Smoothened transduces Hedgehog signals via activity-dependent sequestration of PKA catalytic subunits
Arveseth, Corvin D, Happ, John T, Hedeen, Danielle S, Zhu, Ju-Fen, Capener, Jacob L, Klatt Shaw, Dana, Deshpande, Ishan, Liang, Jiahao, Xu, Jiewei, Stubben, Sara L, Nelson, Isaac B, Walker, Madison F, Kawakami, Kouki, Inoue, Asuka, Krogan, Nevan J, Grunwald, David J, Hüttenhain, Ruth, Manglik, Aashish, Myers, Benjamin R
Published in PLoS biology (22.04.2021)
Published in PLoS biology (22.04.2021)
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Journal Article
A PKA inhibitor motif within SMOOTHENED controls Hedgehog signal transduction
Happ, John T, Arveseth, Corvin D, Bruystens, Jessica, Bertinetti, Daniela, Nelson, Isaac B, Olivieri, Cristina, Zhang, Jingyi, Hedeen, Danielle S, Zhu, Ju-Fen, Capener, Jacob L, Bröckel, Jan W, Vu, Lily, King, C C, Ruiz-Perez, Victor L, Ge, Xuecai, Veglia, Gianluigi, Herberg, Friedrich W, Taylor, Susan S, Myers, Benjamin R
Published in Nature structural & molecular biology (01.10.2022)
Published in Nature structural & molecular biology (01.10.2022)
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Journal Article
Development of SYK NanoBRET cellular target engagement assays for gain–of–function variants
Capener, Jacob L., Vasta, James D., Katis, Vittorio L., Michaud, Ani, Beck, Michael T., Daglish, Sabrina C. D., Cohen-Kedar, Sarit, Shaham Barda, Efrat, Howell, Stefanie, Dotan, Iris, Robers, Matthew B., Axtman, Alison D., Bashore, Frances M.
Published in Frontiers in Chemical Biology (29.07.2024)
Published in Frontiers in Chemical Biology (29.07.2024)
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Journal Article
Development of SYK NanoBRET Cellular Target Engagement Assays for Gain-of-Function Variants
Capener, Jacob L, Vasta, James D, Katis, Vittorio L, Michaud, Ani, Beck, Michael T, Daglish, Sabrina C D, Cohen-Kedar, Sarit, Barda, Efrat Shaham, Howell, Stefanie, Dotan, Iris, Robers, Matthew B, Axtman, Alison D, Bashore, Frances M
Published in bioRxiv (13.06.2024)
Published in bioRxiv (13.06.2024)
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More than an Amide Bioisostere: Discovery of 1,2,4-Triazole-containing Pyrazolo1,5-apyrimidine Host CSNK2 Inhibitors for Combatting β-Coronavirus Replication
Ong, Han Wee, Yang, Xuan, Smith, Jeffery L, Dickmander, Rebekah J, Brown, Jason W, Havener, Tammy M, Taft-Benz, Sharon, Howell, Stefanie, Sanders, Marcia K, Capener, Jacob L, Couñago, Rafael M, Chang, Edcon, Krämer, Andreas, Moorman, Nathaniel J, Heise, Mark, Axtman, Alison D, Drewry, David H, Willson, Timothy M
Published in Journal of medicinal chemistry (25.07.2024)
Published in Journal of medicinal chemistry (25.07.2024)
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Journal Article
More than an Amide Bioisostere: Discovery of 1,2,4-Triazole-containing Pyrazolo[1,5‑a]pyrimidine Host CSNK2 Inhibitors for Combatting β‑Coronavirus Replication
Ong, Han Wee, Yang, Xuan, Smith, Jeffery L., Dickmander, Rebekah J., Brown, Jason W., Havener, Tammy M., Taft-Benz, Sharon, Howell, Stefanie, Sanders, Marcia K., Capener, Jacob L., Couñago, Rafael M., Chang, Edcon, Krämer, Andreas, Moorman, Nathaniel J., Heise, Mark, Axtman, Alison D., Drewry, David H., Willson, Timothy M.
Published in Journal of medicinal chemistry (25.07.2024)
Published in Journal of medicinal chemistry (25.07.2024)
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Journal Article
Smoothened Transduces Hedgehog Signals via Activity-Dependent Sequestration of PKA Catalytic Subunits
Arveseth, Corvin D, Happ, John T, Hedeen, Danielle S, Ju-Fen Zhu, Capener, Jacob L, Dana Klatt Shaw, Deshpande, Ishan, Liang, Jiahao, Xu, Jiewei, Stubben, Sara L, Nelson, Isaac B, Walker, Madison F, Krogan, Nevan J, Grunwald, David J, Hüttenhain, Ruth, Manglik, Aashish, Myers, Benjamin R
Published in bioRxiv (02.07.2020)
Published in bioRxiv (02.07.2020)
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