A highly selective and specific PET tracer for imaging of tau pathologies
Zhang, Wei, Arteaga, Janna, Cashion, Daniel K, Chen, Gang, Gangadharmath, Umesh, Gomez, Luis F, Kasi, Dhanalakshmi, Lam, Chung, Liang, Qianwa, Liu, Changhui, Mocharla, Vani P, Mu, Fanrong, Sinha, Anjana, Szardenings, A Katrin, Wang, Eric, Walsh, Joseph C, Xia, Chunfang, Yu, Chul, Zhao, Tieming, Kolb, Hartmuth C
Published in Journal of Alzheimer's disease (01.01.2012)
Published in Journal of Alzheimer's disease (01.01.2012)
Get more information
Journal Article
Discovery of a Series of Phosphonic Acid-Containing Thiazoles and Orally Bioavailable Diamide Prodrugs That Lower Glucose in Diabetic Animals Through Inhibition of Fructose-1,6-Bisphosphatase
Dang, Qun, Liu, Yan, Cashion, Daniel K, Kasibhatla, Srinivas Rao, Jiang, Tao, Taplin, Frank, Jacintho, Jason D, Li, Haiqing, Sun, Zhili, Fan, Yi, DaRe, Jay, Tian, Feng, Li, Wenyu, Gibson, Tony, Lemus, Robert, van Poelje, Paul D, Potter, Scott C, Erion, Mark D
Published in Journal of medicinal chemistry (13.01.2011)
Published in Journal of medicinal chemistry (13.01.2011)
Get full text
Journal Article
Discovery of Phosphonic Diamide Prodrugs and Their Use for the Oral Delivery of a Series of Fructose 1,6-Bisphosphatase Inhibitors
Dang, Qun, Kasibhatla, Srinivas Rao, Jiang, Tao, Fan, Kevin, Liu, Yan, Taplin, Frank, Schulz, William, Cashion, Daniel K, Reddy, K. Raja, van Poelje, Paul D, Fujitaki, James M, Potter, Scott C, Erion, Mark D
Published in Journal of medicinal chemistry (24.07.2008)
Published in Journal of medicinal chemistry (24.07.2008)
Get full text
Journal Article
Application of Mechanistic Multiparameter Optimization and Large-Scale In Vitro to In Vivo Pharmacokinetics Correlations to Small-Molecule Therapeutic Projects
Broccatelli, Fabio, Veeravalli, Vijayabhaskar, Cashion, Daniel, Baylon, Javier L., Lombardo, Franco, Jia, Lei
Published in Molecular pharmaceutics (02.09.2024)
Published in Molecular pharmaceutics (02.09.2024)
Get full text
Journal Article
Hit-to-Lead Optimization and Discovery of 5‑((5-([1,1′-Biphenyl]-4-yl)-6-chloro‑1H‑benzo[d]imidazol-2-yl)oxy)-2-methylbenzoic Acid (MK-3903): A Novel Class of Benzimidazole-Based Activators of AMP-Activated Protein Kinase
Lan, Ping, Romero, F. Anthony, Wodka, Dariusz, Kassick, Andrew J, Dang, Qun, Gibson, Tony, Cashion, Daniel, Zhou, Gaochao, Chen, Yuli, Zhang, Xiaoping, Zhang, Aihua, Li, Ying, Trujillo, Maria E, Shao, Qing, Wu, Margaret, Xu, Shiyao, He, Huaibing, MacKenna, Deidre, Staunton, Jocelyn, Chapman, Kevin T, Weber, Ann, Sebhat, Iyassu K, Makara, Gergely M
Published in Journal of medicinal chemistry (09.11.2017)
Published in Journal of medicinal chemistry (09.11.2017)
Get full text
Journal Article
Hit-to-Lead Optimization and Discovery of 5-((5-([1,1′-Biphenyl]-4-yl)-6-chloro-1 H -benzo[ d ]imidazol-2-yl)oxy)-2-methylbenzoic Acid (MK-3903): A Novel Class of Benzimidazole-Based Activators of AMP-Activated Protein Kinase
Lan, Ping, Romero, F. Anthony, Wodka, Dariusz, Kassick, Andrew J., Dang, Qun, Gibson, Tony, Cashion, Daniel, Zhou, Gaochao, Chen, Yuli, Zhang, Xiaoping, Zhang, Aihua, Li, Ying, Trujillo, Maria E., Shao, Qing, Wu, Margaret, Xu, Shiyao, He, Huaibing, MacKenna, Deidre, Staunton, Jocelyn, Chapman, Kevin T., Weber, Ann, Sebhat, Iyassu K., Makara, Gergely M.
Published in Journal of medicinal chemistry (09.11.2017)
Published in Journal of medicinal chemistry (09.11.2017)
Get full text
Journal Article
Inhibitor Binding Mode Differences Within the AGC Subfamily
Delker, Silvia, Robinson, Dale, Bahmanyar, Sami, Pagarigan, Barbra, Fang, Wei, Abbasian, Mahan, Mahmoudi, Afshin, Cashion, Daniel, Cathers, Brian, Chamberlain, Philip
Published in Acta crystallographica. Section A, Foundations and advances (05.08.2014)
Published in Acta crystallographica. Section A, Foundations and advances (05.08.2014)
Get full text
Journal Article
SUBSTITUTED DIAMINOPYRIMIDYL COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH
HEGDE SAYEE, RAHEJA RAJ, PLANTEVIN KRENITSKY VERONIQUE, NORRIS STEPHEN, CALABRESE ANDREW ANTONY, SAPIENZA JOHN, LEFTHERIS KATERINA, HANSEN JOSHUA, CORREA MATTHEW, BAHMANYAR SOGOLE, CATHERS BRIAN EDWIN, TORRES EDUARDO, PAPA PATRICK, MORTENSEN DEBORAH, PARNES JASON, WHITEFIELD BRANDON WADE, BENNETT BRYDON, HUANG DEHUA, CASHION DANIEL, DELGADO MARIA MERCEDES
Year of Publication 10.08.2016
Get full text
Year of Publication 10.08.2016
Patent
WEE1 Degrading Compounds and Uses Thereof
Sapienza, John, Riggs, Jennifer R, Cashion, Daniel K, Pierce, Meekyum Olivia, Edwards, Jacob T
Year of Publication 29.02.2024
Get full text
Year of Publication 29.02.2024
Patent
WEE1 DEGRADING COMPOUNDS AND USES THEREOF
PIERCE, Meekyum Olivia, RIGGS, Jennifer R, EDWARDS, Jacob T, SAPIENZA, John, CASHION, Daniel K
Year of Publication 04.01.2024
Get full text
Year of Publication 04.01.2024
Patent
IMAGING AGENTS FOR DETECTING NEUROLOGICAL DISORDERS
KASI DHANALAKSHMI, CHEN GANG, YU CHUL, WALSH JOSEPH C, SINHA ANJANA, GANGADHARMATH UMESH B, KOLB HARTMUTH C, LIU CHANGHUI, CASHION DANIEL KURT, ZHANG WEI, SZARDENINGS ANNA KATRIN, WANG ERIC
Year of Publication 28.02.2013
Get full text
Year of Publication 28.02.2013
Patent
IMAGING AGENTS FOR DETECTING NEUROLOGICAL DISORDERS
YU CHUL, KOLB HARTMUTH C, MOCHARLA VANI P, CASHION DANIEL KURT, WANG ERIC, KASI DHANALAKSHMI, CHEN GANG, WALSH JOSEPH C, GANGADHARMATH UMESH B, SINHA ANJANA, LIU CHANGHUI, ZHANG WEI, SCOTT PETER J.H, SZARDENINGS ANNA KATRIN
Year of Publication 21.12.2011
Get full text
Year of Publication 21.12.2011
Patent
WEE1 degrading compounds and uses thereof
RIGGS, JENNIFER R, PIERCE, MEEKYUM OLIVIA, EDWARDS, JACOB T, SAPIENZA, JOHN, CASHION, DANIEL K
Year of Publication 01.03.2024
Get full text
Year of Publication 01.03.2024
Patent
IMAGING AGENTS FOR DETECTING NEUROLOGICAL DISORDERS
LIU, Changhui, WALSH, Joseph, C, CASHION, Daniel, Kurt, GANGADHARMATH, Umesh, B, MOCHARLA, Vani, P, SCOTT, Peter, J.H, SINHA, Anjana, KASI, Dhanalakshmi, CHEN, Gang, YU, Chul, SZARDENINGS, Anna, Katrin, WANG, Eric, ZHANG, Wei, KOLB, Hartmuth, C
Year of Publication 06.05.2020
Get full text
Year of Publication 06.05.2020
Patent