Abstract 1138: The protein disulfide isomerase inhibitor XCE853 inhibits in vitro , ex-vivo and in vivo growth of human tumors
Prevost, Gregoire Pierre, Chauchereau, Anne, Ladam, Patrick, Seigneuric, Renaud, Carniato, Denis, Pitty, Marc-Henry, Foster, Paul
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Get full text
Journal Article
Abstract 4140: Identification of a selective MKLP2/KIF20A inhibitor with high in-vivo antitumor activity
Collette, Yves, Miserey-Lenkei, Stephanie, Guillou, Catherine, Carniato, Denis, Pau, Bernard, Goud, Bruno, Vey, Norbert, Bougeret, Cecile E.
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Get full text
Journal Article
Abstract 3760: XCE853 is a promising protein disulfide isomerase (PDI) inhibitor exhibiting a strong inhibitory activity in preclinical tumor models
Prevost, Gregoire P., Garrido, Marine, Serova, Maria, Briand, Jean François, Gutmann, Mathieu, Ladam, Patrick, Carniato, Denis, Tijeras-Raballand, Annemilai, De Grammont, Armand, Chauchereau, Anne, Pitty, Marc-Henry, Foster, Paul
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Get full text
Journal Article
Abstract 4466: New biomarkers to optimize preclinical development of the PDI inhibitor XCE853
Prevost, Gregoire Pierre, Garrido, Marine, Xu, Shili, Lefebvre, Celine, Chauchereau, Anne, Carniato, Denis, Briand, Jean François, Gutmann, Mathieu, Serova, Maria, Tijeras-Raballand, Annemilai, De Grammont, Armand, Raymond, Eric, Gespach, Christian, Sabbah, Michèle, Neamati, Nouri, Pitty, Marc-Henry, Foster, Paul
Published in Cancer research (Chicago, Ill.) (01.08.2015)
Published in Cancer research (Chicago, Ill.) (01.08.2015)
Get full text
Journal Article
Abstract 1812: XCE853: A novel PDI inhibitor that inhibits proliferation of human tumor cells in vitro , ex-vivo and in vivo
Prevost, Gregoire P., Xu, Shili, Garrido, Marine, Serova, Maria, Vewer, Olivier D., Gespach, Christian, Briand, Jean-François, Tijeras-Raballand, Annemilaï, Gutmann, Mathieu, Hendrix, An, Sabbah, Michele, Chachereau, Anne, Gramont, Armand de, Neamati, Nouri, Carniato, Denis, Pitty, Marc-Henry, Foster, Paul
Published in Cancer research (Chicago, Ill.) (01.10.2014)
Published in Cancer research (Chicago, Ill.) (01.10.2014)
Get full text
Journal Article
Structure-based design of 7-azaindole-pyrrolidine amides as inhibitors of 11β-hydroxysteroid dehydrogenase type I
Valeur, Eric, Christmann-Franck, Serge, Lepifre, Franck, Carniato, Denis, Cravo, Daniel, Charon, Christine, Bozec, Sophie, Musil, Djordje, Hillertz, Per, Doare, Liliane, Schmidlin, Fabien, Lecomte, Marc, Schultz, Melanie, Roche, Didier
Published in Bioorganic & medicinal chemistry letters (15.09.2012)
Published in Bioorganic & medicinal chemistry letters (15.09.2012)
Get full text
Journal Article
Discovery and structure-guided drug design of inhibitors of 11β-hydroxysteroid-dehydrogenase type I based on a spiro-carboxamide scaffold
Lepifre, Franck, Christmann-Franck, Serge, Roche, Didier, Leriche, Caroline, Carniato, Denis, Charon, Christine, Bozec, Sophie, Doare, Liliane, Schmidlin, Fabien, Lecomte, Marc, Valeur, Eric
Published in Bioorganic & medicinal chemistry letters (01.07.2009)
Published in Bioorganic & medicinal chemistry letters (01.07.2009)
Get full text
Journal Article
신규한 바이사이클릭 리포란티펩티드, 제조 및 항균제로서의 용도
LE BELLER DOMINIQUE, LESQUAME GUILLAUME, CARNIATO DENIS, QUERNIN MARIE HELENE, ASZODI JOSEF
Year of Publication 07.03.2018
Get full text
Year of Publication 07.03.2018
Patent
NEW DERIVATIVES OF INDOLE FOR THE TREATMENT OF CANCER, VIRAL INFECTION AND LUNG DISEASES
BOUGERET CECILE, ROULEAU JULIEN, CARNIATO DENIS, GUILLOU CATHERINE, RIVOLLIER JULIE
Year of Publication 12.08.2015
Get full text
Year of Publication 12.08.2015
Patent
Discovery and structure–activity relationships of pentanedioic acid diamides as potent inhibitors of 11β-hydroxysteroid dehydrogenase type I
Roche, Didier, Carniato, Denis, Leriche, Caroline, Lepifre, Franck, Christmann-Franck, Serge, Graedler, Ulrich, Charon, Christine, Bozec, Sophie, Doare, Liliane, Schmidlin, Fabien, Lecomte, Marc, Valeur, Eric
Published in Bioorganic & medicinal chemistry letters (15.05.2009)
Published in Bioorganic & medicinal chemistry letters (15.05.2009)
Get full text
Journal Article
Structure-based design of 7-azaindole-pyrrolidine amides as inhibitors of 11[beta]-hydroxysteroid dehydrogenase type I
Valeur, Eric, Christmann-Franck, Serge, Lepifre, Franck, Carniato, Denis, Cravo, Daniel, Charon, Christine, Bozec, Sophie, Musil, Djordje, Hillertz, Per, Doare, Liliane, Schmidlin, Fabien, Lecomte, Marc, Schultz, Melanie, Roche, Didier
Published in Bioorganic & medicinal chemistry letters (15.09.2012)
Published in Bioorganic & medicinal chemistry letters (15.09.2012)
Get full text
Journal Article
PIPERAZINYL DERIVATIVES FOR THE TREATMENT OF CANCER
JAILLARDON KARINE, GUTMANN MATHIEU, BRIAND JEAN FRANCOIS, BOUGERET CECILE, DEPREZ BENOIT, CARNIATO DENIS, BUSNEL OLIVIER
Year of Publication 07.10.2014
Get full text
Year of Publication 07.10.2014
Patent
NIP THIAZOLE DERIVATIVES AS INHIBITORS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE-1
LERICHE CAROLINE, CARNIATO DENIS, DOARE LILIANE, ROCHE DIDIER, CHARON CHRISTINE
Year of Publication 13.01.2011
Get full text
Year of Publication 13.01.2011
Patent