Pharmacological Characterization of the Nociceptin/Orphanin FQ Receptor Antagonist SB-612111 [(â)-cis-1-Methyl-7-[[4-(2,6-dichlorophenyl)piperidin-1-yl]methyl]-6,7,8,9-tetrahydro-5H-benzocyclohepten-5-ol]: In Vitro Studies
Barbara Spagnolo, Giacomo CarrÃ, Martina Fantin, Carmela Fischetti, Chris Hebbes, John McDonald, Timothy A. Barnes, Anna Rizzi, Claudio Trapella, Giulia Fanton, Michele Morari, Dave G. Lambert, Domenico Regoli, Girolamo CalÃ
Published in The Journal of pharmacology and experimental therapeutics (01.06.2007)
Published in The Journal of pharmacology and experimental therapeutics (01.06.2007)
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Pharmacological profile of NOP receptors coupled with calcium signaling via the chimeric protein Gαqi5
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Published in Naunyn-Schmiedeberg's archives of pharmacology (01.06.2009)
Published in Naunyn-Schmiedeberg's archives of pharmacology (01.06.2009)
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Rizzi, Anna, Spagnolo, Barbara, Wainford, Richard D., Fischetti, Carmela, Guerrini, Remo, Marzola, Giuliano, Baldisserotto, Anna, Salvadori, Severo, Regoli, Domenico, Kapusta, Daniel R., Calo, Girolamo
Published in Peptides (New York, N.Y. : 1980) (01.06.2007)
Published in Peptides (New York, N.Y. : 1980) (01.06.2007)
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Synthesis and biological activity of nociceptin/orphanin FQ analogues substituted in position 7 or 11 with Cα,α-dialkylated amino acids
Arduin, Marika, Spagnolo, Barbara, Calò, Girolamo, Guerrini, Remo, Carrà, Giacomo, Fischetti, Carmela, Trapella, Claudio, Marzola, Erika, McDonald, John, Lambert, David G., Regoli, Domenico, Salvadori, Severo
Published in Bioorganic & medicinal chemistry (01.07.2007)
Published in Bioorganic & medicinal chemistry (01.07.2007)
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Pharmacological characterization of the nociceptin/orphanin FQ receptor non peptide antagonist Compound 24
Fischetti, Carmela, Camarda, Valeria, Rizzi, Anna, Pelà, Michela, Trapella, Claudio, Guerrini, Remo, McDonald, John, Lambert, David G., Salvadori, Severo, Regoli, Domenico, Calo', Girolamo
Published in European journal of pharmacology (01.07.2009)
Published in European journal of pharmacology (01.07.2009)
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Structure–activity studies on the nociceptin/orphanin FQ receptor antagonist 1-benzyl- N-{3-[spiroisobenzofuran-1(3 H),4′-piperidin-1-yl]propyl} pyrrolidine-2-carboxamide
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Published in Bioorganic & medicinal chemistry (15.07.2009)
Published in Bioorganic & medicinal chemistry (15.07.2009)
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Comparative biochemical and pharmacological characterization of a novel, NOP receptor selective hexapeptide, Ac-RYYRIR-ol
Bojnik, Engin, Babos, Fruzsina, Fischetti, Carmela, Magyar, Anna, Camarda, Valeria, Borsodi, Anna, Bajusz, Sándor, Calo’, Girolamo, Benyhe, Sándor
Published in Brain research bulletin (16.03.2010)
Published in Brain research bulletin (16.03.2010)
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Further studies on the pharmacological features of the nociceptin/orphanin FQ receptor ligand ZP120
Fischetti, Carmela, Rizzi, Anna, Gavioli, Elaine C., Marzola, Giuliano, Trapella, Claudio, Guerrini, Remo, Petersen, Jorgen S., Calo, Girolamo
Published in Peptides (New York, N.Y. : 1980) (01.02.2009)
Published in Peptides (New York, N.Y. : 1980) (01.02.2009)
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Journal Article
Pharmacological Characterization of the Nociceptin/Orphanin FQ Receptor Antagonist SB-612111 [(–)- cis -1-Methyl-7-[[4-(2,6-dichlorophenyl)piperidin-1-yl]methyl]-6,7,8,9-tetrahydro-5 H -benzocyclohepten-5-ol]: In Vitro Studies
Spagnolo, Barbara, Carrà, Giacomo, Fantin, Martina, Fischetti, Carmela, Hebbes, Chris, McDonald, John, Barnes, Timothy A., Rizzi, Anna, Trapella, Claudio, Fanton, Giulia, Morari, Michele, Lambert, Dave G., Regoli, Domenico, Calò, Girolamo
Published in The Journal of pharmacology and experimental therapeutics (01.06.2007)
Published in The Journal of pharmacology and experimental therapeutics (01.06.2007)
Get full text
Journal Article
Synthesis and biological activity of nociceptin/orphanin FQ analogues substituted in position 7 or 11 with Calpha,alpha-dialkylated amino acids
Arduin, Marika, Spagnolo, Barbara, Calò, Girolamo, Guerrini, Remo, Carrà, Giacomo, Fischetti, Carmela, Trapella, Claudio, Marzola, Erika, McDonald, John, Lambert, David G, Regoli, Domenico, Salvadori, Severo
Published in Bioorganic & medicinal chemistry (01.07.2007)
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Published in Bioorganic & medicinal chemistry (01.07.2007)
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