Search Results - "Casper, Martin" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Structure−Activity Relationships of Novel 2-Substituted Quinazoline Antibacterial Agents

Structure−Activity Relationships of Novel 2-Substituted Quinazoline Antibacterial Agents

by Kung, Pei-Pei, Casper, Martin D, Cook, Kimberley L, Wilson-Lingardo, Laura, Risen, Lisa M, Vickers, Timothy A, Ranken, Ray, Blyn, Lawrence B, Wyatt, Jacqueline R, Cook, P. Dan, Ecker, David J
Published in Journal of medicinal chemistry (04.11.1999)

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Journal Article

Discovery and Structure−Activity Relationship of 3-Methoxy-N-(3-(1-methyl-1H-pyrazol-5-yl)-4-(2-morpholinoethoxy)phenyl)benzamide (APD791): A Highly Selective 5-Hydroxytryptamine2A Receptor Inverse Agonist for the Treatment of Arterial Thrombosis

Discovery and Structure−Activity Relationship of 3-Methoxy-N-(3-(1-methyl-1H-pyrazol-5-yl)-4-(2-morpholinoethoxy)phenyl)benzamide (APD791): A Highly Selective 5-Hydroxytryptamine2A Receptor Inverse Agonist for the Treatment of Arterial Thrombosis

by Xiong, Yifeng, Teegarden, Bradley R, Choi, Jin-Sun Karoline, Strah-Pleynet, Sonja, Decaire, Marc, Jayakumar, Honnappa, Dosa, Peter I, Casper, Martin D, Pham, Lan, Feichtinger, Konrad, Ullman, Brett, Adams, John, Yuskin, Diane, Frazer, John, Morgan, Michael, Sadeque, Abu, Chen, Weichao, Webb, Robert R, Connolly, Daniel T, Semple, Graeme, Al-Shamma, Hussien
Published in Journal of medicinal chemistry (10.06.2010)

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Pyrimidine-based antagonists of h-MCH-R1 derived from ATC0175: In vitro profiling and in vivo evaluation

Pyrimidine-based antagonists of h-MCH-R1 derived from ATC0175: In vitro profiling and in vivo evaluation

by Semple, Graeme, Tran, Thuy-Anh, Kramer, Bryan, Hsu, Debbie, Han, Sangdon, Choi, Juyi, Vallar, Pureza, Casper, Martin D., Zou, Ning, Hauser, Erin K., Thomsen, William, Whelan, Kevin, Sengupta, Dipanjan, Morgan, Michael, Sekiguchi, Yoshinori, Kanuma, Kosuke, Chaki, Shigeyuki, Grottick, Andrew J.
Published in Bioorganic & medicinal chemistry letters (01.11.2009)

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Uniformly modified 2'-deoxy-2'-fluoro-phosphorothioate oligonucleotides as nuclease-resistant antisense compounds with high affinity and specificity for RNA targets

Uniformly modified 2'-deoxy-2'-fluoro-phosphorothioate oligonucleotides as nuclease-resistant antisense compounds with high affinity and specificity for RNA targets

by Kawasaki, Andrew M, Casper, Martin D, Freier, Susan M, Lesnik, Elena A, Zounes, Maryann C, Cummins, Lendell L, Gonzalez, Carolyn, Cook, P. Dan
Published in Journal of medicinal chemistry (02.04.1993)

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Allyl Group as a Protecting Group for Internucleotide Phosphate and Thiophosphate Linkages in Oligonucleotide Synthesis: Facile Oxidation and Deprotection Conditions

Allyl Group as a Protecting Group for Internucleotide Phosphate and Thiophosphate Linkages in Oligonucleotide Synthesis: Facile Oxidation and Deprotection Conditions

by Manoharan, Muthiah, Lu, Yixin, Casper, Martin D, Just, George
Published in Organic letters (10.02.2000)

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Discovery and Structure-Activity Relationship of 3-Methoxy-N-(3-(1-methyl-1H-pyrazol-5-yl)-4-(2-morpholinoethoxy)phenyl)benzamide (APD791): A Highly Selective 5-Hydroxytryptamine(2A) Receptor Inverse Agonist for the Treatment of Arterial Thrombosis

Discovery and Structure-Activity Relationship of 3-Methoxy-N-(3-(1-methyl-1H-pyrazol-5-yl)-4-(2-morpholinoethoxy)phenyl)benzamide (APD791): A Highly Selective 5-Hydroxytryptamine(2A) Receptor Inverse Agonist for the Treatment of Arterial Thrombosis

by Xiong, Yifeng, Teegarden, Bradley R., Choi, Jin-Sun Karoline, Strah-Pleynet, Sonja, Decaire, Marc, Jayakumar, Honnappa, Dosa, Peter I., Casper, Martin D., Pham, Lan, Feichtinger, Konrad, Ullman, Brett, Adams, John, Yuskin, Diane, Frazer, John, Morgan, Michael, Sadeque, Abu, Chen, Weichao, Webb, Robert R., Connolly, Daniel T., Semple, Graeme, Al-Shamma, Hussien
Published in Journal of medicinal chemistry (10.06.2010)

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Solubilized phenyl-pyrazole ureas as potent, selective 5-HT2A inverse-agonists and their application as antiplatelet agents

Solubilized phenyl-pyrazole ureas as potent, selective 5-HT2A inverse-agonists and their application as antiplatelet agents

by DOSA, Peter I, STRAH-PLEYNET, Sonja, WEBB, Robert R, ADAMS, John W, RAMIREZ, Juan, RICHMAN, Jeremy G, THOMSEN, William, SEMPLE, Graeme, TEEGARDEN, Bradley R, JAYAKUMAR, Honnappa, CASPER, Martin, DECAIRE, Marc, YIFENG XIONG, LEHMANN, Juerg, CHOI, Karoline, ELWELL, Katie, WONG, Amy
Published in Bioorganic & medicinal chemistry letters (15.09.2009)

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Journal Article

Discovery and Structure−Activity Relationship of 3-Methoxy- N -(3-(1-methyl-1 H -pyrazol-5-yl)-4-(2-morpholinoethoxy)phenyl)benzamide (APD791): A Highly Selective 5-Hydroxytryptamine 2A Receptor Inverse Agonist for the Treatment of Arterial Thrombosis

Discovery and Structure−Activity Relationship of 3-Methoxy- N -(3-(1-methyl-1 H -pyrazol-5-yl)-4-(2-morpholinoethoxy)phenyl)benzamide (APD791): A Highly Selective 5-Hydroxytryptamine 2A Receptor Inverse Agonist for the Treatment of Arterial Thrombosis

by Xiong, Yifeng, Teegarden, Bradley R., Choi, Jin-Sun Karoline, Strah-Pleynet, Sonja, Decaire, Marc, Jayakumar, Honnappa, Dosa, Peter I., Casper, Martin D., Pham, Lan, Feichtinger, Konrad, Ullman, Brett, Adams, John, Yuskin, Diane, Frazer, John, Morgan, Michael, Sadeque, Abu, Chen, Weichao, Webb, Robert R., Connolly, Daniel T., Semple, Graeme, Al-Shamma, Hussien
Published in Journal of medicinal chemistry (10.06.2010)

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Lead optimization of 4-(dimethylamino)quinazolines, potent and selective antagonists for the melanin-concentrating hormone receptor 1

Lead optimization of 4-(dimethylamino)quinazolines, potent and selective antagonists for the melanin-concentrating hormone receptor 1

by Kanuma, Kosuke, Omodera, Katsunori, Nishiguchi, Mariko, Funakoshi, Takeo, Chaki, Shigeyuki, Semple, Graeme, Tran, Thuy-Anh, Kramer, Bryan, Hsu, Debbie, Casper, Martin, Thomsen, Bill, Sekiguchi, Yoshinori
Published in Bioorganic & medicinal chemistry letters (01.09.2005)

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Solubilized phenyl-pyrazole ureas as potent, selective 5-HT sub(2A) inverse-agonists and their application as antiplatelet agents

Solubilized phenyl-pyrazole ureas as potent, selective 5-HT sub(2A) inverse-agonists and their application as antiplatelet agents

by Dosa, Peter I, Strah-Pleynet, Sonja, Jayakumar, Honnappa, Casper, Martin, Decaire, Marc, Xiong, Yifeng, Lehmann, Juerg, Choi, Karoline, Elwell, Katie, Wong, Amy, Webb, Robert R, Adams, John W, Ramirez, Juan, Richman, Jeremy G, Thomsen, William, Semple, Graeme, Teegarden, Bradley R
Published in Bioorganic & medicinal chemistry letters (15.09.2009)

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Journal Article

Discovery of 4-(dimethylamino)quinazolines as potent and selective antagonists for the melanin-concentrating hormone receptor 1

Discovery of 4-(dimethylamino)quinazolines as potent and selective antagonists for the melanin-concentrating hormone receptor 1

by Kanuma, Kosuke, Omodera, Katsunori, Nishiguchi, Mariko, Funakoshi, Takeo, Chaki, Shigeyuki, Semple, Graeme, Tran, Thuy-Anh, Kramer, Bryan, Hsu, Debbie, Casper, Martin, Thomsen, Bill, Beeley, Nigel, Sekiguchi, Yoshinori
Published in Bioorganic & medicinal chemistry letters (16.05.2005)

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Journal Article

Solubilized phenyl-pyrazole ureas as potent, selective 5-HT 2A inverse-agonists and their application as antiplatelet agents

Solubilized phenyl-pyrazole ureas as potent, selective 5-HT 2A inverse-agonists and their application as antiplatelet agents

by Dosa, Peter I., Strah-Pleynet, Sonja, Jayakumar, Honnappa, Casper, Martin, Decaire, Marc, Xiong, Yifeng, Lehmann, Juerg, Choi, Karoline, Elwell, Katie, Wong, Amy, Webb, Robert R., Adams, John W., Ramirez, Juan, Richman, Jeremy G., Thomsen, William, Semple, Graeme, Teegarden, Bradley R.
Published in Bioorganic & medicinal chemistry letters (2009)

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Journal Article

3-PHENYL-PYRAZOLE DERIVATIVES AS MODULATORS OF THE 5-HT2A SEROTONIN RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

3-PHENYL-PYRAZOLE DERIVATIVES AS MODULATORS OF THE 5-HT2A SEROTONIN RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

by XIONG YIFENG, JONES ROBERT M, UNETT DAVID J, JAYAKUMAR HONNAPPA, CHOI JIN SUN KAROLINE, DOSA PETER I, FEICHTINGER KONRAD, CASPER MARTIN, LEHMANN JUERG, TEEGARDEN BRADLEY, STRAH PLEYNET SONJA
Year of Publication 14.03.2013

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Patent

Solubilized phenyl-pyrazole ureas as potent, selective 5-HT(2A) inverse-agonists and their application as antiplatelet agents

Solubilized phenyl-pyrazole ureas as potent, selective 5-HT(2A) inverse-agonists and their application as antiplatelet agents

by Dosa, Peter I, Strah-Pleynet, Sonja, Jayakumar, Honnappa, Casper, Martin, Decaire, Marc, Xiong, Yifeng, Lehmann, Juerg, Choi, Karoline, Elwell, Katie, Wong, Amy, Webb, Robert R, Adams, John W, Ramirez, Juan, Richman, Jeremy G, Thomsen, William, Semple, Graeme, Teegarden, Bradley R
Published in Bioorganic & medicinal chemistry letters (15.09.2009)

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Journal Article

Presenter device

Presenter device

by Wu, Libao, Rüegg, Martin Casper, Phua, Jasper, Helwig, Marten, Mcloughlin, Padraig, Gregoire, Olivier, Chao, Fleming
Year of Publication 21.01.2020

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Patent

Synthesis, hybridization, and nuclease resistance properties of 2′-O-aminooxyethyl ( 2′-O-AOE) modified oligonucleotides

Synthesis, hybridization, and nuclease resistance properties of 2′-O-aminooxyethyl ( 2′-O-AOE) modified oligonucleotides

by Kawasaki, Andrew M., Casper, Martin D., Prakash, Thazha P., Manalili, Sheri, Sasmor, Henri, Manoharan, Muthiah, Cook, P.Dan
Published in Tetrahedron letters (22.01.1999)

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Journal Article

3-phenyl-pyrazole derivatives as modulators of the 5-HT2A serotonin receptor useful for the treatment of disorders related thereto

3-phenyl-pyrazole derivatives as modulators of the 5-HT2A serotonin receptor useful for the treatment of disorders related thereto

by Xiong, Yifeng, Strah-Pleynet, Sonja, Unett, David J, Feichtinger, Konrad, Jones, Robert M, Dosa, Peter I, Teegarden, Bradley, Jayakumar, Honnappa, Casper, Martin, Lehmann, Juerg, Choi, Jin Sun Karoline
Year of Publication 22.09.2020

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Patent

3-PHENYL-PYRAZOLE DERIVATIVES AS MODULATORS OF THE 5-HT2A SEROTONIN RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

3-PHENYL-PYRAZOLE DERIVATIVES AS MODULATORS OF THE 5-HT2A SEROTONIN RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

by Xiong, Yifeng, Strah-Pleynet, Sonja, Unett, David J, Feichtinger, Konrad, Jones, Robert M, Dosa, Peter I, Teegarden, Bradley, Jayakumar, Honnappa, Casper, Martin, Lehmann, Juerg, Choi, Jin Sun Karoline
Year of Publication 29.08.2019

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Patent

3-fenylpyrazol derivater, farmasøytiske sammensetninger inneholdende slike, fremgangsmåte for fremstilling og anvendelse som modulatorer av 5HT2A serotoninreseptoren for behandling av forstyrrelser relatert dertil

3-fenylpyrazol derivater, farmasøytiske sammensetninger inneholdende slike, fremgangsmåte for fremstilling og anvendelse som modulatorer av 5HT2A serotoninreseptoren for behandling av forstyrrelser relatert dertil

by Xiong, Yifeng, Strah-Pleynet, Sonja, Unett, David J, Feichtinger, Konrad, Jones, Robert M, Dosa, Peter I, Teegarden, Bradley, Jayakumar, Honnappa, Casper, Martin, Choi, Jin Sun Karoline, Lehmann, Juerg
Year of Publication 22.05.2017

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Patent

Heat exchanger and heat exchanger arrangement structure

Heat exchanger and heat exchanger arrangement structure

by KLAUS HASDENTOEFEIR, UWE FOSTER, JOHANNS TIM, MARTIN CASPER, PEDRO GONZALEZRACEA, HERBERT HOFFMAN
Year of Publication 08.04.2015

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