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Published in Nature biotechnology (01.07.2012)
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Published in Science (American Association for the Advancement of Science) (13.03.2015)
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Published in Science translational medicine (20.04.2016)
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A small molecule CFTR potentiator restores ATP‐dependent channel gating to the cystic fibrosis mutant G551D‐CFTR
Liu, Jia, Berg, Allison P., Wang, Yiting, Jantarajit, Walailak, Sutcliffe, Katy J., Stevens, Edward B., Cao, Lishuang, Pregel, Marko J., Sheppard, David N.
Published in British journal of pharmacology (01.04.2022)
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GI‐530159, a novel, selective, mechanosensitive two‐pore‐domain potassium (K2P) channel opener, reduces rat dorsal root ganglion neuron excitability
Loucif, Alexandre J C, Saintot, Pierre‐Philippe, Liu, Jia, Antonio, Brett M, Zellmer, Shannon G, Yoger, Katrina, Veale, Emma L, Wilbrey, Anna, Omoto, Kiyoyuki, Cao, Lishuang, Gutteridge, Alex, Castle, Neil A, Stevens, Edward B, Mathie, Alistair
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Published in British journal of pharmacology (01.06.2018)
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Owen, Robert M, Blakemore, David, Cao, Lishuang, Flanagan, Neil, Fish, Rebecca, Gibson, Karl R, Gurrell, Rachel, Huh, Chan Woo, Kammonen, Juha, Mortimer-Cassen, Elisabeth, Nickolls, Sarah A, Omoto, Kiyoyuki, Owen, Dafydd, Pike, Andy, Pryde, David C, Reynolds, David S, Roeloffs, Rosemarie, Rose, Colin, Stead, Clara, Takeuchi, Mifune, Warmus, Joseph S, Watson, Christine
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Published in Journal of medicinal chemistry (27.06.2019)
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Characterizing Human Stem Cell–derived Sensory Neurons at the Single-cell Level Reveals Their Ion Channel Expression and Utility in Pain Research
Young, Gareth T, Gutteridge, Alex, Fox, Heather DE, Wilbrey, Anna L, Cao, Lishuang, Cho, Lily T, Brown, Adam R, Benn, Caroline L, Kammonen, Laura R, Friedman, Julia H, Bictash, Magda, Whiting, Paul, Bilsland, James G, Stevens, Edward B
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Published in Molecular therapy (01.08.2014)
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Pharmacology in translation: the preclinical and early clinical profile of the novel α2/3 functionally selective GABAA receptor positive allosteric modulator PF‐06372865
Nickolls, Sarah A, Gurrell, Rachel, Amerongen, Guido, Kammonen, Juha, Cao, Lishuang, Brown, Adam R, Stead, Clara, Mead, Andy, Watson, Christine, Hsu, Cathleen, Owen, Robert M, Pike, Andy, Fish, Rebecca L, Chen, Laigao, Qiu, Ruolun, Morris, Evan D, Feng, Gang, Whitlock, Mark, Gorman, Donal, Gerven, Joop, Reynolds, David S, Dua, Pinky, Butt, Richard P
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Published in British journal of pharmacology (01.02.2018)
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Design and Identification of a Novel, Functionally Subtype Selective GABA(A) Positive Allosteric Modulator (PF-06372865)
Owen, Robert M., Blakemore, David, Cao, Lishuan, Flanagan, Neil, Fish, Rebecca, Gibson, Karl R., Gurrell, Rachel, Huh, Chan Woo, Kammonen, Juha, Mortimer-Cassen, Elisabeth, Nickolls, Sarah A., Omoto, Kiyoyuki, Owen, Dafydd, Pike, Andy, Pryde, David C., Reynolds, David S., Roeloffs, Rosemarie, Rose, Colin, Stead, Clara, Takeuchi, Mifune, Warmus, Joseph S., Watson, Christine
Published in Journal of medicinal chemistry (27.06.2019)
Published in Journal of medicinal chemistry (27.06.2019)
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Influence of the N terminus on the biophysical properties and pharmacology of TREK1 potassium channels
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Published in Molecular pharmacology (01.05.2014)
Published in Molecular pharmacology (01.05.2014)
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Publisher Correction: Molecular and functional variation in iPSC-derived sensory neurons
Schwartzentruber, Jeremy, Foskolou, Stefanie, Kilpinen, Helena, Rodrigues, Julia, Alasoo, Kaur, Knights, Andrew J, Patel, Minal, Goncalves, Angela, Ferreira, Rita, Benn, Caroline Louise, Wilbrey, Anna, Bictash, Magda, Impey, Emma, Cao, Lishuang, Lainez, Sergio, Loucif, Alexandre Julien, Whiting, Paul John, Gutteridge, Alex, Gaffney, Daniel J
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Published in Nature genetics (01.07.2019)
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Investigation of the structure activity relationship of flufenamic acid derivatives at the human TRESK channel K2P18.1
Monteillier, Aymeric, Loucif, Alexandre, Omoto, Kiyoyuki, Stevens, Edward B., Lainez, Sergio, Saintot, Pierre-Philippe, Cao, Lishuang, Pryde, David C.
Published in Bioorganic & medicinal chemistry letters (15.10.2016)
Published in Bioorganic & medicinal chemistry letters (15.10.2016)
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Corrigendum to “Investigation of the structure activity relationship of flufenamic acid derivatives at the human TRESK channel K2P18.1” [Bioorg. Med. Chem. Lett. 26 (2016) 4919–4924]
Monteillier, Aymeric, Loucif, Alexandre, Omoto, Kiyoyuki, Stevens, Edward B., Lainez, Sergio, Saintot, Pierre-Philippe, Cao, Lishuang, Pryde, David C.
Published in Bioorganic & medicinal chemistry letters (01.05.2017)
Published in Bioorganic & medicinal chemistry letters (01.05.2017)
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Journal Article
Investigation of the structure activity relationship of flufenamic acid derivatives at the human TRESK channel K 2P 18.1
Monteillier, Aymeric, Loucif, Alexandre, Omoto, Kiyoyuki, Stevens, Edward B, Lainez, Sergio, Saintot, Pierre-Philippe, Cao, Lishuang, Pryde, David C
Published in Bioorganic & medicinal chemistry letters (15.10.2016)
Published in Bioorganic & medicinal chemistry letters (15.10.2016)
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