Bioisosteres of Indomethacin as Inhibitors of Aldo-Keto Reductase 1C3
Lolli, Marco L, Carnovale, Irene M, Pippione, Agnese C, Wahlgren, Weixiao Y, Bonanni, Davide, Marini, Elisabetta, Zonari, Daniele, Gallicchio, Margherita, Boscaro, Valentina, Goyal, Parveen, Friemann, Rosmarie, Rolando, Barbara, Bagnati, Renzo, Adinolfi, Salvatore, Oliaro-Bosso, Simonetta, Boschi, Donatella
Published in ACS medicinal chemistry letters (11.04.2019)
Published in ACS medicinal chemistry letters (11.04.2019)
Get full text
Journal Article
Hydroxytriazole derivatives as potent and selective aldo-keto reductase 1C3 (AKR1C3) inhibitors discovered by bioisosteric scaffold hopping approach
Pippione, Agnese C., Giraudo, Alessandro, Bonanni, Davide, Carnovale, Irene M., Marini, Elisabetta, Cena, Clara, Costale, Annalisa, Zonari, Daniele, Pors, Klaus, Sadiq, Maria, Boschi, Donatella, Oliaro-Bosso, Simonetta, Lolli, Marco L.
Published in European journal of medicinal chemistry (20.10.2017)
Published in European journal of medicinal chemistry (20.10.2017)
Get full text
Journal Article