Natural-product-inspired design and synthesis of two series of compounds active against Trypanosoma cruzi: Insights into structure–activity relationship, toxicity, and mechanism of action
da Rosa, Rafael, Dambrós, Bibiana Paula, Höehr de Moraes, Milene, Grand, Lucie, Jacolot, Maïwenn, Popowycz, Florence, Steindel, Mario, Schenkel, Eloir Paulo, Campos Bernardes, Lílian Sibelle
Published in Bioorganic chemistry (01.02.2022)
Published in Bioorganic chemistry (01.02.2022)
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Synthesis and cytotoxic activity evaluation of dihydrocucurbitacin B and cucurbitacin B derivatives
Lang, Karen Luise, Silva, Izabella Thaís, Zimmermann, Lara Almida, Machado, Vanessa Rocha, Teixeira, Marina Rodrigues, Lapuh, María Ivana, Galetti, Mariana Alejandra, Palermo, Jorge Alejandro, Cabrera, Gabriela Myriam, Bernardes, Lílian Sibelle Campos, Simões, Cláudia Maria Oliveira, Schenkel, Eloir Paulo, Caro, Miguel Soriano Balparda, Durán, Fernando Javier
Published in Bioorganic & medicinal chemistry (01.05.2012)
Published in Bioorganic & medicinal chemistry (01.05.2012)
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Journal Article
Chemical Modification Produces Species-Specific Changes in Cucurbitacin Antifeedant Effect
Lang, Karen Luise, Deagosto, Emilio, Zimmermann, Lara Almida, Machado, Vanessa Rocha, Campos Bernardes, Lílian Sibelle, Schenkel, Eloir Paulo, Duran, Fernando Javier, Palermo, Jorge, Rossini, Carmen
Published in Journal of agricultural and food chemistry (12.06.2013)
Published in Journal of agricultural and food chemistry (12.06.2013)
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Journal Article
Design and synthesis of a new series of 3,5-disubstituted isoxazoles active against Trypanosoma cruzi and Leishmania amazonensis
da Rosa, Rafael, de Moraes, Milene Höehr, Zimmermann, Lara Almida, Schenkel, Eloir Paulo, Steindel, Mario, Bernardes, Lílian Sibelle Campos
Published in European journal of medicinal chemistry (10.03.2017)
Published in European journal of medicinal chemistry (10.03.2017)
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Journal Article
Synthesis and trypanocidal activity of 1,4-bis-(3,4,5-trimethoxy-phenyl)-1,4-butanediol and 1,4-bis-(3,4-dimethoxyphenyl)-1,4-butanediol
Bernardes, Lilian Sibelle Campos, Kato, Massuo Jorge, Albuquerque, Sérgio, Carvalho, Ivone
Published in Bioorganic & medicinal chemistry (01.11.2006)
Published in Bioorganic & medicinal chemistry (01.11.2006)
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Journal Article
Synthesis and biological evaluation of isoxazolyl-sulfonamides: A non-cytotoxic scaffold active against Trypanosoma cruzi, Leishmania amazonensis and Herpes Simplex Virus
da Rosa, Rafael, Zimmermann, Lara Almida, de Moraes, Milene Höehr, Schneider, Naira Fernanda Zanchett, Schappo, Alice Duarte, Simões, Claudia Maria de Oliveira, Steindel, Mario, Schenkel, Eloir Paulo, Bernardes, Lílian Sibelle Campos
Published in Bioorganic & medicinal chemistry letters (01.11.2018)
Published in Bioorganic & medicinal chemistry letters (01.11.2018)
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Novel aryl β-aminocarbonyl derivatives as inhibitors of Trypanosoma cruzi trypanothione reductase: binding mode revised by docking and GRIND2-based 3D-QSAR procedures
de Paula da Silva, Carlos Henrique Tomich, Bernardes, Lílian Sibelle Campos, da Silva, Vinícius Barreto, Zani, Carlos Leomar, Carvalho, Ivone
Published in Journal of biomolecular structure & dynamics (01.01.2012)
Published in Journal of biomolecular structure & dynamics (01.01.2012)
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Synthesis and 2D-QSAR studies of neolignan-based diaryltetrahydrofuran and -furan analogues with remarkable activity against Trypanosoma cruzi and assessment of the trypanothione reductase activity
Hartmann, Ana Paula, de Carvalho, Marcelo Rodrigues, Campos Bernardes, Lilian Sibelle, de Moraes, Milena Hoehr, de Melo, Eduardo Borges, Lopes, Carla Duque, Steindel, Mario, da Silva, Joao Santana, Carvalho, Ivone
Published in European journal of medicinal chemistry (10.11.2017)
Published in European journal of medicinal chemistry (10.11.2017)
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Journal Article
Synthesis and 2D-QSAR studies of neolignan-based diaryl-tetrahydrofuran and -furan analogues with remarkable activity against Trypanosoma cruzi and assessment of the trypanothione reductase activity
Hartmann, Ana Paula, de Carvalho, Marcelo Rodrigues, Bernardes, Lilian Sibelle Campos, Moraes, Milena Hoehr de, de Melo, Eduardo Borges, Lopes, Carla Duque, Steindel, Mario, da Silva, João Santana, Carvalho, Ivone
Published in European journal of medicinal chemistry (10.11.2017)
Published in European journal of medicinal chemistry (10.11.2017)
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Journal Article
Qualitative and quantitative chemical characterization of spray‐dried extracts and the development of an innovative oral solid formulation from Lippia alba
Almeida, Maiara Prates, Silva, Lorena Alves de Oliveira, Zimmermann, Lara Almida, Bernardes, Lilian Sibelle Campos, da Silva, Marcelo Aparecido, da Silva, Geraldo Alves, Amaral, Juliano Geraldo, Gomes, Angélica Ferraz, Leite, Mateus Freire
Published in Separation science plus (01.04.2023)
Published in Separation science plus (01.04.2023)
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Journal Article
Combinatorial Chemistry Underpinning Drug Discovery and Development
Bernardes, Lilian Sibelle Campos, Silva, Carlos H. T. P., Taft, Carlton A., Carvalho, Ivone
Published in ChemInform (06.11.2007)
Published in ChemInform (06.11.2007)
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