Probing the aurone scaffold against Plasmodium falciparum: Design, synthesis and antimalarial activity
Carrasco, Marta P., Newton, Ana S., Gonçalves, Lídia, Góis, Ana, Machado, Marta, Gut, Jiri, Nogueira, Fátima, Hänscheid, Thomas, Guedes, Rita C., dos Santos, Daniel J.V.A., Rosenthal, Philip J., Moreira, Rui
Published in European journal of medicinal chemistry (10.06.2014)
Published in European journal of medicinal chemistry (10.06.2014)
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Journal Article
Editorial: Inspired by Nature: Towards Novel Anti-Infective Agents
Ferreira, Ricardo J, Reis, Mariana A, Silva, Daniel, Scapin, Elisandra, Dewanjee, Saikat, Carrasco, Marta P
Published in Frontiers in pharmacology (21.01.2022)
Published in Frontiers in pharmacology (21.01.2022)
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Journal Article
Novel folate-hydroxamate based antimetabolites: synthesis and biological evaluation
Carrasco, Marta P, Enyedy, Eva A, Krupenko, Natalia I, Krupenko, Sergey A, Nuti, Elisa, Tuccinardi, Tiziano, Santamaria, Salvatore, Rossello, Armando, Martinelli, Adriano, Santos, M Amélia
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (01.07.2011)
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (01.07.2011)
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Journal Article
Azaaurones as Potent Antimycobacterial Agents Active against MDR‐ and XDR‐TB
Campaniço, André, Carrasco, Marta P., Njoroge, Mathew, Seldon, Ronnett, Chibale, Kelly, Perdigão, João, Portugal, Isabel, Warner, Digby F., Moreira, Rui, Lopes, Francisca
Published in ChemMedChem (20.08.2019)
Published in ChemMedChem (20.08.2019)
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Journal Article
Design and development of photoswitchable DFG-Out RET kinase inhibitors
Xu, Yongjin, Gao, Chunxia, Andreasson, Måns, Håversen, Liliana, Carrasco, Marta P., Fleming, Cassandra, Lundbäck, Thomas, Andréasson, Joakim, Grøtli, Morten
Published in European journal of medicinal chemistry (15.04.2022)
Published in European journal of medicinal chemistry (15.04.2022)
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Journal Article
Polybenzimidazole for Active Pharmaceutical Ingredient Purification: The Mometasone Furoate Case Study
Ferreira, Flávio Alves, Esteves, Teresa, Carrasco, Marta P, Bandarra, João, Afonso, Carlos A. M, Ferreira, Frederico Castelo
Published in Industrial & engineering chemistry research (19.06.2019)
Published in Industrial & engineering chemistry research (19.06.2019)
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Combination of hyaluronic acid and PLGA particles as hybrid systems for viscosupplementation in osteoarthritis
Mota, Ana Henriques, Direito, Rosa, Carrasco, Marta P., Rijo, Patrícia, Ascensão, Lia, Viana, Ana Silveira, Rocha, João, Eduardo-Figueira, Maria, Rodrigues, Maria João, Custódio, Luísa, Kuplennik, Nataliya, Sosnik, Alejandro, Almeida, António José, Gaspar, Maria Manuela, Reis, Catarina Pinto
Published in International journal of pharmaceutics (25.03.2019)
Published in International journal of pharmaceutics (25.03.2019)
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Journal Article
Plasmodium dihydrofolate reductase is a second enzyme target for the antimalarial action of triclosan
Bilsland, Elizabeth, van Vliet, Liisa, Williams, Kevin, Feltham, Jack, Carrasco, Marta P, Fotoran, Wesley L, Cubillos, Eliana F G, Wunderlich, Gerhard, Grøtli, Morten, Hollfelder, Florian, Jackson, Victoria, King, Ross D, Oliver, Stephen G
Published in Scientific reports (18.01.2018)
Published in Scientific reports (18.01.2018)
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Journal Article
Probing the Azaaurone Scaffold against the Hepatic and Erythrocytic Stages of Malaria Parasites
Carrasco, Marta P., Machado, Marta, Gonçalves, Lídia, Sharma, Moni, Gut, Jiri, Lukens, Amanda K., Wirth, Dyann F., André, Vânia, Duarte, Maria Teresa, Guedes, Rita C., dos Santos, Daniel J. V. A., Rosenthal, Philip J., Mazitschek, Ralph, Prudêncio, Miguel, Moreira, Rui
Published in ChemMedChem (06.10.2016)
Published in ChemMedChem (06.10.2016)
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Flavones as isosteres of 4(1H)-quinolones: Discovery of ligand efficient and dual stage antimalarial lead compounds
Rodrigues, Tiago, Ressurreição, Ana S., da Cruz, Filipa P., Albuquerque, Inês S., Gut, Jiri, Carrasco, Marta P., Gonçalves, Daniel, Guedes, Rita C., dos Santos, Daniel J.V.A., Mota, Maria M., Rosenthal, Philip J., Moreira, Rui, Prudêncio, Miguel, Lopes, Francisca
Published in European journal of medicinal chemistry (01.11.2013)
Published in European journal of medicinal chemistry (01.11.2013)
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Exploring the Molecular Basis of Qo bc1 Complex Inhibitors Activity to Find Novel Antimalarials Hits
Carrasco, Marta P., Gut, Jiri, Rodrigues, Tiago, Ribeiro, Maria H. L., Lopes, Francisca, Rosenthal, Philip J., Moreira, Rui, dos Santos, Daniel J. V. A.
Published in Molecular informatics (01.07.2013)
Published in Molecular informatics (01.07.2013)
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Journal Article
Exploring the Molecular Basis of Q sub(o) bc sub(1) Complex Inhibitors Activity to Find Novel Antimalarials Hits
Carrasco, Marta P, Gut, Jiri, Rodrigues, Tiago, Ribeiro, Maria HL, Lopes, Francisca, Rosenthal, Philip J, Moreira, Rui, dosSantos, Daniel JVA
Published in Molecular informatics (01.07.2013)
Published in Molecular informatics (01.07.2013)
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