Structural Determinants for Small-Molecule Activation of Skeletal Muscle AMPK α2β2γ1 by the Glucose Importagog SC4
Ngoei, Kevin R.W., Langendorf, Christopher G., Ling, Naomi X.Y., Hoque, Ashfaqul, Varghese, Swapna, Camerino, Michelle A., Walker, Scott R., Bozikis, Ylva E., Dite, Toby A., Ovens, Ashley J., Smiles, William J., Jacobs, Roxane, Huang, He, Parker, Michael W., Scott, John W., Rider, Mark H., Foitzik, Richard C., Kemp, Bruce E., Baell, Jonathan B., Oakhill, Jonathan S.
Published in Cell chemical biology (21.06.2018)
Published in Cell chemical biology (21.06.2018)
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The structure-activity relationships of L3MBTL3 inhibitors: flexibility of the dimer interface
Camerino, Michelle A, Zhong, Nan, Dong, Aiping, Dickson, Bradley M, James, Lindsey I, Baughman, Brandi M, Norris, Jacqueline L, Kireev, Dmitri B, Janzen, William P, Arrowsmith, Cheryl H, Frye, Stephen V
Published in MedChemComm (01.11.2013)
Published in MedChemComm (01.11.2013)
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Solid Phase Synthesis and Circular Dichroism Analysis of (i → i + 4) Cyclic Lactam Analogues of Kisspeptin
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Published in International journal of peptide research and therapeutics (01.12.2008)
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(S)-(−)-Fluorenylethylchloroformate (FLEC); preparation using asymmetric transfer hydrogenation and application to the analysis and resolution of amines
Amin, Mohammad A., Camerino, Michelle A., Mountford, Simon J., Ma, Xiao, Manallack, David T., Chalmers, David K., Wills, Martin, Thompson, Philip E.
Published in Tetrahedron (25.10.2019)
Published in Tetrahedron (25.10.2019)
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Discovery of a highly potent, selective, orally bioavailable inhibitor of KAT6A/B histone acetyltransferases with efficacy against KAT6A-high ER+ breast cancer
Sharma, Shikhar, Chung, Chi-Yeh, Uryu, Sean, Petrovic, Jelena, Cao, Joan, Rickard, Amanda, Nady, Nataliya, Greasley, Samantha, Johnson, Eric, Brodsky, Oleg, Khan, Showkhin, Wang, Hui, Wang, Zhenxiong, Zhang, Yong, Tsaparikos, Konstantinos, Chen, Lei, Mazurek, Anthony, Lapek, John, Kung, Pei-Pei, Sutton, Scott, Richardson, Paul F., Greenwald, Eric C., Yamazaki, Shinji, Jones, Rhys, Maegley, Karen A., Bingham, Patrick, Lam, Hieu, Stupple, Alexandra E., Kamal, Aileen, Chueh, Anderly, Cuzzupe, Anthony, Morrow, Benjamin J., Ren, Bin, Carrasco-Pozo, Catalina, Tan, Chin Wee, Bhuva, Dharmesh D., Allan, Elizabeth, Surgenor, Elliot, Vaillant, François, Pehlivanoglu, Havva, Falk, Hendrik, Whittle, James R., Newman, Janet, Cursons, Joseph, Doherty, Judy P., White, Karen L., MacPherson, Laura, Devlin, Mark, Dennis, Matthew L., Hattarki, Meghan K., De Silva, Melanie, Camerino, Michelle A., Butler, Miriam S., Dolezal, Olan, Pilling, Patricia, Foitzik, Richard, Stupple, Paul A., Lagiakos, H. Rachel, Walker, Scott R., Hediyeh-Zadeh, Soroor, Nuttall, Stewart, Spall, Sukhdeep K., Charman, Susan A., Connor, Theresa, Peat, Thomas S., Avery, Vicky M., Bozikis, Ylva E., Yang, Yuqing, Zhang, Ming, Monahan, Brendon J., Voss, Anne K., Thomas, Tim, Street, Ian P., Dawson, Sarah-Jane, Dawson, Mark A., Lindeman, Geoffrey J., Davis, Melissa J., Visvader, Jane E., Paul, Thomas A.
Published in Cell chemical biology (19.10.2023)
Published in Cell chemical biology (19.10.2023)
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Abstract 1130: First-in-class KAT6A/KAT6B inhibitor CTx-648 (PF-9363) demonstrates potent anti-tumor activity in ER+ breast cancer with KAT6A dysregulation
Sharma, Shikhar, Chung, Jay, Uryu, Sean, Rickard, Amanda, Nady, Natalie, Khan, Showkhin, Wang, Zhenxiong, Zhang, Yong, Zhang, Haikuo, Kung, Pei-Pei, Greenwald, Eric, Maegley, Karen, Bingham, Patrick, Lam, Hieu, Bozikis, Ylva E., Falk, Hendrik, Allan, Elizabeth, Avery, Vicky M., Butler, Miriam S., Camerino, Michelle A., Carrasco-Pozo, Catalina, Charman, Susan A., Davis, Melissa J., Dawson, Mark A., Sarah-Jane, Dawson, de Silva, Melanie, Dennis, Matthew L., Dolezal, Olan, Lagiakos, Rachel, Lindeman, Geoffrey J., MacPherson, Laura, Nuttall, Stewart, Peat, Thomas S., Ren, Bin, Stupple, Alexandra E., Surgenor, Elliot, Tan, Chin Wee, Thomas, Tim, Visvader, Jane E., Voss, Anne K., Vaillant, Francois, White, Karen L., Whittle, James, Yang, Yuqing, Hediyeh-Zadeh, Soroor, Stupple, Paul A., Street, Ian P., Monahan, Brendon J., Paul, Thomas
Published in Cancer research (Chicago, Ill.) (01.07.2021)
Published in Cancer research (Chicago, Ill.) (01.07.2021)
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(+)-Fluorenylethylchloroformate (FLEC) - improved synthesis for application in chiral analysis and peptidomimetic synthesisElectronic supplementary information (ESI) available: Full experimental details relating to all syntheses are available as supplementary data. See DOI: 10.1039/c3ob40218e
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Abstract 5371: PRMT5 inhibitors as novel treatment for cancers
Falk, Hendrik, Foitzik, Richard C., Allan, Elizabeth, deSilva, Melanie, Yang, Hong, Bozikis, Ylva E., Nikac, Marica, Walker, Scott R., Camerino, Michelle A., Morrow, Ben J., Stupple, Alexandra E., Lagiakos, Rachel, Pinson, Jo-Anne, Lessene, Romina, Kersten, Wilhelmus JA, Ganame, Danny G., Holmes, Ian P., Lunniss, Gill E., Chung, Matthew, Hermans, Stefan J., Parker, Michael W., Thistlethwaite, Alison, White, Karen, Charman, Susan A., Monahan, Brendon J., Pilling, Patricia, Grusovin, Julian, Peat, Thomas S., Sonderegger, Stefan, Toulmin, Emma, Jane, Stephen M., Curtis, David J., Stupple, Paul A., Street, Ian P.
Published in Cancer research (Chicago, Ill.) (01.08.2015)
Published in Cancer research (Chicago, Ill.) (01.08.2015)
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The structure-activity relationships of L3MBTL3 inhibitors: flexibility of the dimer interfaceElectronic supplementary information (ESI) available: Experimental procedures including spectra for all final compounds, crystallographic methods, in vitro assay conditions and representative ITC binding curves. See DOI: 10.1039/c3md00197k
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COMPOUND
MORROW BENJAMIN J, BOZIKIS YLVA E B, LAGIAKOS HELEN R, WALKER SCOTT R, FOITZIK RICHARD C, CAMERINO MICHELLE A, HEMLEY CATHERINE F, STUPPLE PAUL A
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Compounds
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SUBSTITUTED CONDENSED THIOPHENES AS MODULATORS OF STING
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Compounds
HEMLEY, CATHERINE FAE, STUPPLE, PAUL ANTHONY, LAGIAKOS, HELEN RACHEL, MORROW, BENJAMIN JOSEPH, CAMERINO, MICHELLE ANG, WALKER, SCOTT RAYMOND, FOITZIK, RICHARD CHARLES, BOZIKIS, YLVA ELISABET BERGMAN
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화합물
HEMLEY CATHERINE FAE, MORROW BENJAMIN JOSEPH, LAGIAKOS HELEN RACHEL, WALKER SCOTT RAYMOND, STUPPLE PAUL ANTHONY, FOITZIK RICHARD CHARLES, BOZIKIS YLVA ELISABET BERGMAN, CAMERINO MICHELLE ANG
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