Stereoselective block of hERG channel by (S)-methadone and QT interval prolongation in CYP2B6 slow metabolizers
Eap, C B, Crettol, S, Rougier, J-S, Schläpfer, J, Sintra Grilo, L, Déglon, J-J, Besson, J, Croquette-Krokar, M, Carrupt, P-A, Abriel, H
Published in Clinical pharmacology and therapeutics (01.05.2007)
Published in Clinical pharmacology and therapeutics (01.05.2007)
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Journal Article
QSAR analysis and molecular modeling of ABCG2-specific inhibitors
Nicolle, E., Boumendjel, A., Macalou, S., Genoux, E., Ahmed-Belkacem, A., Carrupt, P.-A., Di Pietro, A.
Published in Advanced drug delivery reviews (31.01.2009)
Published in Advanced drug delivery reviews (31.01.2009)
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Journal Article
Targeting the multidrug ABCG2 transporter with flavonoidic inhibitors: in vitro optimization and in vivo validation
Boumendjel, A, Macalou, S, Valdameri, G, Pozza, A, Gauthier, C, Arnaud, O, Nicolle, E, Magnard, S, Falson, P, Terreux, R, Carrupt, P-A, Payen, L, Di Pietro, A
Published in Current medicinal chemistry (01.08.2011)
Published in Current medicinal chemistry (01.08.2011)
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Journal Article
Predicting Blood−Brain Barrier Permeation from Three-Dimensional Molecular Structure
Crivori, Patrizia, Cruciani, Gabriele, Carrupt, Pierre-Alain, Testa, Bernard
Published in Journal of medicinal chemistry (01.06.2000)
Published in Journal of medicinal chemistry (01.06.2000)
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Journal Article
Xanthones from Gentianella amarella ssp. acuta with Acetylcholinesterase and Monoamine Oxidase Inhibitory Activities
Urbain, A., Marston, A., Grilo, L. Sintra, Bravo, J., Purev, O., Purevsuren, B., Batsuren, D., Reist, M., Carrupt, P.-A., Hostettmann, K.
Published in Journal of natural products (Washington, D.C.) (01.05.2008)
Published in Journal of natural products (Washington, D.C.) (01.05.2008)
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Journal Article
Coumarins Derivatives as Dual Inhibitors of Acetylcholinesterase and Monoamine Oxidase
Brühlmann, Corinne, Ooms, Frédéric, Carrupt, Pierre-Alain, Testa, Bernard, Catto, Marco, Leonetti, Francesco, Altomare, Cosimo, Carotti, Angelo
Published in Journal of medicinal chemistry (13.09.2001)
Published in Journal of medicinal chemistry (13.09.2001)
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Inhibition of Monoamine Oxidases by Functionalized Coumarin Derivatives: Biological Activities, QSARs, and 3D-QSARs
Gnerre, Carmela, Catto, Marco, Leonetti, Francesco, Weber, Peter, Carrupt, Pierre-Alain, Altomare, Cosimo, Carotti, Angelo, Testa, Bernard
Published in Journal of medicinal chemistry (14.12.2000)
Published in Journal of medicinal chemistry (14.12.2000)
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Journal Article
Anti-inflammatory, antimicrobial and antioxidant activities of Diospyros bipindensis (Gürke) extracts and its main constituents
Cesari, I., Hoerlé, M., Simoes-Pires, C., Grisoli, P., Queiroz, E.F., Dacarro, C., Marcourt, L., Moundipa, P.F., Carrupt, P.A., Cuendet, M., Caccialanza, G., Wolfender, J.L., Brusotti, G.
Published in Journal of ethnopharmacology (07.03.2013)
Published in Journal of ethnopharmacology (07.03.2013)
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Journal Article
Antioxidant potential and radical-scavenging effects of flavonoids from the leaves of Psidium cattleianum grown in French Polynesia
Ho, R., Violette, A., Cressend, D., Raharivelomanana, P., Carrupt, P.A., Hostettmann, K.
Published in Natural product research (01.02.2012)
Published in Natural product research (01.02.2012)
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Journal Article
Antifungals and acetylcholinesterase inhibitors from the stem bark of Croton heliotropiifolius
Queiroz, M.M.F., Queiroz, E.F., Zeraik, M.L., Marti, G., Favre-Godal, Q., Simões-Pires, C., Marcourt, L., Carrupt, P.A., Cuendet, M., Paulo, M.Q., Bolzani, V.S., Wolfender, J.L.
Published in Phytochemistry letters (01.12.2014)
Published in Phytochemistry letters (01.12.2014)
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Journal Article
Generalization of Ionic Partition Diagrams to Lipophilic Compounds and to Biphasic Systems with Variable Phase Volume Ratios
Gobry, Véronique, Ulmeanu, Sorina, Reymond, Frédéric, Bouchard, Géraldine, Carrupt, Pierre-Alain, Testa, Bernard, Girault, Hubert H
Published in Journal of the American Chemical Society (31.10.2001)
Published in Journal of the American Chemical Society (31.10.2001)
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Journal Article
Chiral Inversion and Hydrolysis of Thalidomide: Mechanisms and Catalysis by Bases and Serum Albumin, and Chiral Stability of Teratogenic Metabolites
Reist, Marianne, Carrupt, Pierre-Alain, Francotte, Eric, Testa, Bernard
Published in Chemical research in toxicology (01.12.1998)
Published in Chemical research in toxicology (01.12.1998)
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Journal Article
Isoquinoline derivatives as endogenous neurotoxins in the aetiology of Parkinson’s disease
McNaught, Kevin St.P., Carrupt, Pierre-Alain, Altomare, Cosimo, Cellamare, Saverio, Carotti, Angelo, Testa, Bernard, Jenner, Peter, Marsden, C.David
Published in Biochemical pharmacology (15.10.1998)
Published in Biochemical pharmacology (15.10.1998)
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Journal Article
Fast determination of lipophilicity by HPLC
AYOUNI, L, CAZORLA, G, CHAILLOU, D, HERBRETEAU, B, RUDAZ, S, LANTERI, P, CORRUPT, P.-A
Published in Chromatographia (01.09.2005)
Published in Chromatographia (01.09.2005)
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Journal Article
Inhibition of Monoamine Oxidase-B by Condensed Pyridazines and Pyrimidines: Effects of Lipophilicity and Structure−Activity Relationships
Altomare, Cosimo, Cellamare, Saverio, Summo, Luciana, Catto, Marco, Carotti, Angelo, Thull, Ulrike, Carrupt, Pierre-Alain, Testa, Bernard, Stoeckli-Evans, Helen
Published in Journal of medicinal chemistry (24.09.1998)
Published in Journal of medicinal chemistry (24.09.1998)
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Journal Article
Lipophilicity in molecular modeling
Testa, B, Carrupt, P A, Gaillard, P, Billois, F, Weber, P
Published in Pharmaceutical research (01.03.1996)
Published in Pharmaceutical research (01.03.1996)
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Journal Article
Evaluation and prediction of drug permeation
Pagliara, A, Reist, M, Geinoz, S, Carrupt, P A, Testa, B
Published in Journal of pharmacy and pharmacology (01.12.1999)
Published in Journal of pharmacy and pharmacology (01.12.1999)
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Journal Article
Molecular Properties and Pharmacokinetic Behavior of Cetirizine, a Zwitterionic H1-Receptor Antagonist
Pagliara, Alessandra, Testa, Bernard, Carrupt, Pierre-Alain, Jolliet, Pascale, Morin, Christophe, Morin, Didier, Urien, Saïk, Tillement, Jean-Paul, Rihoux, Jean-Pierre
Published in Journal of medicinal chemistry (12.03.1998)
Published in Journal of medicinal chemistry (12.03.1998)
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Journal Article
Inhibition of monoamine oxidase by isoquinoline derivatives: Qualitative and 3D-quantitative structure-activity relationships
Thull, Ulrike, Kneubühler, Silvia, Gaillard, Patrick, Carrupt, Pierre-Alain, Testa, Bernard, Altomare, Cosimo, Carotti, Angelo, Jenner, Peter, St. P. McNaught, Kevin
Published in Biochemical pharmacology (07.09.1995)
Published in Biochemical pharmacology (07.09.1995)
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