Search Results - "Caignard, Daniel H." :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Synthesis and Structure–Affinity Relationships of Selective High-Affinity 5‑HT4 Receptor Antagonists: Application to the Design of New Potential Single Photon Emission Computed Tomography Tracers

Synthesis and Structure–Affinity Relationships of Selective High-Affinity 5‑HT4 Receptor Antagonists: Application to the Design of New Potential Single Photon Emission Computed Tomography Tracers

by Dubost, Emmanuelle, Dumas, Noé, Fossey, Christine, Magnelli, Rosa, Butt-Gueulle, Sabrina, Ballandonne, Céline, Caignard, Daniel H, Dulin, Fabienne, Sopkova de-Oliveira Santos, Jana, Millet, Philippe, Charnay, Yves, Rault, Sylvain, Cailly, Thomas, Fabis, Frederic
Published in Journal of medicinal chemistry (26.11.2012)

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Journal Article

Design and synthesis of benzofuranic derivatives as new ligands at the melatonin-binding site MT3

Design and synthesis of benzofuranic derivatives as new ligands at the melatonin-binding site MT3

by ETTAOUSSI, Mohamed, PERES, Basile, YOUS, Saïd, KLUPSCH, Frederique, DELAGRANGE, Philippe, BOUTIN, Jean-A, RENARD, Pierre, CAIGNARD, Daniel-H, CHAVATTE, Philippe, BERTHELOT, Pascal, LESIEUR, Daniel
Published in Bioorganic & medicinal chemistry (01.05.2008)

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Journal Article

Quinazoline and phthalazine derivatives as novel melatonin receptor ligands analogues of agomelatine

Quinazoline and phthalazine derivatives as novel melatonin receptor ligands analogues of agomelatine

by Bolteau, Raphaël, Descamps, Florian, Ettaoussi, Mohamed, Caignard, Daniel H., Delagrange, Philippe, Melnyk, Patricia, Yous, Saïd
Published in European journal of medicinal chemistry (01.03.2020)

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Journal Article

Syntheses and Antitumor Targeting G1 Phase of the Cell Cycle of Benzoyldihydroisoquinolines and Related 1-Substituted Isoquinolines

Syntheses and Antitumor Targeting G1 Phase of the Cell Cycle of Benzoyldihydroisoquinolines and Related 1-Substituted Isoquinolines

by Bermejo, Almudena, Andreu, Inmaculada, Suvire, Fernando, Léonce, Stephane, Caignard, Daniel H, Renard, Pierre, Pierré, Alain, Enriz, Ricardo D, Cortes, Diego, Cabedo, Nuria
Published in Journal of medicinal chemistry (07.11.2002)

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Journal Article

Substituted tetrahydroisoquinolines: synthesis, characterization, antitumor activity and other biological properties

Substituted tetrahydroisoquinolines: synthesis, characterization, antitumor activity and other biological properties

by Capilla, A. Sergi, Soucek, Richard, Grau, Laura, Romero, Manel, Rubio-Martínez, Jaime, Caignard, Daniel H., Pujol, Maria Dolors
Published in European journal of medicinal chemistry (10.02.2018)

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Journal Article

Polycerasoidol, a Natural Prenylated Benzopyran with a Dual PPARα/PPARγ Agonist Activity and Anti-inflammatory Effect

Polycerasoidol, a Natural Prenylated Benzopyran with a Dual PPARα/PPARγ Agonist Activity and Anti-inflammatory Effect

by Bermejo, Almudena, Collado, Aida, Barrachina, Isabel, Marqués, Patrice, El Aouad, Noureddine, Franck, Xavier, Garibotto, Francisco, Dacquet, Catherine, Caignard, Daniel H, Suvire, Fernando D, Enriz, Ricardo D, Piqueras, Laura, Figadère, Bruno, Sanz, María-Jesús, Cabedo, Nuria, Cortes, Diego
Published in Journal of natural products (Washington, D.C.) (26.07.2019)

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Journal Article

Synthesis of benzopyran derivatives as PPARα and/or PPARγ activators

Synthesis of benzopyran derivatives as PPARα and/or PPARγ activators

by Bermejo, Almudena, Barrachina, Isabel, El Aouad, Noureddine, Franck, Xavier, Chahboune, Nadia, Andreu, Inmaculada, Figadère, Bruno, Vila, Laura, Hennuyer, Nathalie, Staels, Bart, Dacquet, Catherine, Caignard, Daniel H., Sanz, María-Jesús, Cortes, Diego, Cabedo, Nuria
Published in Bioorganic & medicinal chemistry (15.12.2019)

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Journal Article

Novel 2(3H)-Benzothiazolones as Highly Potent and Selective Sigma-1 Receptor Ligands

Novel 2(3H)-Benzothiazolones as Highly Potent and Selective Sigma-1 Receptor Ligands

by Yous, Saïd, Wallez, Valérie, Belloir, Mirabelle, Caignard, Daniel H., McCurdy, Christopher R., Poupaert, Jacques H.
Published in Medicinal chemistry research (01.01.2005)

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Journal Article

Design and synthesis of 1-(2-alkanamidoethyl)-6-methoxy-7-azaindole derivatives as potent melatonin agonists

Design and synthesis of 1-(2-alkanamidoethyl)-6-methoxy-7-azaindole derivatives as potent melatonin agonists

by Jeanty, Matthieu, Suzenet, Franck, Delagrange, Philippe, Nosjean, Olivier, Boutin, Jean A., Caignard, Daniel H., Guillaumet, Gérald
Published in Bioorganic & medicinal chemistry letters (15.04.2011)

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Journal Article

Semisynthesis and Cytotoxicity of Styryl-Lactone Derivatives

Semisynthesis and Cytotoxicity of Styryl-Lactone Derivatives

by Bermejo, Almudena, Léonce, Stéphane, Cabedo, Nuria, Andreu, Inmaculada, Caignard, Daniel H, Atassi, Ghanem, Cortes, Diego
Published in Journal of natural products (Washington, D.C.) (01.08.1999)

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Journal Article

Synthesis and Structure–Affinity Relationships of Selective High-Affinity 5-HT 4 Receptor Antagonists: Application to the Design of New Potential Single Photon Emission Computed Tomography Tracers

Synthesis and Structure–Affinity Relationships of Selective High-Affinity 5-HT 4 Receptor Antagonists: Application to the Design of New Potential Single Photon Emission Computed Tomography Tracers

by Dubost, Emmanuelle, Dumas, Noé, Fossey, Christine, Magnelli, Rosa, Butt-Gueulle, Sabrina, Ballandonne, Céline, Caignard, Daniel H., Dulin, Fabienne, Sopkova de-Oliveira Santos, Jana, Millet, Philippe, Charnay, Yves, Rault, Sylvain, Cailly, Thomas, Fabis, Frederic
Published in Journal of medicinal chemistry (26.11.2012)

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Journal Article

Design and synthesis of 3-phenyltetrahydronaphthalenic derivatives as new selective MT2 melatoninergic ligands. Part II

Design and synthesis of 3-phenyltetrahydronaphthalenic derivatives as new selective MT2 melatoninergic ligands. Part II

by DURIEUX, Sophie, CHANU, Angéline, LESIEUR, Daniel, BERTHELOT, Pascal, YOUS, Saïd, BOCHU, Christophe, AUDINOT, Valérie, COUMAILLEAU, Sophie, BOUTIN, Jean A, DELAGRANGE, Philippe, CAIGNARD, Daniel H, BENNEJEAN, Caroline, RENARD, Pierre
Published in Bioorganic & medicinal chemistry (15.04.2009)

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Journal Article

Antitumor agents. Synthesis and biological evaluation of new compounds related to podophyllotoxin, containing the 2,3-dihydro-1,4-benzodioxin system

Antitumor agents. Synthesis and biological evaluation of new compounds related to podophyllotoxin, containing the 2,3-dihydro-1,4-benzodioxin system

by Capilla, Alfons Sergi, Sánchez, Isabel, Caignard, Daniel H., Renard, Pierre, Pujol, Maria Dolors
Published in European journal of medicinal chemistry (01.04.2001)

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Journal Article

An efficient method for the preparation of antitumoral alpha-keto-imines benzyldihydroisoquinolines by selective benzylic oxidation with C/Pd in acetonitrile

An efficient method for the preparation of antitumoral alpha-keto-imines benzyldihydroisoquinolines by selective benzylic oxidation with C/Pd in acetonitrile

by Andreu, Cabedo, N, Atassi, G, Pierre, A, Caignard, DH, Renard, P, Cortes, D, Bermejo, A
Published in Tetrahedron letters (28.01.2002)

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Journal Article

Synthesis and cytotoxic activity of 2-dialkylaminoethylamino substituted xanthenone and thioxanthenone derivatives

Synthesis and cytotoxic activity of 2-dialkylaminoethylamino substituted xanthenone and thioxanthenone derivatives

by Kostakis, Ioannis, Ghirtis, Konstantinos, Pouli, Nicole, Marakos, Panagiotis, Skaltsounis, Alexios-Leandros, Leonce, Stephane, Caignard, Daniel H, Atassi, Ghanem
Published in Farmaco (Società chimica italiana : 1989) (01.06.2000)

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Journal Article

6-(N-IMIDOALKYL)AMINOALKYLBENZOTHIAZOLIN-2-ONES AS LIGANDS OF THE SEROTONINERGIC 5-HT1A RECEPTORS

6-(N-IMIDOALKYL)AMINOALKYLBENZOTHIAZOLIN-2-ONES AS LIGANDS OF THE SEROTONINERGIC 5-HT1A RECEPTORS

by DIOUF, O, DEPREUX, P, LESIEUR, D, POUPAERT, JH, CAIGNARD, DH
Published in Heterocycles (01.06.1995)

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Journal Article

Design, synthesis and pharmacological evaluation of novel naphthalenic derivatives as selective MT1 melatoninergic ligands

Design, synthesis and pharmacological evaluation of novel naphthalenic derivatives as selective MT1 melatoninergic ligands

by Mésangeau, Christophe, Pérès, Basile, Descamps-François, Carole, Chavatte, Philippe, Audinot, Valérie, Coumailleau, Sophie, Boutin, Jean A., Delagrange, Philippe, Bennejean, Caroline, Renard, Pierre, Caignard, Daniel H., Berthelot, Pascal, Yous, Saïd
Published in Bioorganic & medicinal chemistry (15.05.2010)

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Journal Article

PROCESS FOR PREPARING BENZOXAZOLINONES

PROCESS FOR PREPARING BENZOXAZOLINONES

by LESIEUR, DANIEL, BUSCH, NORBERT, CAIGNARD, DANIEL H, LESPAGNOL, CHARLES
Year of Publication 25.01.1991

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Patent

Design, synthesis and pharmacological evaluation of novel naphthalenic derivatives as selective MT 1 melatoninergic ligands

Design, synthesis and pharmacological evaluation of novel naphthalenic derivatives as selective MT 1 melatoninergic ligands

by Mésangeau, Christophe, Pérès, Basile, Descamps-François, Carole, Chavatte, Philippe, Audinot, Valérie, Coumailleau, Sophie, Boutin, Jean A., Delagrange, Philippe, Bennejean, Caroline, Renard, Pierre, Caignard, Daniel H., Berthelot, Pascal, Yous, Saïd
Published in Bioorganic & medicinal chemistry (2010)

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Journal Article

Design and synthesis of 3-phenyltetrahydronaphthalenic derivatives as new selective MT 2 melatoninergic ligands. Part II

Design and synthesis of 3-phenyltetrahydronaphthalenic derivatives as new selective MT 2 melatoninergic ligands. Part II

by Durieux, Sophie, Chanu, Angéline, Bochu, Christophe, Audinot, Valérie, Coumailleau, Sophie, Boutin, Jean A., Delagrange, Philippe, Caignard, Daniel H., Bennejean, Caroline, Renard, Pierre, Lesieur, Daniel, Berthelot, Pascal, Yous, Saïd
Published in Bioorganic & medicinal chemistry (2009)

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Journal Article