Synthesis of 2-(Pyridin-3-yl)-1-azabicyclo[3.2.2]nonane, 2-(Pyridin-3-yl)-1-azabicyclo[2.2.2]octane, and 2-(Pyridin-3-yl)-1-azabicyclo[3.2.1]octane, a Class of Potent Nicotinic Acetylcholine Receptor–Ligands
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Published in Journal of organic chemistry (02.05.2008)
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Published in Bioorganic & medicinal chemistry letters (15.01.2012)
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Discovery of novel α7 nicotinic acetylcholine receptor ligands via pharmacophoric and docking studies of benzylidene anabaseine analogs
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Published in Bioorganic & medicinal chemistry letters (15.01.2012)
Published in Bioorganic & medicinal chemistry letters (15.01.2012)
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Docking studies of benzylidene anabaseine interactions with α7 nicotinic acetylcholine receptor (nAChR) and acetylcholine binding proteins (AChBPs): Application to the design of related α7 selective ligands
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First Total Synthesis of (±)-3-Hydroxy-11-norcytisine: Structure Confirmation and Biological Characterization
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Bohme, Georg Andrees, Letchworth, Sharon R., Piot-Grosjean, Odile, Gatto, Gregory J., Obinu, Marie-Carmen, Caldwell, William S., Laville, Michel, Brunel, Pascale, Pellerin, Rachel, Leconte, Jean-Pierre, Genevois-Borella, Arielle, Dubedat, Pierre, Mazadier, Martine, Pradier, Laurent, Bencherif, Merouane, Benavides, Jesus
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Kinetic Isotope Effects on Substrate Association: Reactions of Phosphoenolpyruvate with Phosphoenolpyruvate Carboxylase and Pyruvate Kinase
Gawlita, Ewa, Caldwell, William S, O'Leary, Marion H, Paneth, Piotr, Anderson, Vernon E
Published in Biochemistry (Easton) (28.02.1995)
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TC‐1734: An Orally Active Neuronal Nicotinic Acetylcholine Receptor Modulator with Antidepressant, Neuroprotective and Long‐Lasting Cognitive Effects
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Docking studies of benzylidene anabaseine interactions with alpha 7 nicotinic acetylcholine receptor (nAChR) and acetylcholine binding proteins (AChBPs): Application to the design of related alpha 7 selective ligands
Kombo, David C., Mazurov, Anatoly, Tallapragada, Kartik, Hammond, Philip S., Chewning, Joseph, Hauser, Terry A., Vasquez-Valdivieso, Montserrat, Yohannes, Daniel, Talley, Todd T., Taylor, Palmer, Caldwell, William S.
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The nitrosation of nicotine: a kinetic study
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Published in Chemical research in toxicology (01.09.1991)
Published in Chemical research in toxicology (01.09.1991)
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In vitro and in vivo characterization of TC‐1827, a novel brain α 4 β 2 nicotinic receptor agonist with pro‐cognitive activity
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Published in Drug development research (01.05.2004)
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In vitro and in vivo characterization of TC-1827, a novel brain [alpha] sub(4)[beta] sub(2) nicotinic receptor agonist with pro-cognitive activity
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Correlation between Hydrophobicity of Short-Chain Aliphatic Alcohols and Their Ability to Alter Plasma Membrane Integrity
MCKARNS, SUSAN C., HANSCH, CORWIN, CALDWELL, WILLIAM S., MORGAN, WALTER T., MOORE, SARAH K., DOOLITTLE, DAVID J.
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Published in Toxicological sciences (1997)
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Compounds capable of activating cholinergic receptors
MEROUANE BENCHERIF, WILLIAM S. CALDWELL, PATRICK LIPPIELLO, JARED M. WAGNER
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COMPOUNDS CAPABLE OF ACTIVATING CHOLINERGIC RECEPTORS
CALDWELL, WILLIAM S, CROOKS, PETER A, PARK, HAEIL, BENCHERIF, MEROUANE, BHATTI, BALWINDER S, HADIMANI, SRISHAILKUMAR, DULL, GARY M, LIPPIELLO, PATRICK M, WAGNER, JARED M
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Modern Instrumental Methods for Studying Mechanisms of Toxicology
Published in Principles and Methods of Toxicology
(2008)
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