Design and synthesis of novel sulfonamide-containing bradykinin hB(2) receptor antagonists. 2. Synthesis and structure - Activity relationships of alpha,alpha-cycloalkylglycine sulfonamides
Fattori, Daniela, Rossi, Cristina, Fincham, Christopher I., Caciagli, VAlerio, Catrambone, Fernando, D'Andrea, Piero, Felicetti, Patrizia, Gensini, Martina, Marastoni, Elena, Nannicini, Rossano, Paris, Marielle, Terracciano, Rosa, Bressan, Alessandro, Giuliani, Sandro, Maggi, Carlo A., Meini, Stefania, Valenti, Claudio, Quartara, Laura
Published in Journal of medicinal chemistry (08.02.2007)
Published in Journal of medicinal chemistry (08.02.2007)
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Journal Article
Design and Synthesis of Novel Sulfonamide-Containing Bradykinin hB 2 Receptor Antagonists. 2. Synthesis and Structure−Activity Relationships of α,α-Cycloalkylglycine Sulfonamides
Fattori, Daniela, Rossi, Cristina, Fincham, Christopher I., Caciagli, Valerio, Catrambone, Fernando, D'Andrea, Piero, Felicetti, Patrizia, Gensini, Martina, Marastoni, Elena, Nannicini, Rossano, Paris, Marielle, Terracciano, Rosa, Bressan, Alessandro, Giuliani, Sandro, Maggi, Carlo A., Meini, Stefania, Valenti, Claudio, Quartara, Laura
Published in Journal of medicinal chemistry (08.02.2007)
Published in Journal of medicinal chemistry (08.02.2007)
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Novel applications of the potassium chlorate-osmium tetroxide oxidizing system. Synthesis of .alpha.-dicarbonyl derivatives from acetylenic compounds. Synthesis of a 2,3-dihydroxy-1,4-dione from a 2,5-dialkylfuran
Bassignani, Luciano, Brandt, Alberto, Caciagli, Valerio, Re, Luciano
Published in Journal of organic chemistry (01.10.1978)
Published in Journal of organic chemistry (01.10.1978)
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Journal Article
Design and Synthesis of Novel Sulfonamide-Containing Bradykinin hB2 Receptor Antagonists. 2. Synthesis and Structure−Activity Relationships of α,α-Cycloalkylglycine Sulfonamides
Fattori, Daniela, Rossi, Cristina, Fincham, Christopher I, Caciagli, Valerio, Catrambone, Fernando, D'Andrea, Piero, Felicetti, Patrizia, Gensini, Martina, Marastoni, Elena, Nannicini, Rossano, Paris, Marielle, Terracciano, Rosa, Bressan, Alessandro, Giuliani, Sandro, Maggi, Carlo A, Meini, Stefania, Valenti, Claudio, Quartara, Laura
Published in Journal of medicinal chemistry (08.02.2007)
Published in Journal of medicinal chemistry (08.02.2007)
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Journal Article
Large-scale production of peptides using the solid phase continuous flow method. Part 2: preparative synthesis of a 26-mer peptide thrombin inhibitor
Caciagli, Valerio, Cardinali, Franco, Bonelli, Fabio, Lombardi, Paolo
Published in Journal of peptide science (01.08.1998)
Published in Journal of peptide science (01.08.1998)
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Journal Article
Large-scale production of peptides using the solid-phase continuous flow method. Preparative synthesis of the novel tachykinin antagonist MEN 10627
Caciagli, Valerio, Cardinali, Franco, Hänsicke, Andre, Tuchalski, Gisbert, Lombardi, Paolo
Published in Journal of peptide science (01.05.1997)
Published in Journal of peptide science (01.05.1997)
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Journal Article
LINEAR BASIC COMPOUNDS HAVING NK-2 ANTAGONIST ACTIVITY AND FORMULATIONS THEREOF
ALTAMURA, MARIA, NANNICINI, ROSSANO, CACIAGLI, VALERIO, HARMAT, NICHOLAS, SISTO, ALESSANDRO, FEDI, VALENTINA, GUIDI, ANTONIO, PASQUI, FRANCO, MAGGI, CARLO ALBERTO, GIOLITTI, ALESSANDRO, GIANNOTTI, DANILO
Year of Publication 28.05.2013
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Year of Publication 28.05.2013
Patent
compostos básicos lineares apresentando atividade antagonista do nk-2 e formulações contendo os mesmos
Altamura, Maria, Giannotti, Danilo, Guidi, Antonio, Fedi, Valentina, Harmat, Nicholas, Giolitti, Alessandro, Nannicini, Rossano, Maggi, Carlo, Alberto, Pasqui, Franco, Sisto, Alessandro, Caciagli, Valerio
Year of Publication 10.04.2018
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Year of Publication 10.04.2018
Patent
Linear basic compounds having NK-2 antagonist activity and formulations thereof
ALTAMURA, MARIA, CACIAGLI, VALERIO, SISTO, ALESSANDRO, GIOLITTI, ALESSANDRO, FEDI, VALENTINA+
Year of Publication 21.07.2006
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Year of Publication 21.07.2006
Patent
LINEAR BASIC COMPOUNDS HAVING NK-2 ANTAGONIST ACTIVITY AND FORMULATIONS THEREOF
GIOLITTI ALESSANDRO, FEDI VALENTINA, NANNICINI ROSSANO, GUIDI ANTONIO, SISTO ALESSANDRO, PASQUI FRANCO, HARMAT NICHOLAS, CACIAGLI VALERIO, ALTAMURA MARIA, GIANNOTTI DANILO, MAGGI CARLO ALBERTO
Year of Publication 31.08.2011
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Year of Publication 31.08.2011
Patent