Allosteric Effects of Sodium Ion Binding on Activation of the M3 Muscarinic G-Protein-Coupled Receptor
Miao, Yinglong, Caliman, Alisha D., McCammon, J. Andrew
Published in Biophysical journal (07.04.2015)
Published in Biophysical journal (07.04.2015)
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Journal Article
Mapping the allosteric sites of the A 2A adenosine receptor
Caliman, Alisha D, Miao, Yinglong, McCammon, James A
Published in Chemical biology & drug design (01.01.2018)
Published in Chemical biology & drug design (01.01.2018)
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Journal Article
Activation of atypical protein kinase C by sphingosine 1-phosphate revealed by an aPKC-specific activity reporter
Kajimoto, Taketoshi, Caliman, Alisha D, Tobias, Irene S, Okada, Taro, Pilo, Caila A, Van, An-Angela N, Andrew McCammon, J, Nakamura, Shun-Ichi, Newton, Alexandra C
Published in Science signaling (01.01.2019)
Published in Science signaling (01.01.2019)
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Journal Article
Allosteric inhibition of PPM1D serine/threonine phosphatase via an altered conformational state
Miller, Peter G, Sathappa, Murugappan, Moroco, Jamie A, Jiang, Wei, Qian, Yue, Iqbal, Sumaiya, Guo, Qi, Giacomelli, Andrew O, Shaw, Subrata, Vernier, Camille, Bajrami, Besnik, Yang, Xiaoping, Raffier, Cerise, Sperling, Adam S, Gibson, Christopher J, Kahn, Josephine, Jin, Cyrus, Ranaghan, Matthew, Caliman, Alisha, Brousseau, Merissa, Fischer, Eric S, Lintner, Robert, Piccioni, Federica, Campbell, Arthur J, Root, David E, Garvie, Colin W, Ebert, Benjamin L
Published in Nature communications (30.06.2022)
Published in Nature communications (30.06.2022)
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Journal Article
Investigation of the conformational dynamics of the apo A2A adenosine receptor
Caliman, Alisha D., Swift, Sara E., Wang, Yi, Miao, Yinglong, McCammon, J. Andrew
Published in Protein science (01.06.2015)
Published in Protein science (01.06.2015)
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Journal Article
Mapping the allosteric sites of the A2A adenosine receptor
Caliman, Alisha D., Miao, Yinglong, McCammon, James A.
Published in Chemical biology & drug design (01.01.2018)
Published in Chemical biology & drug design (01.01.2018)
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Journal Article
S1P-aPKCシグナリングが制御するアポトーシス抵抗性の新たな分子メカニズム
梶本, 武利, キャリマン, アリシャ, トバイアス, アイリーン, 岡田, 太郎, パイロ, ケイラ, ヴァン, アンジェラ, マキャモン, アンドリュー, 中村, 俊一, ニュートン, アレキサンドラ
Published in 日本薬理学会年会要旨集 (2023)
Published in 日本薬理学会年会要旨集 (2023)
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Journal Article
Investigation of the conformational dynamics of the apo A 2A adenosine receptor
Caliman, Alisha D., Swift, Sara E., Wang, Yi, Miao, Yinglong, McCammon, J. Andrew
Published in Protein science (01.06.2015)
Published in Protein science (01.06.2015)
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Journal Article
Abstract 3588: Discovery of potent and selective CSNK1A1 inhibitors for solid tumor therapy
Corsello, Steven M., Zhang, Huajia, Rupaimoole, Rajesha, Schulze, Volker K., Lemos, Clara, Handing, Kasia B., Orsi, Douglas L., Shekhar, Mrinal, Sack, Ulrike, Christian, Sven, Bone, Wilhelm, Humeidi, Ranad, Colgan, William, Hoyt, Stephanie, Cherniack, Andrew, Schroder, Jens, Kaulfuss, Stefan, Brzezinka, Krzysztof, von Ahsen, Oliver, Mengel, Anne, Hillig, Roman C., Suelzle, Detlev, Mortier, Jeremie, Harrington, Caitlin, Nagari, Rohith, Wierzbinska, Justyna, Chiang, Derek, Beckmann, Georg, Olive, Meagan, Udeshi, Namrata, Apffel, Annie, Carr, Steven, Lienau, Philip, Lechner, Christian, Boemer, Ulf, Caliman, Alisha, McKinney, David, Wagner, Florence, Mumberg, Dominik, Bauser, Marcus, Haegebarth, Andrea, Eis, Knut, Eheim, Ashley, Golub, Todd R.
Published in Cancer research (Chicago, Ill.) (15.06.2022)
Published in Cancer research (Chicago, Ill.) (15.06.2022)
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Journal Article
A novel molecular mechanism of apoptosis resistance regulated by S1P-aPKC signaling
Kajimoto, Taketoshi, Caliman, Alisha D., Tobias, Irene S., Okada, Taro, Pilo, Caila A., Van, An-Angela, McCammon, J. Andrew, Nakamura, Shun-ichi, Newton, Alexandra C.
Published in Proceedings for Annual Meeting of The Japanese Pharmacological Society (2023)
Published in Proceedings for Annual Meeting of The Japanese Pharmacological Society (2023)
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Journal Article
HETEROAROMATIC COMPOUNDS
VERANO, Alyssa Leigh, ZHENG, Xiaolan, CALIMAN, Alisha Danielle, JOHANNES, Jeffrey Wallace, LIANG, Yufan, MLYNARSKI, Scott Nathan, ZIEGLER, Robert Evans, READ, Jonathan Anthony
Year of Publication 11.04.2024
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Year of Publication 11.04.2024
Patent
BICYCLIC HETEROAROMATIC COMPOUNDS AND THEIR APPLICATION IN THE TREATMENT OF CANCER
VERANO, Alyssa Leigh, ZHENG, Xiaolan, CALIMAN, Alisha Danielle, JOHANNES, Jeffrey Wallace, LIANG, Yufan, MLYNARSKI, Scott Nathan, ZIEGLER, Robert Evans, READ, Jonathan Anthony
Year of Publication 02.11.2023
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Year of Publication 02.11.2023
Patent
SUBSTITUTED PYRROLO-PYRIDINONE DERIVATIVES AND THERAPEUTIC USES THEREOF
Schulze, Volker, Caliman, Alisha, Bömer, Ulf, Lechner, Christian, Mengel, Anne, Rauh, Ulrike, Hillig, Roman, Faria Alvares De Lemos, Adelaide Clara, Mortier, Jeremie Xavier G, Madec, Amael, Sülzle, Detlev, Corsello, Steven, Handing, Katarzyna, Kaulfuss, Stefan
Year of Publication 16.11.2023
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Year of Publication 16.11.2023
Patent
3-AMINO-2-[2-(ACYLAMINO)PYRIDIN-4-YL]-1,5,6,7-TETRAHYDRO-4H-PYRROLO[3,2-C]PYRIDIN-4-ONE AS CSNK1 INHIBITORS
SÜLZLE, Detlev, MORTIER, Jérémie, FARIA ALVARES DE LEMOS, Adelaide, Clara, BÖMER, Ulf, LECHNER, Christian, CORSELLO, Steven, CALIMAN, Alisha, KAULFUSS, Stefan, CHRIST, Clara, SCHULZE, Volker, MENGEL, Anne, HANDING, Katarzyna, RAUH, Ulrike, Schröder, Jens, BONE, Wilhelm, HILLIG, Roman
Year of Publication 02.08.2023
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Year of Publication 02.08.2023
Patent
SUBSTITUTED PYRROLO-PYRIDINONE DERIVATIVES AND THERAPEUTIC USES THEREOF
SÜLZLE, Detlev, FARIA ALVARES DE LEMOS, Adelaide, Clara, MADEC, Amael, BÖMER, Ulf, LECHNER, Christian, CORSELLO, Steven, CALIMAN, Alisha, KAULFUSS, Stefan, SCHULZE, Volker, MENGEL, Anne, RAUH, Ulrike, HANDING, Katarzyna, HILLIG, Roman, MORTIER, Jeremie, Xavier, G
Year of Publication 07.06.2023
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Year of Publication 07.06.2023
Patent
3-AMINO-2-[2-(ACYLAMINO)PYRIDIN-4-YL]-1,5,6,7-TETRAHYDRO-4H-PYRROLO[3,2-C]PYRIDIN-4-ONE AS CSNK1 INHIBITORS
Schulze, Volker, Schroeder, Jens, Caliman, Alisha, Lechner, Christian, Sulzle, Detlev, Mengel, Anne, Christ, Clara, Rauh, Ulrike, Hillig, Roman, Faria Alvares De Lemos, Adelaide Clara, Bomer, Ulf, Handing, Kasia, Bone, Wilhelm, Corsello, Steven, Kaulfuss, Stefan, Mortier, Jérémie
Year of Publication 16.02.2023
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Year of Publication 16.02.2023
Patent