Selective and reversible modification of kinase cysteines with chlorofluoroacetamides
Shindo, Naoya, Fuchida, Hirokazu, Sato, Mami, Watari, Kosuke, Shibata, Tomohiro, Kuwata, Keiko, Miura, Chizuru, Okamoto, Kei, Hatsuyama, Yuji, Tokunaga, Keisuke, Sakamoto, Seiichi, Morimoto, Satoshi, Abe, Yoshito, Shiroishi, Mitsunori, Caaveiro, Jose M M, Ueda, Tadashi, Tamura, Tomonori, Matsunaga, Naoya, Nakao, Takaharu, Koyanagi, Satoru, Ohdo, Shigehiro, Yamaguchi, Yasuchika, Hamachi, Itaru, Ono, Mayumi, Ojida, Akio
Published in Nature chemical biology (01.03.2019)
Published in Nature chemical biology (01.03.2019)
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Journal Article
Affinity improvement of a therapeutic antibody by structure-based computational design: generation of electrostatic interactions in the transition state stabilizes the antibody-antigen complex
Kiyoshi, Masato, Caaveiro, Jose M M, Miura, Eri, Nagatoishi, Satoru, Nakakido, Makoto, Soga, Shinji, Shirai, Hiroki, Kawabata, Shigeki, Tsumoto, Kouhei
Published in PloS one (27.01.2014)
Published in PloS one (27.01.2014)
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Journal Article
Structural basis for the recognition of human hemoglobin by the heme-acquisition protein Shr from Streptococcus pyogenes
Senoo, Akinobu, Hoshino, Masato, Shiomi, Toshiki, Nakakido, Makoto, Nagatoishi, Satoru, Kuroda, Daisuke, Nakagawa, Ichiro, Tame, Jeremy R H, Caaveiro, Jose M M, Tsumoto, Kouhei
Published in Scientific reports (05.03.2024)
Published in Scientific reports (05.03.2024)
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Journal Article
Structural analysis of Fc/FcγR complexes: a blueprint for antibody design
Caaveiro, Jose M. M., Kiyoshi, Masato, Tsumoto, Kouhei
Published in Immunological reviews (01.11.2015)
Published in Immunological reviews (01.11.2015)
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Journal Article
Discovery and Optimization of Inhibitors of the Parkinson’s Disease Associated Protein DJ‑1
Tashiro, Shinya, Caaveiro, Jose M. M, Nakakido, Makoto, Tanabe, Aki, Nagatoishi, Satoru, Tamura, Yasushi, Matsuda, Noriyuki, Liu, Dali, Hoang, Quyen Q, Tsumoto, Kouhei
Published in ACS chemical biology (21.09.2018)
Published in ACS chemical biology (21.09.2018)
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Journal Article
Molecular basis for thermal stability and affinity in a VHH: Contribution of the framework region and its influence in the conformation of the CDR3
Kinoshita, Seisho, Nakakido, Makoto, Mori, Chinatsu, Kuroda, Daisuke, Caaveiro, Jose M.M., Tsumoto, Kouhei
Published in Protein science (01.11.2022)
Published in Protein science (01.11.2022)
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Journal Article
Glycosylation of IgG-Fc: a molecular perspective
Kiyoshi, Masato, Tsumoto, Kouhei, Ishii-Watabe, Akiko, Caaveiro, Jose M M
Published in International immunology (01.07.2017)
Published in International immunology (01.07.2017)
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Journal Article
Tyrosine Sulfation Restricts the Conformational Ensemble of a Flexible Peptide, Strengthening the Binding Affinity for an Antibody
Miyanabe, Kazuhiro, Yamashita, Takefumi, Abe, Yoshito, Akiba, Hiroki, Takamatsu, Yuichiro, Nakakido, Makoto, Hamakubo, Takao, Ueda, Tadashi, Caaveiro, Jose M. M, Tsumoto, Kouhei
Published in Biochemistry (Easton) (17.07.2018)
Published in Biochemistry (Easton) (17.07.2018)
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Journal Article
Differential Effect of Membrane Composition on the Pore-Forming Ability of Four Different Sea Anemone Actinoporins
García-Linares, Sara, Rivera-de-Torre, Esperanza, Morante, Koldo, Tsumoto, Kouhei, Caaveiro, Jose M. M, Gavilanes, José G, Slotte, J. Peter, Martínez-del-Pozo, Álvaro
Published in Biochemistry (Easton) (06.12.2016)
Published in Biochemistry (Easton) (06.12.2016)
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Journal Article
Discovery of Chlorofluoroacetamide-Based Covalent Inhibitors for Severe Acute Respiratory Syndrome Coronavirus 2 3CL Protease
Hirose, Yuya, Shindo, Naoya, Mori, Makiko, Onitsuka, Satsuki, Isogai, Hikaru, Hamada, Rui, Hiramoto, Tadanari, Ochi, Jinta, Takahashi, Daisuke, Ueda, Tadashi, Caaveiro, Jose M. M., Yoshida, Yuya, Ohdo, Shigehiro, Matsunaga, Naoya, Toba, Shinsuke, Sasaki, Michihito, Orba, Yasuko, Sawa, Hirofumi, Sato, Akihiko, Kawanishi, Eiji, Ojida, Akio
Published in Journal of medicinal chemistry (27.10.2022)
Published in Journal of medicinal chemistry (27.10.2022)
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Journal Article
Structural and Thermodynamic Basis of Epitope Binding by Neutralizing and Nonneutralizing Forms of the Anti-HIV-1 Antibody 4E10
Rujas, Edurne, Gulzar, Naveed, Morante, Koldo, Tsumoto, Kouhei, Scott, Jamie K, Nieva, José L, Caaveiro, Jose M M
Published in Journal of virology (01.12.2015)
Published in Journal of virology (01.12.2015)
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Journal Article
Ca2+‐induced structural changes and intramolecular interactions in N‐terminal region of diacylglycerol kinase alpha
Takahashi, Daisuke, Yonezawa, Kento, Okizaki, Yuki, Caaveiro, Jose M. M., Ueda, Tadashi, Shimada, Atsushi, Sakane, Fumio, Shimizu, Nobutaka
Published in Protein science (01.07.2022)
Published in Protein science (01.07.2022)
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Journal Article
Heme Binding Mechanism of Structurally Similar Iron-Regulated Surface Determinant Near Transporter Domains of Staphylococcus aureus Exhibiting Different Affinities for Heme
Moriwaki, Yoshitaka, Terada, Tohru, Caaveiro, Jose M. M, Takaoka, Yousuke, Hamachi, Itaru, Tsumoto, Kouhei, Shimizu, Kentaro
Published in Biochemistry (Easton) (10.12.2013)
Published in Biochemistry (Easton) (10.12.2013)
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Journal Article
Testing Geometrical Discrimination within an Enzyme Active Site: Constrained Hydrogen Bonding in the Ketosteroid Isomerase Oxyanion Hole
Sigala, Paul A, Kraut, Daniel A, Caaveiro, Jose M. M, Pybus, Brandon, Ruben, Eliza A, Ringe, Dagmar, Petsko, Gregory A, Herschlag, Daniel
Published in Journal of the American Chemical Society (15.10.2008)
Published in Journal of the American Chemical Society (15.10.2008)
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Journal Article
Molecular recognition of a membrane-anchored HIV-1 pan-neutralizing epitope
Torralba, Johana, de la Arada, Igor, Partida-Hanon, Angélica, Rujas, Edurne, Arribas, Madalen, Insausti, Sara, Valotteau, Claire, Valle, Javier, Andreu, David, Caaveiro, José M M, Jiménez, María Angeles, Apellániz, Beatriz, Redondo-Morata, Lorena, Nieva, José L
Published in Communications biology (18.11.2022)
Published in Communications biology (18.11.2022)
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Journal Article
Molecular Basis of Recognition of Antibacterial Porphyrins by Heme-Transporter IsdH-NEAT3 of Staphylococcus aureus
Moriwaki, Yoshitaka, Caaveiro, Jose M. M, Tanaka, Yoshikazu, Tsutsumi, Hiroshi, Hamachi, Itaru, Tsumoto, Kouhei
Published in Biochemistry (Easton) (30.08.2011)
Published in Biochemistry (Easton) (30.08.2011)
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Journal Article
Unfolding is the driving force for mitochondrial import and degradation of the Parkinson's disease-related protein DJ-1
Queliconi, Bruno Barros, Kojima, Waka, Kimura, Mayumi, Imai, Kenichiro, Udagawa, Chisato, Motono, Chie, Hirokawa, Takatsugu, Tashiro, Shinya, Caaveiro, Jose M M, Tsumoto, Kouhei, Yamano, Koji, Tanaka, Keiji, Matsuda, Noriyuki
Published in Journal of cell science (15.11.2021)
Published in Journal of cell science (15.11.2021)
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Journal Article