relationship of 3-Methoxy-N-(3-(1-methyl-1H-pyrazol-5-yl)-4-(2-morpholinoethoxy)phenyl)benzamide (APD791): A Highly Selective 5-Hydroxytryptamine2A Receptor Inverse Agonist for the Treatment of Arterial Thrombosis
Xiong, Yifeng, Teegarden, Bradley R, Choi, Jin-Sun Karoline, Strah-Pleynet, Sonja, Decaire, Marc, Jayakumar, Honnappa, Dosa, Peter I, Casper, Martin D, Pham, Lan, Feichtinger, Konrad, Ullman, Brett, Adams, John, Yuskin, Diane, Frazer, John, Morgan, Michael, Sadeque, Abu, Chen, Weichao, Webb, Robert R, Connolly, Daniel T, Semple, Graeme, Al-Shamma, Hussien
Published in Journal of medicinal chemistry (10.06.2010)
Published in Journal of medicinal chemistry (10.06.2010)
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Pyrimidine-based antagonists of h-MCH-R1 derived from ATC0175: In vitro profiling and in vivo evaluation
Semple, Graeme, Tran, Thuy-Anh, Kramer, Bryan, Hsu, Debbie, Han, Sangdon, Choi, Juyi, Vallar, Pureza, Casper, Martin D., Zou, Ning, Hauser, Erin K., Thomsen, William, Whelan, Kevin, Sengupta, Dipanjan, Morgan, Michael, Sekiguchi, Yoshinori, Kanuma, Kosuke, Chaki, Shigeyuki, Grottick, Andrew J.
Published in Bioorganic & medicinal chemistry letters (01.11.2009)
Published in Bioorganic & medicinal chemistry letters (01.11.2009)
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Uniformly modified 2'-deoxy-2'-fluoro-phosphorothioate oligonucleotides as nuclease-resistant antisense compounds with high affinity and specificity for RNA targets
Kawasaki, Andrew M, Casper, Martin D, Freier, Susan M, Lesnik, Elena A, Zounes, Maryann C, Cummins, Lendell L, Gonzalez, Carolyn, Cook, P. Dan
Published in Journal of medicinal chemistry (02.04.1993)
Published in Journal of medicinal chemistry (02.04.1993)
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Journal Article
Discovery and Structure-Activity Relationship of 3-Methoxy-N-(3-(1-methyl-1H-pyrazol-5-yl)-4-(2-morpholinoethoxy)phenyl)benzamide (APD791): A Highly Selective 5-Hydroxytryptamine(2A) Receptor Inverse Agonist for the Treatment of Arterial Thrombosis
Xiong, Yifeng, Teegarden, Bradley R., Choi, Jin-Sun Karoline, Strah-Pleynet, Sonja, Decaire, Marc, Jayakumar, Honnappa, Dosa, Peter I., Casper, Martin D., Pham, Lan, Feichtinger, Konrad, Ullman, Brett, Adams, John, Yuskin, Diane, Frazer, John, Morgan, Michael, Sadeque, Abu, Chen, Weichao, Webb, Robert R., Connolly, Daniel T., Semple, Graeme, Al-Shamma, Hussien
Published in Journal of medicinal chemistry (10.06.2010)
Published in Journal of medicinal chemistry (10.06.2010)
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Journal Article
Discovery and Structure−Activity Relationship of 3-Methoxy- N -(3-(1-methyl-1 H -pyrazol-5-yl)-4-(2-morpholinoethoxy)phenyl)benzamide (APD791): A Highly Selective 5-Hydroxytryptamine 2A Receptor Inverse Agonist for the Treatment of Arterial Thrombosis
Xiong, Yifeng, Teegarden, Bradley R., Choi, Jin-Sun Karoline, Strah-Pleynet, Sonja, Decaire, Marc, Jayakumar, Honnappa, Dosa, Peter I., Casper, Martin D., Pham, Lan, Feichtinger, Konrad, Ullman, Brett, Adams, John, Yuskin, Diane, Frazer, John, Morgan, Michael, Sadeque, Abu, Chen, Weichao, Webb, Robert R., Connolly, Daniel T., Semple, Graeme, Al-Shamma, Hussien
Published in Journal of medicinal chemistry (10.06.2010)
Published in Journal of medicinal chemistry (10.06.2010)
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Synthesis, hybridization, and nuclease resistance properties of 2′-O-aminooxyethyl ( 2′-O-AOE) modified oligonucleotides
Kawasaki, Andrew M., Casper, Martin D., Prakash, Thazha P., Manalili, Sheri, Sasmor, Henri, Manoharan, Muthiah, Cook, P.Dan
Published in Tetrahedron letters (22.01.1999)
Published in Tetrahedron letters (22.01.1999)
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Carbohydrate Modifications in Antisense Oligonucleotide Therapy: New Kids on the Block
Manoharan, Muthiah, Kawasaki, Andrew M., Prakash, Thazha P., Fraser, Allister S., Prhavc, Marija, Inamati, Gopal B., Casper, Martin D., Cook, P. Dan
Published in Nucleosides & nucleotides (01.06.1999)
Published in Nucleosides & nucleotides (01.06.1999)
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Synthesis, Hybridization, and Nuclease Resistance Properties of 2′-O-Aminooxyethyl Modified Oligonucleotides
Kawasaki, Andrew M., Casper, Martin D., Prakash, Thazha P., Manalili, Sheri, Sasmor, Henri, Manoharan, Muthiah, Cook, P. Dan
Published in Nucleosides & nucleotides (01.06.1999)
Published in Nucleosides & nucleotides (01.06.1999)
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Solution Phase Combinatorial Chemistry. Purine- and Pyrimidine-Based Libraries with Antibacterial Activity via Solution Phase Simultaneous Addition of Functionalities
Kawasaki, Andrew M., Casper, Martin D., Gaus, Hans J., Herrmann, Rigo, Griffey, Richard H., Cook, P. Dan
Published in Nucleosides & nucleotides (01.04.1999)
Published in Nucleosides & nucleotides (01.04.1999)
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