Structural basis of the effect of activating mutations on the EGF receptor
Galdadas, Ioannis, Carlino, Luca, Ward, Richard A, Hughes, Samantha J, Haider, Shozeb, Gervasio, Francesco Luigi
Published in eLife (28.07.2021)
Published in eLife (28.07.2021)
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Journal Article
The role of histone demethylases in cancer therapy
Hoffmann, Inga, Roatsch, Martin, Schmitt, Martin L., Carlino, Luca, Pippel, Martin, Sippl, Wolfgang, Jung, Manfred
Published in Molecular oncology (01.12.2012)
Published in Molecular oncology (01.12.2012)
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Journal Article
Synthesis, biological activity and molecular modeling studies on 1H-benzimidazole derivatives as acetylcholinesterase inhibitors
Alpan, Ayşe Selcen, Parlar, Sülünay, Carlino, Luca, Tarikogullari, Ayse Hande, Alptüzün, Vildan, Güneş, Hasan Semih
Published in Bioorganic & medicinal chemistry (01.09.2013)
Published in Bioorganic & medicinal chemistry (01.09.2013)
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Journal Article
Improving Localization by Testing Mobility
Carlino, Luca, Bandiera, Francesco, Coluccia, Angelo, Ricci, Giuseppe
Published in IEEE transactions on signal processing (01.07.2019)
Published in IEEE transactions on signal processing (01.07.2019)
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Journal Article
Merging Nucleophilic Phosphine Catalysis and Photocatalysis for the Rapid Assembly of 2-Oxabicyclo-[2.1.1]hexane Scaffolds from Feedstock Allyl Alcohols
Whalley, David Michael, Carlino, Luca, Putra, Okky Dwichandra, Anderson, Niall, Coote, Susannah Clare, Lorthioir, Olivier Eric
Published in Chemical science (Cambridge) (2024)
Published in Chemical science (Cambridge) (2024)
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Journal Article
Access to 2‑Oxabicyclo[2.1.1]hexanes and their use in Scaffold Hopping
Lorthioir, Olivier, Anderson, Niall, Boyd, Scott, Carlino, Luca, Davey, Paul, Hodds, William, Howard, Megan, Lindhagen, Marika, Proctor, Katie, Putra, Okky Dwichandra, Smith, Theo, Turner, Oliver, Woodhouse, Alfie, Woodward, Millie
Published in Organic letters (01.11.2024)
Published in Organic letters (01.11.2024)
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Journal Article
Access to 2-Oxabicyclo2.1.1hexanes and their use in Scaffold Hopping
Lorthioir, Olivier, Anderson, Niall, Boyd, Scott, Carlino, Luca, Davey, Paul, Hodds, William, Howard, Megan, Lindhagen, Marika, Proctor, Katie, Putra, Okky Dwichandra, Smith, Theo, Turner, Oliver, Woodhouse, Alfie, Woodward, Millie
Published in Organic letters (01.11.2024)
Published in Organic letters (01.11.2024)
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Journal Article
Identification of Novel Potent NSD2-PWWP1 Ligands Using Structure-Based Design and Computational Approaches
Carlino, Luca, Astles, Peter C., Ackroyd, Bryony, Ahmed, Afshan, Chan, Christina, Collie, Gavin W., Dale, Ian L., O’Donovan, Daniel H., Fawcett, Caroline, di Fruscia, Paolo, Gohlke, Andrea, Guo, Xiaoxiao, Hao-Ru Hsu, Jessie, Kaplan, Bethany, Milbradt, Alexander G., Northall, Sarah, Petrović, Dušan, Rivers, Emma L., Underwood, Elizabeth, Webb, Alice
Published in Journal of medicinal chemistry (13.06.2024)
Published in Journal of medicinal chemistry (13.06.2024)
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Journal Article
Nonpeptidic Propargylamines as Inhibitors of Lysine Specific Demethylase 1 (LSD1) with Cellular Activity
Schmitt, Martin L, Hauser, Alexander-Thomas, Carlino, Luca, Pippel, Martin, Schulz-Fincke, Johannes, Metzger, Eric, Willmann, Dominica, Yiu, Teresa, Barton, Michelle, Schüle, Roland, Sippl, Wolfgang, Jung, Manfred
Published in Journal of medicinal chemistry (26.09.2013)
Published in Journal of medicinal chemistry (26.09.2013)
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Journal Article
Identification and Structure-Activity Relationship Studies of Small-Molecule Inhibitors of the Methyllysine Reader Protein Spindlin1
Robaa, Dina, Wagner, Tobias, Luise, Chiara, Carlino, Luca, McMillan, Joel, Flaig, Ralf, Schüle, Roland, Jung, Manfred, Sippl, Wolfgang
Published in ChemMedChem (19.10.2016)
Published in ChemMedChem (19.10.2016)
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Journal Article
Computer- and structure-based lead design for epigenetic targets
Heinke, Ralf, Carlino, Luca, Kannan, Srinivasaraghavan, Jung, Manfred, Sippl, Wolfgang
Published in Bioorganic & medicinal chemistry (15.06.2011)
Published in Bioorganic & medicinal chemistry (15.06.2011)
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Journal Article
Structure–Activity Relationships of Hexahydrocyclopenta[c]quinoline Derivatives as Allosteric Inhibitors of CDK2 and EGFR
Carlino, Luca, Christodoulou, Michael S., Restelli, Valentina, Caporuscio, Fabiana, Foschi, Francesca, Semrau, Marta S., Costanzi, Elisa, Tinivella, Annachiara, Pinzi, Luca, Lo Presti, Leonardo, Battistutta, Roberto, Storici, Paola, Broggini, Massimo, Passarella, Daniele, Rastelli, Giulio
Published in ChemMedChem (20.12.2018)
Published in ChemMedChem (20.12.2018)
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Journal Article
Probing an Allosteric Pocket of CDK2 with Small Molecules
Christodoulou, Michael S., Caporuscio, Fabiana, Restelli, Valentina, Carlino, Luca, Cannazza, Giuseppe, Costanzi, Elisa, Citti, Cinzia, Lo Presti, Leonardo, Pisani, Pasquale, Battistutta, Roberto, Broggini, Massimo, Passarella, Daniele, Rastelli, Giulio
Published in ChemMedChem (05.01.2017)
Published in ChemMedChem (05.01.2017)
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Journal Article
Inhibition of bromodomain-mediated protein–protein interactions as a novel therapeutic strategy
Furdas, Silviya D., Carlino, Luca, Sippl, Wolfgang, Jung, Manfred
Published in MedChemComm (01.02.2012)
Published in MedChemComm (01.02.2012)
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Journal Article
Abstract B81: Analogues of the chromenone namoline as inhibitors of lysine specific demethylase 1 (LSD1)
Schulz-Fincke, Johannes, Schmitt, Martin L., Carlino, Luca, Haydn, Tinka, Willmann, Dominica, Metzger, Eric, Fulda, Simone, Schüle, Roland, Sippl, Wolfgang, Jung, Manfred
Published in Molecular cancer therapeutics (01.12.2015)
Published in Molecular cancer therapeutics (01.12.2015)
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Journal Article
1H-benzimidazole derivatives as butyrylcholinesterase inhibitors: synthesis and molecular modeling studies
Coban, Gunes, Carlino, Luca, Tarikogullari, Ayse Hande, Parlar, Sülünay, Sarıkaya, Görkem, Alptüzün, Vildan, Alpan, Ayşe Selcen, Güneş, Hasan Semih, Erciyas, Erçin
Published in Medicinal chemistry research (01.09.2016)
Published in Medicinal chemistry research (01.09.2016)
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Journal Article